Affinity DataKi: 0.0460nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu
Curated by ChEMBL
Chaminade University Of Honolulu
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu
Curated by ChEMBL
Chaminade University Of Honolulu
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu
Curated by ChEMBL
Chaminade University Of Honolulu
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu
Curated by ChEMBL
Chaminade University Of Honolulu
Curated by ChEMBL
Affinity DataKi: 0.470nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.741nMAssay Description:Binding Affinity was determined against Dopamine receptor D1 in rat striatal membranes using [3H]- SCH 23390 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu
Curated by ChEMBL
Chaminade University Of Honolulu
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding Affinity was determined against Dopamine receptor D2 in rat striatal membranes using [3H]- spiperone radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair