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Found 30 with Last Name = 'onose' and Initial = 'j'
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  930nMAssay Description:Binding affinity to recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  1.07E+3nMAssay Description:Binding affinity to full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  1.25E+4nMAssay Description:Competitive inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  300nMAssay Description:Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of mouse anti-DNP IgE-stimulated beta-hexosaminidase release preincubated for 15 mins fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  500nMAssay Description:Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of anti-DNP IgE-stimulated TNFalpha release preincubated for 15 mins followed by mouse a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  800nMAssay Description:Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of ionomycin-stimulated beta-hexosaminidase release preincubated for 15 mins followed by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of ionomycin-stimulated TNFalpha release preincubated for 15 mins followed by ionomycin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 4(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human USP4 using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536673(CHEMBL4587307)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536673(CHEMBL4587307)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536672(CHEMBL2012939)
Affinity DataIC50:  2.71E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable ubiquitin carboxyl-terminal hydrolase FAF-X(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of USP9x in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of USP5 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of UCH-L1 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536672(CHEMBL2012939)
Affinity DataIC50:  3.76E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536674(CHEMBL4593579)
Affinity DataIC50:  3.79E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437694(CHEMBL1410015)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human USP14More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536674(CHEMBL4593579)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536671(CHEMBL2013072)
Affinity DataIC50:  9.73E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50539389(CHEMBL4636684)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of PKCbeta in rat RBL2H3 cells assessed as inhibition of mouse anti-DNP IgE-stimulated beta-hexosaminidase release preincubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50539389(CHEMBL4636684)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of PKCbeta in rat RBL2H3 cells assessed as inhibition of anti-DNP IgE-stimulated TNFalpha release preincubated for 15 mins followed by mou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50539389(CHEMBL4636684)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of PKCbeta in rat RBL2H3 cells assessed as inhibition of ionomycin-stimulated TNFalpha release preincubated for 15 mins followed by ionomy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50539389(CHEMBL4636684)
Affinity DataIC50:  2.22E+4nMAssay Description:Inhibition of PKCbeta in rat RBL2H3 cells assessed as inhibition of ionomycin-stimulated beta-hexosaminidase release preincubated for 15 mins followe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibition of human UCH-L1 using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50539389(CHEMBL4636684)
Affinity DataIC50:  3.62E+4nMAssay Description:Inhibition of recombinant full-length N-temrinal GST-tagged human PKC beta1 expressed in baculovirus infected Sf9 cells using TMB as substrate incuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536671(CHEMBL2013072)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed