Compile Data Set for Download or QSAR
maximum 50k data
Found 136 with Last Name = 'pérez' and Initial = 'y'
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443182(CHEMBL3086538)
Affinity DataKi:  0.5nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443181(CHEMBL3086535)
Affinity DataKi:  0.600nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443180(CHEMBL3086536)
Affinity DataKi:  0.700nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443178(CHEMBL3086537)
Affinity DataKi:  1.90nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443177(CHEMBL3086533)
Affinity DataKi:  2.5nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443189(CHEMBL3086327)
Affinity DataKi:  5.30nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443188(CHEMBL3086329)
Affinity DataKi:  6.40nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443187(CHEMBL3086328)
Affinity DataKi:  6.60nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443175(CHEMBL3086534)
Affinity DataKi:  8.40nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443186(CHEMBL3086331)
Affinity DataKi:  30nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443185(CHEMBL3086330)
Affinity DataKi:  43nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443184(CHEMBL3086544)
Affinity DataKi:  50nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443183(CHEMBL3086545)
Affinity DataKi:  85nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443194(CHEMBL3086542)
Affinity DataKi:  230nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443193(CHEMBL3086540)
Affinity DataKi:  380nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443192(CHEMBL3086539)
Affinity DataKi:  460nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443179(CHEMBL3086332)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443191(CHEMBL3086541)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443176(CHEMBL3086326)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443190(CHEMBL3086543)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371120(CHEMBL242173)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371127(CHEMBL244681)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371125(CHEMBL244088)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371131(CHEMBL390874)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371118(CHEMBL244693)
Affinity DataKi:  1.70E+5nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371123(CHEMBL244090)
Affinity DataKi:  2.40E+5nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM38435(9-ethyl-1-oxo-2,3,4,9-tetrahydro-1H-carbazole-6-ca...)
Affinity DataKi:  6.10E+5nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371126(CHEMBL438508)
Affinity DataKi:  8.80E+5nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371130(CHEMBL390873)
Affinity DataKi:  9.10E+5nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371117(CHEMBL242146)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371116(CHEMBL242148)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371119(CHEMBL244696)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371121(CHEMBL440951)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371122(CHEMBL242363)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371124(CHEMBL244694)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371129(CHEMBL244328)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow molecular weight phosphotyrosine protein phosphatase(Bos taurus)
Institute For Research In Biomedicine (Irb)

Curated by ChEMBL
LigandPNGBDBM50371128(CHEMBL390401)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of bovine low molecular weight PTP expressed in Escherichia coli BL21(D3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50355323(CHEMBL1835228)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50355325(CHEMBL1835231)
Affinity DataIC50:  0.740nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50300895(3-(3-methoxyphenyl)-6-methyl-2H-chromen-2-one | CH...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50355320(CHEMBL1835224)
Affinity DataIC50:  1.52nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50443493(CHEMBL3087777)
Affinity DataIC50:  2nMAssay Description:Inhibition of full-length aurora-B (unknown origin) using 5FAMLRRASLG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50355318(CHEMBL1835230)
Affinity DataIC50:  2.73nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50355326(CHEMBL1835232)
Affinity DataIC50:  3.25nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50443493(CHEMBL3087777)
Affinity DataIC50:  4nMAssay Description:Inhibition of N-terminal HIS-tagged aurora-A (unknown origin) using 5FAM-LRRASLG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50443508(CHEMBL3087781)
Affinity DataIC50:  5nMAssay Description:Inhibition of N-terminal HIS-tagged aurora-A (unknown origin) using 5FAM-LRRASLG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50443510(CHEMBL3087779)
Affinity DataIC50:  5nMAssay Description:Inhibition of N-terminal HIS-tagged aurora-A (unknown origin) using 5FAM-LRRASLG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50443509(CHEMBL3087780)
Affinity DataIC50:  7nMAssay Description:Inhibition of N-terminal HIS-tagged aurora-A (unknown origin) using 5FAM-LRRASLG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50443492(CHEMBL3087778)
Affinity DataIC50:  7nMAssay Description:Inhibition of full-length aurora-B (unknown origin) using 5FAMLRRASLG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50443510(CHEMBL3087779)
Affinity DataIC50:  8nMAssay Description:Inhibition of full-length aurora-B (unknown origin) using 5FAMLRRASLG-CONH2 as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 136 total ) | Next | Last >>
Jump to: