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Found 21 with Last Name = 'lesnard' and Initial = 'a'
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170158(1-(2-Methoxy-phenyl)-4-(1-o-tolyl-1H-pyrrol-3-ylme...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170156(2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210122(CHEMBL234881 | [2-(2',6'-dimethyl-biphenyl-3-yl)-e...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210124(2-(2'-methyl-biphenyl-3-yl)-ethylamine | CHEMBL234...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210123(CHEMBL395870 | N,N-dimethyl-2-(2'-methylbiphenyl-3...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210126(CHEMBL232792 | [2-(2'-methoxy-biphenyl-3-yl)-ethyl...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210125(CHEMBL232791 | [2-(2',6'-dimethoxy-biphenyl-3-yl)-...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170158(1-(2-Methoxy-phenyl)-4-(1-o-tolyl-1H-pyrrol-3-ylme...)
Affinity DataKi:  9.90nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170159(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-p...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170159(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-p...)
Affinity DataKi:  18.5nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170156(2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1...)
Affinity DataKi:  33.7nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50210123(CHEMBL395870 | N,N-dimethyl-2-(2'-methylbiphenyl-3...)
Affinity DataKi:  443nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50210126(CHEMBL232792 | [2-(2'-methoxy-biphenyl-3-yl)-ethyl...)
Affinity DataKi:  531nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50210124(2-(2'-methyl-biphenyl-3-yl)-ethylamine | CHEMBL234...)
Affinity DataKi:  1.47E+3nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50210122(CHEMBL234881 | [2-(2',6'-dimethyl-biphenyl-3-yl)-e...)
Affinity DataKi:  2.25E+3nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50210125(CHEMBL232791 | [2-(2',6'-dimethoxy-biphenyl-3-yl)-...)
Affinity DataKi:  4.83E+3nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Universit?? Pierre Et Marie Curie

LigandPNGBDBM32021(4,5-bis(oxidanyl)-9,10-bis(oxidanylidene)anthracen...)
Affinity DataKd:  9.60E+3nMpH: 7.5 T: 2°CAssay Description:We incubated human recombinant CDK2/cyclin A with small molecules at the indicatedconcentrations in buffer A (Tris真HCl (25 mm, pH 7.5), MgCl2 (10 mm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Universit?? Pierre Et Marie Curie

LigandPNGBDBM150754(11-O-acetyl-aloe-emodin | 3-[(acetyloxy)methyl]-1,...)
Affinity DataKd:  1.78E+4nMpH: 7.5 T: 2°CAssay Description:We incubated human recombinant CDK2/cyclin A with small molecules at the indicatedconcentrations in buffer A (Tris真HCl (25 mm, pH 7.5), MgCl2 (10 mm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Universit?? Pierre Et Marie Curie

LigandPNGBDBM43654(7,8-dihydro-6H-cyclopenta[4,5]thieno[1,2-c]pyrimid...)
Affinity DataKd:  2.87E+5nMpH: 7.5 T: 2°CAssay Description:We incubated human recombinant CDK2/cyclin A with small molecules at the indicatedconcentrations in buffer A (Tris真HCl (25 mm, pH 7.5), MgCl2 (10 mm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Universit?? Pierre Et Marie Curie

LigandPNGBDBM150753(4-hydrazino-6,7,8,9-tetrahydro-5H-cyclohepta[4,5]t...)
Affinity DataKd:  3.25E+4nMpH: 7.5 T: 2°CAssay Description:We incubated human recombinant CDK2/cyclin A with small molecules at the indicatedconcentrations in buffer A (Tris真HCl (25 mm, pH 7.5), MgCl2 (10 mm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Universit?? Pierre Et Marie Curie

LigandPNGBDBM150752(4-hydrazino-5,6,7,8-tetrahydro[1]benzothieno[2,3-d...)
Affinity DataKd:  2.83E+4nMpH: 7.5 T: 2°CAssay Description:We incubated human recombinant CDK2/cyclin A with small molecules at the indicatedconcentrations in buffer A (Tris真HCl (25 mm, pH 7.5), MgCl2 (10 mm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed