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Found 20 with Last Name = 'soeiro' and Initial = 'mnc'
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510706(CHEMBL4515068)
Affinity DataKi:  1.70E+4nMAssay Description:Non-competitive inhibition of Leishmania amazonensis arginase using L-arginine as substrate incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50181473(4-(4-(4-(4-(((3R,5R)-5-((1H-1,2,4-triazol-1-yl)met...)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Tulahuen CYP51 expressed in Escherichia coli JM109 cell membranes assessed as inhibition of microbe growt...More data for this Ligand-Target Pair
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50458303(CHEMBL4208391)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Tulahuen CYP51 expressed in Escherichia coli JM109 cell membranes assessed as inhibition of microbe growt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM25817(2-(2,4-difluorophenyl)-1,3-bis(1H-1,2,4-triazol-1-...)
Affinity DataIC50:  880nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Tulahuen CYP51 expressed in Escherichia coli JM109 cell membranes assessed as inhibition of microbe growt...More data for this Ligand-Target Pair
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510709(CHEMBL4571367)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510706(CHEMBL4515068)
Affinity DataIC50:  1.65E+4nMAssay Description:Non-competitive inhibition of Leishmania amazonensis arginase using L-arginine as substrate incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510706(CHEMBL4515068)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510711(CHEMBL4467463)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510708(CHEMBL4456185)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510712(CHEMBL4570250)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510710(CHEMBL4438412)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase(Leishmania amazonensis)
Instituto De Tecnologia Em Farmacos

Curated by ChEMBL
LigandPNGBDBM50510707(CHEMBL4541649)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant Leishmania amazonensis arginase expressed in Escherichia coli using L-arginine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM213825(VNI)
Affinity DataKd:  8.30nMAssay Description:Binding affinity to Trypanosoma cruzi Y CYP51A expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50276214(CHEMBL4129161)
Affinity DataKd:  4.20nMAssay Description:Binding affinity to Trypanosoma cruzi Y CYP51A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative lanosterol 14-alpha-demethylase(Leishmania infantum)
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50465949(CHEMBL4276822)
Affinity DataKd:  24nMAssay Description:Binding affinity to Leishmania infantum CYP51 expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50465948(CHEMBL3629567)
Affinity DataKd:  6.80nMAssay Description:Binding affinity to Trypanosoma cruzi Y CYP51A expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50465949(CHEMBL4276822)
Affinity DataKd:  8.40nMAssay Description:Binding affinity to Trypanosoma cruzi Y CYP51A expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPutative lanosterol 14-alpha-demethylase(Leishmania infantum)
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50465948(CHEMBL3629567)
Affinity DataKd:  8.40nMAssay Description:Binding affinity to Leishmania infantum CYP51 expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPutative lanosterol 14-alpha-demethylase(Leishmania infantum)
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM213825(VNI)
Affinity DataKd:  2nMAssay Description:Binding affinity to Leishmania infantum CYP51 expressed in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPutative lanosterol 14-alpha-demethylase(Leishmania infantum)
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50276214(CHEMBL4129161)
Affinity DataKd:  1.70nMAssay Description:Binding affinity to Leishmania infantum CYP51 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed