Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]-sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 1.87nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.96nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.13nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 2.81nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Dissociation constant(Ki) of compound was determined to measure PNMT-inhibitory potencyMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.25nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity against dopamine receptor D2 from rat corpus striatum by using radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.43nMAssay Description:In vitro binding affinity towards dopamine receptor D2 in rat striatal membranes by [3H]sulpiride displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.70nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity against D2 receptor in rat corpus striatum using [3H]-sulpiride as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.11nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 8.54nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2 receptor in rat striatal membranes by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor from rat cortical synaptosomal membrane using radioligand [3H]ketanserin.More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to human 11beta-HSD1 by SPA assayMore data for this Ligand-Target Pair