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Found 228 with Last Name = 'kwong' and Initial = 'aj'
TargetDual specificity mitogen-activated protein kinase kinase 5(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50434072(CHEMBL2381342)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of MEK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559800(CHEMBL3329977)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 5(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559802(CHEMBL4303171)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of MEK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50553870(CHEMBL4749823)
Affinity DataIC50:  5nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50206444(CHEMBL3901151)
Affinity DataIC50:  6nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615119(CHEMBL5284723)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559801(CHEMBL4787266)
Affinity DataIC50:  14nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)
Affinity DataIC50:  41nMAssay Description:Inhibition of MEK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)
Affinity DataIC50:  41nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615123(CHEMBL5283781)
Affinity DataIC50:  42nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615102(CHEMBL5271442)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558862(US11370770, Compound 6n)
Affinity DataIC50:  60nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50577661(CHEMBL4879048)
Affinity DataIC50:  61nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558880(US11370770, Compound 6ee)
Affinity DataIC50:  63nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615113(CHEMBL5267499)
Affinity DataIC50:  66nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)
Affinity DataIC50:  66nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615120(CHEMBL5279577)
Affinity DataIC50:  74nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50577689(CHEMBL4866649)
Affinity DataIC50:  83nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50577657(CHEMBL4848865)
Affinity DataIC50:  96nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50577689(CHEMBL4866649)
Affinity DataIC50:  96nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK7 expressed in Sf21 cells using JNK1 as substrate pre-incubated for 30 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558875(US11370770, Compound 6z)
Affinity DataIC50:  100nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)
Affinity DataIC50:  100nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558864(US11370770, Compound 6p)
Affinity DataIC50:  110nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615118(CHEMBL5271266)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615122(CHEMBL5267684)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558878(US11370770, Compound 6cc)
Affinity DataIC50:  120nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558862(US11370770, Compound 6n)
Affinity DataIC50:  130nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558867(US11370770, Compound 6s)
Affinity DataIC50:  150nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558848(US11370770, Compound 6a)
Affinity DataIC50:  180nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558867(US11370770, Compound 6s)
Affinity DataIC50:  180nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50559799(CHEMBL4748767)
Affinity DataIC50:  190nMAssay Description:Inhibition of MEK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558866(US11370770, Compound 6r)
Affinity DataIC50:  200nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558865(US11370770, Compound 6q)
Affinity DataIC50:  210nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558867(US11370770, Compound 6s)
Affinity DataIC50:  220nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50504351(CHEMBL100206)
Affinity DataIC50:  230nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558858(US11370770, Compound 6j)
Affinity DataIC50:  240nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558858(US11370770, Compound 6j)
Affinity DataIC50:  250nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615109(CHEMBL5282673)
Affinity DataIC50:  260nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558880(US11370770, Compound 6ee)
Affinity DataIC50:  260nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615129(CHEMBL5277855)
Affinity DataIC50:  260nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM31085(1-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluorom...)
Affinity DataIC50:  260nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615110(CHEMBL5271906)
Affinity DataIC50:  270nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50577686(CHEMBL4865159)
Affinity DataIC50:  290nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615128(CHEMBL5272546)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50577671(CHEMBL4872723)
Affinity DataIC50:  310nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50577647(CHEMBL4849172)
Affinity DataIC50:  310nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))
Northwestern University

US Patent
LigandPNGBDBM558875(US11370770, Compound 6z)
Affinity DataIC50:  350nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615121(CHEMBL5271334)
Affinity DataIC50:  360nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 7(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50615130(CHEMBL5271519)
Affinity DataIC50:  360nMAssay Description:Inhibition of human recombinant full-length MEK7 using JNK1 as substrate incubated for 30 mins followed by ATP addition measured after 1 hr by ADP Gl...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM558875(US11370770, Compound 6z)
Affinity DataIC50:  360nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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