Affinity DataIC50: 1.60nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 118nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 206nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 252nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 328nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 332nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Affinity DataIC50: 404nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 407nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 518nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 628nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 633nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 729nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 972nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Istituto Di Scienze E Tecnologie Molecolari (Istm)
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.59E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 3.14E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair