Affinity DataKi: 0.25nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24.5nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 202nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 215nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 331nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 431nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 478nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.65E+3nMAssay Description:Binding affinity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Antagonist activity in human bradykinin B1 receptor by FLIPR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Antagonist activity in human bradykinin B1 receptor by FLIPR methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of MK-499 from human ERG channel in HEK293 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Displacement of MK-499 from human ERG channel in HEK293 cellsMore data for this Ligand-Target Pair