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Found 246 with Last Name = 'sbacchi' and Initial = 'm'
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110268(CHEMBL2369895 | CSNLSTCVLGKLSQELc[DKLQK]YPRTNTGSGT...)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50024170(CHEMBL2369912)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110272(CHEMBL2369907 | CSNLSTCVLGKLSQELc[DKLHK]YPRTNTGSGT...)
Affinity DataKi:  0.0510nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110265(CHEMBL2369886 | CSNLSTCVLGKLSQELc[DKLHO]YPRTNTGSGT...)
Affinity DataKi:  0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110275(CGNLSTCBLGTYTQDF[DKFHO]YPQTAIGVGAP-amide | CHEMBL2...)
Affinity DataKi:  0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001107(2-(3,4-Dichloro-phenyl)-1-(5-hydroxy-1-pyrrolidin-...)
Affinity DataKi:  0.0900nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity of compound was determined against Opioid receptor delta 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50027063(CHEMBL2111838)
Affinity DataKi:  0.170nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50027063(CHEMBL2111838)
Affinity DataKi:  0.170nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50027064(CHEMBL2111836)
Affinity DataKi:  0.190nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001108(2-(3,4-Dichloro-phenyl)-1-(1-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001108(2-(3,4-Dichloro-phenyl)-1-(1-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  0.200nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007159(2-(3,4-Dichloro-phenyl)-1-(4-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity determined against Opioid receptor delta 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50453089(CHEMBL2114225)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131967(CHEMBL123898 | N-[2-(5-Phenyl-2,3-dihydro-1H-benzo...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131967(CHEMBL123898 | N-[2-(5-Phenyl-2,3-dihydro-1H-benzo...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131972(4-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.280nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131972(4-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.280nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049802(4-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049802(4-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007158((S)-2-(3,4-Dichloro-phenyl)-1-(2-pyrrolidin-1-ylme...)
Affinity DataKi:  0.310nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049807(2-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049807(2-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131968(CHEMBL127828 | Thiophene-3-carboxylic acid {2-[5-(...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001104(2-(3,4-Dichloro-phenyl)-1-(3-methyl-1-pyrrolidin-1...)
Affinity DataKi:  0.430nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50027064(CHEMBL2111836)
Affinity DataKi:  0.430nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50027064(CHEMBL2111836)
Affinity DataKi:  0.430nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131969(CHEMBL126688 | Thiophene-2-carboxylic acid [2-(5-p...)
Affinity DataKi:  0.450nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131969(CHEMBL126688 | Thiophene-2-carboxylic acid [2-(5-p...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007166(2-(3,4-Dichloro-phenyl)-1-(7-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007165(2-(3,4-Dichloro-phenyl)-1-(4-piperidin-1-ylmethyl-...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131973(CHEMBL338391 | N-[2-(1-Methyl-5-phenyl-2,3-dihydro...)
Affinity DataKi:  0.470nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131973(CHEMBL338391 | N-[2-(1-Methyl-5-phenyl-2,3-dihydro...)
Affinity DataKi:  0.480nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001107(2-(3,4-Dichloro-phenyl)-1-(5-hydroxy-1-pyrrolidin-...)
Affinity DataKi:  0.490nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049806(CHEMBL127969 | Thiophene-2-carboxylic acid [2-(1-m...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049806(CHEMBL127969 | Thiophene-2-carboxylic acid [2-(1-m...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig using [3H]-U-65,693 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049806(CHEMBL127969 | Thiophene-2-carboxylic acid [2-(1-m...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50453088(CHEMBL2114226)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131970(2-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50131970(2-Fluoro-N-[2-(5-phenyl-2,3-dihydro-1H-benzo[e][1,...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049808(CHEMBL127968 | N-[2-(7-Chloro-1-methyl-5-phenyl-2,...)
Affinity DataKi:  0.550nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Calcitonin receptor (1)(Homo sapiens (Human))
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50110273(CGNLSTCMLGTYTQDFc[DKFHK]FPQTAIGVGAP-amide | CHEMBL...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049802(4-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049802(4-Fluoro-N-[2-(1-methyl-5-phenyl-2,3-dihydro-1H-be...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig using [3H]-U-65,693 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007167(1-(4-Piperidin-1-ylmethyl-6,7-dihydro-4H-thieno[3,...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001105(2-(3,4-Dichloro-phenyl)-1-(4-methyl-1-pyrrolidin-1...)
Affinity DataKi:  0.600nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007157((-)-1-(1-Piperidin-1-ylmethyl-3,4-dihydro-1H-isoqu...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007164((S)-1-(2-Pyrrolidin-1-ylmethyl-piperidin-1-yl)-2-(...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Smithkline Beecham Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50007164((S)-1-(2-Pyrrolidin-1-ylmethyl-piperidin-1-yl)-2-(...)
Affinity DataKi:  0.640nMAssay Description:Evaluated for the binding affinity at kappa receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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