Compile Data Set for Download or QSAR
maximum 50k data
Found 386 with Last Name = 'hadari' and Initial = 'yr'
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179883((4-Isopropylphenyl)-(4-isoquinolin-5-yl-phthalazin...)
Affinity DataIC50:  17nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  45nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179881((4-Chlorophenyl)-(4-isoquinolin-5-yl-phthalazin-1-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262214((2-((1H-indazol-6-yl)methylamino)phenyl)(5-methyl-...)
Affinity DataIC50:  52nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  74nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179890((4-tert-Butylphenyl)-(4-isoquinolin-5-yl-phthalazi...)
Affinity DataIC50:  75nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262274((2-((1H-indazol-6-yl)methylamino)phenyl)(6-methyl-...)
Affinity DataIC50:  76nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173019(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  78nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179889(CHEMBL382818 | N-(4-(chlorodifluoromethoxy)phenyl)...)
Affinity DataIC50:  79nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173031(4-(4-(4-bromophenylamino)phthalazin-1-yl)benzamide...)
Affinity DataIC50:  100nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  100nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179888((3,4-Dichloro-phenyl)-(4-isoquinolin-5-yl-phthalaz...)
Affinity DataIC50:  110nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179891((4-Chloro-3-trifluoromethylphenyl)-(4-isoquinolin-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  120nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50:  130nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173045(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)-N-m...)
Affinity DataIC50:  130nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262057((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50:  140nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192487((7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-...)
Affinity DataIC50:  150nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262105((5-methyl-1H-indol-3-yl)(2-(quinolin-6-ylmethylami...)
Affinity DataIC50:  160nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262057((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262106((1,5-dimethyl-1H-indol-3-yl)(2-(quinolin-6-ylmethy...)
Affinity DataIC50:  180nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173049(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50:  190nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192474(CHEMBL215191 | benzyl-(7,8-dimethoxy-10,11-dihydro...)
Affinity DataIC50:  200nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50:  230nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179893((4-Isoquinolin-5-yl-phthalazin-1-yl)-(2-methyl-1Hi...)
Affinity DataIC50:  230nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262056((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indol-...)
Affinity DataIC50:  240nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262274((2-((1H-indazol-6-yl)methylamino)phenyl)(6-methyl-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262278((2-((1H-indazol-6-yl)methylamino)phenyl)(6-fluoro-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262054((2-((1H-indazol-6-yl)methylamino)phenyl)(1-methyl-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262277((2-((1H-indazol-6-yl)methylamino)phenyl)(5-fluoro-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261960((2-((1H-indazol-6-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  270nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179884((4-Isoquinolin-5-yl-phthalazin-1-yl)-m-tolylamine ...)
Affinity DataIC50:  270nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261961((1H-indazol-3-yl)(2-(quinolin-6-ylmethylamino)phen...)
Affinity DataIC50:  300nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50180448((3-Bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-ox...)
Affinity DataIC50:  300nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262054((2-((1H-indazol-6-yl)methylamino)phenyl)(1-methyl-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192477((3-chloro-2-fluoro-phenyl)-(7,8-dimethoxy-10,11-di...)
Affinity DataIC50:  300nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192498((3-chloro-4-fluoro-benzyl)-(7,8-dimethoxy-10,11-di...)
Affinity DataIC50:  300nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262007((2-((1H-benzo[d]imidazol-5-yl)methylamino)phenyl)(...)
Affinity DataIC50:  310nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50174697(3-fluoro-N-[5-(7-methoxy-10,11-dihydro-5-oxa-2,4,1...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50174698(4-fluoro-N-[5-(7-methoxy-10,11-dihydro-5-oxa-2,4,1...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50180448((3-Bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-ox...)
Affinity DataIC50:  340nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262275((2-((1H-indazol-6-yl)methylamino)phenyl)(7-methyl-...)
Affinity DataIC50:  355nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179894((4-Isoquinolin-5-yl-phthalazin-1-yl)-(4-morpholin-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173022(3-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  400nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179882((2-Fluoro-4-methylphenyl)-(4-isoquinolin-5-ylphtha...)
Affinity DataIC50:  430nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50174686(1-(1-chloro-5-oxa-2,4,11-triaza-dibenzo[a,d]cycloh...)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity against FLT3 kinase in a HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50262157((5-methoxy-1H-indol-3-yl)(2-(quinolin-6-ylmethylam...)
Affinity DataIC50:  450nMAssay Description:Inhibition of KDR (unknown origin) autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50261959((2-((1H-indazol-5-yl)methylamino)phenyl)(1H-indazo...)
Affinity DataIC50:  460nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173034(4-(4-(3-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  470nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50180448((3-Bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-ox...)
Affinity DataIC50:  470nMAssay Description:Inhibition of EGFR autophosphorylation in DiFi cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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