Affinity DataKi: 0.0230nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0510nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0690nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.0900nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity of compound was determined against Opioid receptor delta 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity determined against Opioid receptor delta 1 from human cloned receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.470nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Binding constant towards human Opioid receptor kappa 1 was reportedMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Receptor binding affinity towards opioid receptor muMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig using [3H]-U-65,693 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Inhibition of [125I]-salmon calcitonin (sCT) binding to human calcitonin receptor I1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig using [3H]-U-65,693 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Receptor binding affinity towards opioid receptor kappaMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.620nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.640nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Smithkline Beecham Farmaceutici
Curated by ChEMBL
Smithkline Beecham Farmaceutici
Curated by ChEMBL
Affinity DataKi: 0.640nMAssay Description:Evaluated for the binding affinity at kappa receptorMore data for this Ligand-Target Pair