Affinity DataKi: 24nMAssay Description:Inhibition constant against HIV protease was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 57nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 69nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 84nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 107nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition constant against HIV protease was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 365nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 404nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 635nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HIV protease cleavage of V-S-Q-N-(b-naphthylalanine)-P-I-VMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Boehringer Ingelheim Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.11E+4nMpH: 7.5Assay Description:Inhibitory activity against human leukocyte elastase (HLE) at pH 7.5More data for this Ligand-Target Pair