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Found 204 with Last Name = 'kläss' and Initial = 't'
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50111026(9-[1-(5-Methyl-thiophen-2-yl)-meth-(Z)-ylidene]-7-...)
Affinity DataKi:  4.90nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166332(9-[1-(3'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50366567(ATOMOXETINE)
Affinity DataKi:  5nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50111028(9-[1-(5-Iodo-thiophen-2-yl)-meth-(Z)-ylidene]-7-az...)
Affinity DataKi:  5nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166328(9-[3-(2,6-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  5.30nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166336(9-[1-[2,3']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  5.90nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166339(9-[1-(2'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  6.5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133744(9-[1-(5-Bromo-4-methyl-thiophen-2-yl)-meth-(Z)-yli...)
Affinity DataKi:  6.80nMAssay Description:Ability to inhibit reuptake of serotonin ([3H]5-HT) at serotonin transporter of rat midbrianMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  7.36nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  7.40nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166333(9-[1-(3'-Trifluoromethyl-biphenyl-4-yl)-meth-(Z)-y...)
Affinity DataKi:  8.80nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166334(9-[1-(3'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  9.40nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133753(9-[1-(5-Chloro-thiophen-2-yl)-meth-(Z)-ylidene]-7-...)
Affinity DataKi:  9.70nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127626(5-(3',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  9.70nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133740(9-[1-[5-(4-Methoxy-phenyl)-thiophen-2-yl]-meth-(Z)...)
Affinity DataKi:  10nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127627(5-[5-(4-Methoxy-phenyl)-thiophen-2-ylmethylene]-3-...)
Affinity DataKi:  10.3nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127641(5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  13.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127642(5-(4-Furan-2-yl-benzylidene)-3-aza-tricyclo[4.4.2....)
Affinity DataKi:  13.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133745(9-[1-(5-Phenyl-thiophen-2-yl)-meth-(Z)-ylidene]-7-...)
Affinity DataKi:  14nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166341(9-[3-(4-Fluoro-phenyl)-prop-2-yn-(Z)-ylidene]-7-az...)
Affinity DataKi:  17nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127644(5-(3'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  17.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127625(5-(4-Thiophen-2-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  19.8nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133748(9-[1-(5-Bromo-thiophen-2-yl)-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  20nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127635(5-(4-Thiophen-3-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  20.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166329(9-[3-Thiophen-3-yl-prop-2-yn-(Z)-ylidene]-7-aza-tr...)
Affinity DataKi:  22nMAssay Description:Inhibitory constant for [3H]-NE reuptake at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127624(5-[4-(5-Methyl-thiophen-2-yl)-benzylidene]-3-aza-t...)
Affinity DataKi:  22.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127634(5-(4'-Methyl-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  22.7nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50111025(9-[1-Thiophen-2-yl-meth-(Z)-ylidene]-7-aza-tricycl...)
Affinity DataKi:  26nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50111028(9-[1-(5-Iodo-thiophen-2-yl)-meth-(Z)-ylidene]-7-az...)
Affinity DataKi:  29nMAssay Description:Ability to inhibit reuptake of serotonin ([3H]5-HT) at serotonin transporter of rat midbrianMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166336(9-[1-[2,3']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166328(9-[3-(2,6-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127630(5-(4'-Cyano-biphenyl-4-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  32.4nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133751(9-[1-Thiophen-3-yl-meth-(Z)-ylidene]-7-aza-tricycl...)
Affinity DataKi:  33nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133748(9-[1-(5-Bromo-thiophen-2-yl)-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  36nMAssay Description:Ability to inhibit reuptake of serotonin ([3H]5-HT) at serotonin transporter of rat midbrianMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133744(9-[1-(5-Bromo-4-methyl-thiophen-2-yl)-meth-(Z)-yli...)
Affinity DataKi:  37nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127638(5-(4'-Methoxy-biphenyl-4-ylmethylene)-3-aza-tricyc...)
Affinity DataKi:  39nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127628(5-(4-Pyrrol-1-yl-benzylidene)-3-aza-tricyclo[4.4.2...)
Affinity DataKi:  45.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127632(Acetic acid 5-biphenyl-4-ylmethylene-3-aza-tricycl...)
Affinity DataKi:  46nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127630(5-(4'-Cyano-biphenyl-4-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  47nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133738(9-[1-[2,2']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  48nMAssay Description:Ability to inhibit reuptake of serotonin ([3H]5-HT) at serotonin transporter of rat midbrianMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166330(9-[3-(3-Fluoro-4-methyl-phenyl)-prop-2-yn-(Z)-ylid...)
Affinity DataKi:  52nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166326(9-[1-(4'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  53nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133753(9-[1-(5-Chloro-thiophen-2-yl)-meth-(Z)-ylidene]-7-...)
Affinity DataKi:  53nMAssay Description:Ability to inhibit reuptake of serotonin ([3H]5-HT) at serotonin transporter of rat midbrianMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127632(Acetic acid 5-biphenyl-4-ylmethylene-3-aza-tricycl...)
Affinity DataKi:  57nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127622(5-(4'-Methylamino-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  57.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133756(9-[1-(5'-Chloro-[2,2']bithiophenyl-5-yl)-meth-(Z)-...)
Affinity DataKi:  58nMAssay Description:Ability to inhibit reuptake of norepinephrine ([3H]NE) at norepinephrine transporter of rat parietal/occipital regionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127643(5-(3',5'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  61nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166327(9-[1-(4'-Methylsulfanyl-biphenyl-4-yl)-meth-(Z)-yl...)
Affinity DataKi:  62nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50166337(9-[3-(3,4-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  69nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50127641(5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  71nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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