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Found 963 with Last Name = 'lau' and Initial = 'f'
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.0460nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389778(CHEMBL2070251)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389773(CHEMBL2070246)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389771(CHEMBL2070243)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389780(CHEMBL2069317)
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu

Curated by ChEMBL
LigandPNGBDBM50171394(2-Decyl-2H-pyrazolo[3,4-d]pyrimidin-4-ylamine | CH...)
Affinity DataKi:  0.130nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389777(CHEMBL2070250)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389776(CHEMBL2070249)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389774(CHEMBL2070247)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389769(BREMELANOTIDE)
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389779(CHEMBL2070252)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu

Curated by ChEMBL
LigandPNGBDBM50171396(1-((R)-4-Amino-pyrazolo[3,4-d]pyrimidin-2-yl)-deca...)
Affinity DataKi:  0.280nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389775(CHEMBL2070248)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054088((2R,3R)-2-(Methyl-propyl-amino)-3-phenyl-indan-5-o...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054088((2R,3R)-2-(Methyl-propyl-amino)-3-phenyl-indan-5-o...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataKi:  0.370nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu

Curated by ChEMBL
LigandPNGBDBM50213599((6aR,10aR)-3-(6-bromo-2-methylhexan-2-yl)-6,6,9-tr...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054084((2R,3R)-2-(Allyl-methyl-amino)-3-phenyl-indan-5-ol...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054084((2R,3R)-2-(Allyl-methyl-amino)-3-phenyl-indan-5-ol...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu

Curated by ChEMBL
LigandPNGBDBM50171395(2-Undecyl-2H-pyrazolo[3,4-d]pyrimidin-4-ylamine | ...)
Affinity DataKi:  0.470nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataKi:  0.470nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.480nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389782(CHEMBL2070374)
Affinity DataKi:  0.580nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054089((2R,3R)-2-Amino-3-phenyl-indan-5-ol | CHEMBL135224)
Affinity DataKi:  0.590nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054089((2R,3R)-2-Amino-3-phenyl-indan-5-ol | CHEMBL135224)
Affinity DataKi:  0.590nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.730nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.741nMAssay Description:Binding Affinity was determined against Dopamine receptor D1 in rat striatal membranes using [3H]- SCH 23390 radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataKi:  0.780nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054084((2R,3R)-2-(Allyl-methyl-amino)-3-phenyl-indan-5-ol...)
Affinity DataKi:  0.790nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054084((2R,3R)-2-(Allyl-methyl-amino)-3-phenyl-indan-5-ol...)
Affinity DataKi:  0.790nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054091((2R,3R)-2-Dipropylamino-3-phenyl-indan-5-ol | CHEM...)
Affinity DataKi:  0.840nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054091((2R,3R)-2-Dipropylamino-3-phenyl-indan-5-ol | CHEM...)
Affinity DataKi:  0.840nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal homogenate by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054088((2R,3R)-2-(Methyl-propyl-amino)-3-phenyl-indan-5-o...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054088((2R,3R)-2-(Methyl-propyl-amino)-3-phenyl-indan-5-o...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389772(CHEMBL2070244)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389773(CHEMBL2070246)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chaminade University Of Honolulu

Curated by ChEMBL
LigandPNGBDBM50337798((6aR,10aR)-3-(8-bromo-2-methyloctan-2-yl)-6,6,9-tr...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human recombinant His-tagged VEGFR2 assessed as infrared absorptionChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389771(CHEMBL2070243)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054090((1R,2R)-2-Dipropylamino-1-phenyl-indan-5-ol | CHEM...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054090((1R,2R)-2-Dipropylamino-1-phenyl-indan-5-ol | CHEM...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389783(CHEMBL2070245)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  2.10nMAssay Description:Binding Affinity was determined against Dopamine receptor D2 in rat striatal membranes using [3H]- spiperone radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50389771(CHEMBL2070243)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054089((2R,3R)-2-Amino-3-phenyl-indan-5-ol | CHEMBL135224)
Affinity DataKi:  2.5nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50054089((2R,3R)-2-Amino-3-phenyl-indan-5-ol | CHEMBL135224)
Affinity DataKi:  2.5nMAssay Description:Binding affinity at Dopamine receptor D1 in rat neostriatum by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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