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Found 85 with Last Name = 'nobusada' and Initial = 'h'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344330((S)-2-(3-((4-(4-Fluorophenoxy)benzamido)methyl)-4-...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344331(CHEMBL270587 | rac-2-(3-{[(biphenyl-4-carbonyl)-am...)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344332(2-(4-methoxy-3-((4-phenoxybenzamido)methyl)benzyl)...)
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344333(CHEMBL1779473 | rac-2-(4-Methoxy-3-((4-(trifluorom...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344334((S)-2-(3-((4-(4-Chlorophenoxy)benzamido)methyl)-4-...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344335((S)-2-(3-((4-(4-bromophenoxy)benzamido)methyl)-4-m...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344336(CHEMBL1779474 | rac-2-(4-Methoxy-3-((3-phenoxybenz...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344337(CHEMBL1779478 | rac-2-(3-((4-(Benzyloxy)benzamido)...)
Affinity DataEC50:  52nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344338(CHEMBL1779479 | rac-2-(4-Methoxy-3-((4-phenethoxyb...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344339(CHEMBL1779476 | rac-2-(4-Methoxy-3-((3-phenylbenza...)
Affinity DataEC50:  74nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344340(CHEMBL255392 | rac-2-(3-(4-Methylbenzamidomethyl)-...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344333(CHEMBL1779473 | rac-2-(4-Methoxy-3-((4-(trifluorom...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344332(2-(4-methoxy-3-((4-phenoxybenzamido)methyl)benzyl)...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344331(CHEMBL270587 | rac-2-(3-{[(biphenyl-4-carbonyl)-am...)
Affinity DataEC50:  210nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344330((S)-2-(3-((4-(4-Fluorophenoxy)benzamido)methyl)-4-...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344331(CHEMBL270587 | rac-2-(3-{[(biphenyl-4-carbonyl)-am...)
Affinity DataEC50:  340nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344340(CHEMBL255392 | rac-2-(3-(4-Methylbenzamidomethyl)-...)
Affinity DataEC50:  360nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344337(CHEMBL1779478 | rac-2-(3-((4-(Benzyloxy)benzamido)...)
Affinity DataEC50:  460nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344334((S)-2-(3-((4-(4-Chlorophenoxy)benzamido)methyl)-4-...)
Affinity DataEC50:  580nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344339(CHEMBL1779476 | rac-2-(4-Methoxy-3-((3-phenylbenza...)
Affinity DataEC50:  710nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344338(CHEMBL1779479 | rac-2-(4-Methoxy-3-((4-phenethoxyb...)
Affinity DataEC50:  780nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344335((S)-2-(3-((4-(4-bromophenoxy)benzamido)methyl)-4-m...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344332(2-(4-methoxy-3-((4-phenoxybenzamido)methyl)benzyl)...)
Affinity DataEC50:  820nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344334((S)-2-(3-((4-(4-Chlorophenoxy)benzamido)methyl)-4-...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344330((S)-2-(3-((4-(4-Fluorophenoxy)benzamido)methyl)-4-...)
Affinity DataEC50:  920nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344335((S)-2-(3-((4-(4-bromophenoxy)benzamido)methyl)-4-m...)
Affinity DataEC50:  990nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344337(CHEMBL1779478 | rac-2-(3-((4-(Benzyloxy)benzamido)...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344338(CHEMBL1779479 | rac-2-(4-Methoxy-3-((4-phenethoxyb...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344341(CHEMBL255593 | rac-2-(3-(benzamidomethyl)-4-methox...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344342(CHEMBL1779475 | rac-2-(4-Methoxy-3-((2-phenoxybenz...)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344343(CHEMBL1779477 | rac-2-(4-Methoxy-3-((2-phenylbenza...)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344339(CHEMBL1779476 | rac-2-(4-Methoxy-3-((3-phenylbenza...)
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344333(CHEMBL1779473 | rac-2-(4-Methoxy-3-((4-(trifluorom...)
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344336(CHEMBL1779474 | rac-2-(4-Methoxy-3-((3-phenoxybenz...)
Affinity DataEC50:  4.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344336(CHEMBL1779474 | rac-2-(4-Methoxy-3-((3-phenoxybenz...)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344341(CHEMBL255593 | rac-2-(3-(benzamidomethyl)-4-methox...)
Affinity DataEC50:  8.10E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344340(CHEMBL255392 | rac-2-(3-(4-Methylbenzamidomethyl)-...)
Affinity DataEC50:  9.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344342(CHEMBL1779475 | rac-2-(4-Methoxy-3-((2-phenoxybenz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344343(CHEMBL1779477 | rac-2-(4-Methoxy-3-((2-phenylbenza...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344341(CHEMBL255593 | rac-2-(3-(benzamidomethyl)-4-methox...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344342(CHEMBL1779475 | rac-2-(4-Methoxy-3-((2-phenoxybenz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344343(CHEMBL1779477 | rac-2-(4-Methoxy-3-((2-phenylbenza...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50231507((2S)-2-(4-propoxy-3-{[({4-[(3S,5S,7S)-tricyclo[3.3...)
Affinity DataEC50:  54nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176605((S)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  12nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176605((S)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  23nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176609((R)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  150nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176609((R)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  840nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50214207((2S)-2-{4-butoxy-3-[({[2-fluoro-4-(trifluoromethyl...)
Affinity DataEC50:  250nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50214207((2S)-2-{4-butoxy-3-[({[2-fluoro-4-(trifluoromethyl...)
Affinity DataEC50:  0.720nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50214209((R)-2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)be...)
Affinity DataEC50:  620nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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