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Found 35 with Last Name = 'pengsuparp' and Initial = 't'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50002662((+)-calanolide A | (+)-calnolide A | (10R,11S,12S)...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50002662((+)-calanolide A | (+)-calnolide A | (10R,11S,12S)...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50050430((10S,12S)-12-Hydroxy-6,6,10,11-tetramethyl-4-propy...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50050430((10S,12S)-12-Hydroxy-6,6,10,11-tetramethyl-4-propy...)
Affinity DataIC50:  970nMAssay Description:Inhibitory activity against RNA-dependent DNA polymerase(RDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292441(1beta-hydroxyaleuritolic acid 3-p-hydroxybenzoate ...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478513(2Alpha-Hydroxymaprounic Acid | CHEMBL469925)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478517(CHEBI:66672 | CHEMBL472320)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478511(CHEBI:66671 | CHEMBL449431)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478512(1Beta-Hydroxymaprounic Acid | CHEMBL512314)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50250356((+)-protolichesterinic acid | CHEMBL490329 | proto...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50002662((+)-calanolide A | (+)-calnolide A | (10R,11S,12S)...)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibitory activity against TIBO-resistant HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50370476(Combivir | ZIDOVUDINE TRIPHOSPHATE)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478514(Fagaronine | Fagaronine Chloride)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50336799(5,5',5''-[1,3,6-naphthalenetriyltris(sulfonylimino...)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478516(CHEBI:81067 | CHEMBL471812 | O-Methylpsychotrine)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50370476(Combivir | ZIDOVUDINE TRIPHOSPHATE)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of DNA polymerase betaMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50050430((10S,12S)-12-Hydroxy-6,6,10,11-tetramethyl-4-propy...)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibitory activity against TIBO-resistant HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478515(Aleuritolic Acid | CHEBI:73107 | Maprounic Acid)
Affinity DataIC50:  2.49E+4nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50050431((-)-calanolide B | (10S,11R,12S)-12-Hydroxy-6,6,10...)
Affinity DataIC50:  2.78E+4nMAssay Description:Inhibitory activity against RNA-dependent DNA polymerase(RDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50412092(SWERTIFRANCHESIDE)
Affinity DataIC50:  5.77E+4nMAssay Description:Inhibition of DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50323214(6-[4-(5,7-Dihydroxy-4-oxo-4H-chromen-2-yl)-phenoxy...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50323212(6-[5-(5,7-Dihydroxy-4-oxo-4H-chromen-2-yl)-2-hydro...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478418(Agathisflavone | CHEBI:2512)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478419((+)-Morelloflavone | Morelloflavone)
Affinity DataIC50:  1.16E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50129952(2-(3-(5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4H-c...)
Affinity DataIC50:  1.19E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478510(3-Acetylaleuritolic Acid | Acetyl Aleuritolic Acid...)
Affinity DataIC50:  1.36E+5nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Medichem Research

Curated by ChEMBL
LigandPNGBDBM50050431((-)-calanolide B | (10S,11R,12S)-12-Hydroxy-6,6,10...)
Affinity DataIC50:  1.56E+5nMAssay Description:Inhibitory activity against DNA -dependent DNA polymerase(DDDP) of HIV-1 RT Nucleic Acid polymeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478414(CHEBI:66626 | Nigranoic Acid)
Affinity DataIC50:  1.59E+5nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478421(CHEMBL445452)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002662((+)-calanolide A | (+)-calnolide A | (10R,11S,12S)...)
Affinity DataIC50:  2.05E+5nMAssay Description:Inhibition of DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50368352(Cerubidine | DAUNORUBICIN)
Affinity DataIC50:  2.36E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50478420(CHEMBL456859)
Affinity DataIC50:  2.36E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  4.43E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase p66/p51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292362(CHEMBL466773 | Soulattrolide)
Affinity DataIC50: >4.95E+5nMAssay Description:Inhibition of DNA polymerase betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed