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Found 48 with Last Name = 'skoog' and Initial = 'm'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284925(CHEMBL288759 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataKi:  24nMAssay Description:Inhibition constant against HIV protease was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM914(Aminodiol deriv. 9a | BMS-186318 analog 1 | [(S,R)...)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284924(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284924(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286514(CHEMBL357009 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  16nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286502(CHEMBL143470 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  35nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284937(CHEMBL45838 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284925(CHEMBL288759 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284937(CHEMBL45838 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284929(CHEMBL48917 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004182(2-Acetylamino-6-(4-{2-[(2-benzyloxycarbonylamino-3...)
Affinity DataIC50:  57nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284930(CHEMBL49305 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284930(CHEMBL49305 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004192(CHEMBL344981 | [2-(4-{2-[(2-Benzyloxycarbonylamino...)
Affinity DataIC50:  69nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004184(4-(4-Chloro-benzenesulfonylaminocarbonyl)-N-((S)-1...)
Affinity DataIC50:  84nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286504(CHEMBL435594 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286513(CHEMBL343727 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  105nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004190(3-Acetoxymethyl-7-methyl-5,5,8-trioxo-5lambda*6*-t...)
Affinity DataIC50:  107nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284932(CHEMBL45699 | {(1S,2R)-1-Benzyl-3-[(2R,3S)-3-(2,4-...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM914(Aminodiol deriv. 9a | BMS-186318 analog 1 | [(S,R)...)
Affinity DataIC50:  125nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM914(Aminodiol deriv. 9a | BMS-186318 analog 1 | [(S,R)...)
Affinity DataIC50:  125nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284932(CHEMBL45699 | {(1S,2R)-1-Benzyl-3-[(2R,3S)-3-(2,4-...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286511(CHEMBL140062 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  160nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286503(CHEMBL142990 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286508(CHEMBL356345 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284934(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50:  220nMAssay Description:Inhibition constant against HIV protease was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284934(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50:  220nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286509(CHEMBL143415 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  230nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284935(CHEMBL445886 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284931(CHEMBL49773 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  320nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004187(((S)-1-{Indan-2-yl-[(3,3,3-trifluoro-1-isopropyl-2...)
Affinity DataIC50:  365nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004185(4-[2-({2-[4-(4-Chloro-benzenesulfonylaminocarbonyl...)
Affinity DataIC50:  404nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286506(CHEMBL344953 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  420nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284926(CHEMBL46020 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  450nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004183(4-{2-[(2-Benzyloxycarbonylamino-3-methyl-butyryl)-...)
Affinity DataIC50:  635nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284933(CHEMBL48921 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  900nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286507(CHEMBL348226 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284927(CHEMBL297829 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286512(CHEMBL346860 | {(1S,2R)-1-Benzyl-3-[(2R,3S)-3-(2-f...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM924((1S-(1R*,2S*(2S*,3R*)))-[3-[[3-[(3,3-Dimethyl-1-ox...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004189(4-[2-({2-[4-(4-Chloro-benzenesulfonylaminocarbonyl...)
Affinity DataIC50:  4.90E+3nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004188(4-[2-({2-[4-(4-Chloro-benzenesulfonylaminocarbonyl...)
Affinity DataIC50: >5.00E+3nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004186(4-{2-[(2-Benzyloxycarbonylamino-3-methyl-butyryl)-...)
Affinity DataIC50: >5.00E+3nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284936(CHEMBL48993 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3...)
Affinity DataIC50:  6.50E+3nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286510(CHEMBL141252 | {(1S,2R)-3-[(2R,3S)-3-(2-Amino-1,1-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284928(CHEMBL301382 | {(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286505(CHEMBL140755 | [(1S,2R)-3-((2R,3S)-3-Amino-2-hydro...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004191(4-{2-[(2-Benzyloxycarbonylamino-3-methyl-butyryl)-...)
Affinity DataIC50:  1.11E+4nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed