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Found 33 with Last Name = 'liu' and Initial = 'wq'
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080832(CHEMBL334099 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataIC50:  11nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213228(2-(4-((S)-3-((S)-1-((S)-2-(((S)-5-amino-1-((2S,3R)...)
Affinity DataIC50:  108nMAssay Description:Inhibition of STAT3 dimer DNA binding activity by ELISA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080831(CHEMBL434413 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataIC50:  120nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080836(4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-phos...)
Affinity DataIC50:  153nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080834(CHEMBL409455 | {4-[2-[2-(3-Amino-benzyloxycarbonyl...)
Affinity DataIC50:  198nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080830(CHEMBL333070 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataIC50:  235nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080833(CHEMBL264635 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataIC50:  497nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213225((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-3-(4-(2...)
Affinity DataIC50: >800nMAssay Description:Inhibition of STAT3 dimer DNA binding activity by ELISA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213227((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-3-(4-((...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of STAT3 dimer DNA binding activity by ELISA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213226((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-aceta...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of STAT3 dimer DNA binding activity by ELISA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080835(CHEMBL333527 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataIC50:  1.10E+3nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213224((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-aceta...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of STAT3 dimer DNA binding activity by ELISA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50257256(CHEMBL4092853)
Affinity DataIC50:  1.04E+4nMAssay Description:Displacement of biotinylated VEGF-A (165 residues) from humanized recombinant C-terminal His-tagged VEGFR-1 extracellular domain expressed in baculov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50257258(CHEMBL4062433)
Affinity DataIC50:  5.04E+4nMAssay Description:Displacement of biotinylated VEGF-A (165 residues) from humanized recombinant C-terminal His-tagged VEGFR-1 extracellular domain expressed in baculov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50257253(CHEMBL4077087)
Affinity DataIC50:  5.60E+4nMAssay Description:Displacement of biotinylated VEGF-A (165 residues) from humanized recombinant C-terminal His-tagged VEGFR-1 extracellular domain expressed in baculov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50257257(CHEMBL4071072)
Affinity DataIC50:  7.51E+4nMAssay Description:Displacement of biotinylated VEGF-A (165 residues) from humanized recombinant C-terminal His-tagged VEGFR-1 extracellular domain expressed in baculov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50257259(CHEMBL4083044)
Affinity DataIC50:  1.30E+5nMAssay Description:Displacement of biotinylated VEGF-A (165 residues) from humanized recombinant C-terminal His-tagged VEGFR-1 extracellular domain expressed in baculov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50213223((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-aceta...)
Affinity DataIC50:  1.38E+5nMAssay Description:Inhibition of STAT3 dimer DNA binding activity by ELISA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50257261(CHEMBL4090414)
Affinity DataIC50:  1.57E+5nMAssay Description:Displacement of biotinylated VEGF-A (165 residues) from humanized recombinant C-terminal His-tagged VEGFR-1 extracellular domain expressed in baculov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50521337(CHEMBL4592007)
Affinity DataIC50:  1.96E+5nMAssay Description:Displacement of biotinylated VEGF-A165 from human VEGFR-1 ECD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50257260(CHEMBL4090834)
Affinity DataIC50:  2.71E+5nMAssay Description:Displacement of biotinylated VEGF-A (165 residues) from humanized recombinant C-terminal His-tagged VEGFR-1 extracellular domain expressed in baculov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Umr 8638 Cnrs

Curated by ChEMBL
LigandPNGBDBM50521337(CHEMBL4592007)
Affinity DataKd:  6.21E+5nMAssay Description:Binding affinity to 15N-labeled VEGFR1 domain 2 (unknown origin) at 26 mM by TROSY [1H-15N] spectroscopic analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50087245(CHEMBL345170 | Pro-Ser-Pmp-Val-Asn-Val-Gln-Asn)
Affinity DataKd:  260nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50087244(Ac-Pro-Phe-pTyr-Val-Asn-Val-Pro-NH2 | CHEMBL237124...)
Affinity DataKd:  30nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50087243(CHEMBL436789 | Pro-Ser-F2Pmp-Val-Asn-Val-Gln-Asn)
Affinity DataKd:  200nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50087242(CHEMBL422705 | Pro-Ser-pTyr-Val-Asn-Val-Gln-Asn)
Affinity DataKd:  18nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080836(4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-phos...)
Affinity DataKd:  45nMAssay Description:The copound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Ment...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080835(CHEMBL333527 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataKd:  250nMAssay Description:The copound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Ment...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080832(CHEMBL334099 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataKd:  3nMAssay Description:The copound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Ment...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080830(CHEMBL333070 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataKd:  60nMAssay Description:The copound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Ment...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080833(CHEMBL264635 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataKd:  155nMAssay Description:The copound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Ment...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080834(CHEMBL409455 | {4-[2-[2-(3-Amino-benzyloxycarbonyl...)
Affinity DataKd:  60nMAssay Description:The copound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Ment...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50080831(CHEMBL434413 | [1-[1-(1,2-Dicarbamoyl-ethylcarbamo...)
Affinity DataKd:  30nMAssay Description:The copound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Ment...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed