Affinity DataKi: 0.400nMAssay Description:Binding affinity towards Serotonin 5-hydroxytryptamine 1A receptor by displacement of [3H]-(+)-8-OH-DPAT.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]-U-86,170.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.70nMAssay Description:Binding affinity towards Dopamine receptor D3 by displacement of [3H]-(+)-7-OH-DPAT.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]-U-86,170.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity of compound towards 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards Serotonin 5-hydroxytryptamine 1A receptor by displacement of [3H]-(+)-8-OH-DPAT.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]-U-86,170.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards Dopamine receptor D3 by displacement of [3H]-(+)-7-OH-DPAT.More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 6.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]-U-86,170.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]-U-86,170.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]-U-86,170.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]-U-86,170.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 18nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity towards Dopamine receptor D3 by displacement of [3H]-(+)-7-OH-DPAT.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 23nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards Serotonin 5-hydroxytryptamine 1A receptor by displacement of [3H]-(+)-8-OH-DPAT.More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity towards Dopamine receptor D3 by displacement of [3H]-(+)-7-OH-DPAT.More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of North Carolina
Curated by PDSP Ki Database
University of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 54nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair