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Found 543 with Last Name = 'rief' and Initial = 's'
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492784(CHEMBL2413837)
Affinity DataKi:  0.0450nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492781(CHEMBL2413835)
Affinity DataKi:  0.0570nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326663(CHEMBL1255022)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326662(10-hydroxy-17-methoxy-4-methyl-(13R,17S)-12-oxa-4-...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492783(CHEMBL2413824)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326662(10-hydroxy-17-methoxy-4-methyl-(13R,17S)-12-oxa-4-...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50166216(17-benzyloxy-10-hydroxy-4-methyl-(13R,17S)-12-oxa-...)
Affinity DataKi:  0.120nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492772(CHEMBL2413828)
Affinity DataKi:  0.130nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50127165(10-hydroxy-17-methoxy-4,13-dimethyl-(13R,17S)-12-o...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50166212(17-ethoxy-10-hydroxy-13-methyl-4-phenethyl-(13R,17...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492769(CHEMBL2413836)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50166214(10-hydroxy-4-methyl-17-(1-naphthylmethoxy)-(13R,17...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50166215(17-benzyloxy-10-hydroxy-4,13-dimethyl-(13R,17S)-12...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548314(CHEMBL4793888)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492780(CHEMBL2413833)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50186290(3-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50412447(CHEMBL380101)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50186269(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50186309(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548310(CHEMBL4755067)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548285(CHEMBL4792012)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492782(CHEMBL2413829)
Affinity DataKi:  0.490nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50259267(CHEMBL4099779)
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492774(CHEMBL2413825)
Affinity DataKi:  0.510nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492773(CHEMBL2413827)
Affinity DataKi:  0.530nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548313(CHEMBL4741873)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50186283(2-ethyl-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.540nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492768(CHEMBL2413838)
Affinity DataKi:  0.549nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50325744(CHEMBL1223683 | N-(4-(4-(2,3-dichlorophenyl)pipera...)
Affinity DataKi:  0.600nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50166213(17-allyloxy-10-hydroxy-4-methyl-(13R,17S)-12-oxa-4...)
Affinity DataKi:  0.610nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548296(CHEMBL4757240)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492767(CHEMBL2413839)
Affinity DataKi:  0.640nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548309(CHEMBL4788003)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492770(CHEMBL2413832)
Affinity DataKi:  0.655nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492777(CHEMBL2413834)
Affinity DataKi:  0.670nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548300(CHEMBL4777389)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548292(CHEMBL4797321)
Affinity DataKi:  0.760nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548322(CHEMBL4782642)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548288(CHEMBL4743953)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548286(CHEMBL4789014)
Affinity DataKi:  0.820nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548323(CHEMBL4755734)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548312(CHEMBL4753934)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50336592(2-{[(1S,5R,13R,14S,17S)-10-hydroxy-17-methoxy-4-me...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50492766(CHEMBL2413840)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]iodoproxyfan from histamine H3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50166214(10-hydroxy-4-methyl-17-(1-naphthylmethoxy)-(13R,17...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of [3H]U-69593 binding to opioid receptor kappa from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50548320(CHEMBL4754944)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes incubated for 45 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50001707(10,17-dihydroxy-4-methyl-(13R,17S)-12-oxa-4-azapen...)
Affinity DataKi:  0.970nMAssay Description:Inhibition of [3H]DAMGO binding to opioid receptor mu from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50325748(CHEMBL1223750 | N-(4-(4-(3-(trifluoromethyl)phenyl...)
Affinity DataKi:  1nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50325746(CHEMBL1223748 | N-(4-(4-(2-methoxyphenyl)piperazin...)
Affinity DataKi:  1nMAssay Description:Antagonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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