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Found 434 with Last Name = 'spadari' and Initial = 's'
TargetThymidine kinase(Human herpesvirus 2)
Glsynthesis

LigandPNGBDBM21885(2,9-disubstituted 6-oxopurine, 12i | 9-[4-(decahyd...)
Affinity DataKi:  5nM IC50:  13nMAssay Description:Recombinant HSV TKs were assayed in reaction mixture containing substrate [3H-methyl]TdR and test compounds. After reaction was stopped, the radioact...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102265(1-(5-Bromo-pyridin-2-yl)-3-[2-(6-fluoro-4-oxo-4H-p...)
Affinity DataKi:  9nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102271(1-(5-Bromo-pyridin-2-yl)-3-[2-(4-oxo-4H-5,9,9b-tri...)
Affinity DataKi:  9nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082061((+/-)-5-ethyl-5-(3-methoxy-phenyl)-6-oxa-10b-aza-b...)
Affinity DataKi:  10nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082061((+/-)-5-ethyl-5-(3-methoxy-phenyl)-6-oxa-10b-aza-b...)
Affinity DataKi:  11nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102265(1-(5-Bromo-pyridin-2-yl)-3-[2-(6-fluoro-4-oxo-4H-p...)
Affinity DataKi:  15nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102268(1-(5-Bromo-pyridin-2-yl)-3-[2-(5-oxo-pyrazolo[1,5-...)
Affinity DataKi:  15nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102276(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-chloro-4-oxo-4H-p...)
Affinity DataKi:  20nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102276(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-chloro-4-oxo-4H-p...)
Affinity DataKi:  20nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102268(1-(5-Bromo-pyridin-2-yl)-3-[2-(5-oxo-pyrazolo[1,5-...)
Affinity DataKi:  21nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082055(5-Ethyl-5-m-tolyl-6-oxa-10,10b-diaza-benzo[e]azule...)
Affinity DataKi:  21nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102277(1-(5-Bromo-pyridin-2-yl)-3-[2-(7,9-difluoro-4-oxo-...)
Affinity DataKi:  22nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082061((+/-)-5-ethyl-5-(3-methoxy-phenyl)-6-oxa-10b-aza-b...)
Affinity DataKi:  22nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082060(5-Ethyl-5-phenyl-6-oxa-10,10b-diaza-benzo[e]azulen...)
Affinity DataKi:  22nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102266(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-fluoro-4-oxo-4H-p...)
Affinity DataKi:  29nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102273(1-(5-Bromo-pyridin-2-yl)-3-[2-(6-fluoro-pyrrolo[1,...)
Affinity DataKi:  29nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1)
Glsynthesis

LigandPNGBDBM21885(2,9-disubstituted 6-oxopurine, 12i | 9-[4-(decahyd...)
Affinity DataKi:  30nM ΔG°:  -44.7kJ/mole IC50:  150nMpH: 7.5 T: 2°CAssay Description:Recombinant HSV TKs were assayed in reaction mixture containing substrate [3H-methyl]TdR and test compounds. After reaction was stopped, the radioact...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082062(5-Ethyl-5-thiophen-2-yl-6-oxa-10b-aza-benzo[e]azul...)
Affinity DataKi:  30nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102277(1-(5-Bromo-pyridin-2-yl)-3-[2-(7,9-difluoro-4-oxo-...)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082055(5-Ethyl-5-m-tolyl-6-oxa-10,10b-diaza-benzo[e]azule...)
Affinity DataKi:  30nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102266(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-fluoro-4-oxo-4H-p...)
Affinity DataKi:  40nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  40nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102270(1-(5-Bromo-pyridin-2-yl)-3-[2-(9-fluoro-4-oxo-4H-p...)
Affinity DataKi:  40nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082060(5-Ethyl-5-phenyl-6-oxa-10,10b-diaza-benzo[e]azulen...)
Affinity DataKi:  40nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082055(5-Ethyl-5-m-tolyl-6-oxa-10,10b-diaza-benzo[e]azule...)
Affinity DataKi:  44nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082056(5-Ethyl-5-thiophen-2-yl-6-oxa-10,10b-diaza-benzo[e...)
Affinity DataKi:  45nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
University Of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM21866(2-phenylamino-9-(4-hydroxybutyl)-6-oxopurine | 9-(...)
Affinity DataKi:  50nMAssay Description:Binding affinity of the compound towards HSV-1 thymidine kinase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102271(1-(5-Bromo-pyridin-2-yl)-3-[2-(4-oxo-4H-5,9,9b-tri...)
Affinity DataKi:  50nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102267(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-chloro-pyrrolo[1,...)
Affinity DataKi:  53nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102273(1-(5-Bromo-pyridin-2-yl)-3-[2-(6-fluoro-pyrrolo[1,...)
Affinity DataKi:  58nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102275(1-(5-Bromo-pyridin-2-yl)-3-[2-(4-oxo-4H-pyrrolo[1,...)
Affinity DataKi:  58nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102270(1-(5-Bromo-pyridin-2-yl)-3-[2-(9-fluoro-4-oxo-4H-p...)
Affinity DataKi:  60nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082061((+/-)-5-ethyl-5-(3-methoxy-phenyl)-6-oxa-10b-aza-b...)
Affinity DataKi:  60nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102267(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-chloro-pyrrolo[1,...)
Affinity DataKi:  70nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution V179DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082057((+/-)-5-ethyl-5-m-tolyl-6-oxa-10b-aza-benzo[e]azul...)
Affinity DataKi:  70nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082060(5-Ethyl-5-phenyl-6-oxa-10,10b-diaza-benzo[e]azulen...)
Affinity DataKi:  70nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082062(5-Ethyl-5-thiophen-2-yl-6-oxa-10b-aza-benzo[e]azul...)
Affinity DataKi:  70nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082059(5-Ethyl-5-(3-fluoro-phenyl)-6-oxa-10b-aza-benzo[e]...)
Affinity DataKi:  70nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082056(5-Ethyl-5-thiophen-2-yl-6-oxa-10,10b-diaza-benzo[e...)
Affinity DataKi:  90nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102267(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-chloro-pyrrolo[1,...)
Affinity DataKi:  90nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution Y181IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082056(5-Ethyl-5-thiophen-2-yl-6-oxa-10,10b-diaza-benzo[e...)
Affinity DataKi:  90nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082056(5-Ethyl-5-thiophen-2-yl-6-oxa-10,10b-diaza-benzo[e...)
Affinity DataKi:  93nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102271(1-(5-Bromo-pyridin-2-yl)-3-[2-(4-oxo-4H-5,9,9b-tri...)
Affinity DataKi:  95nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution L1001More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082057((+/-)-5-ethyl-5-m-tolyl-6-oxa-10b-aza-benzo[e]azul...)
Affinity DataKi:  100nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102268(1-(5-Bromo-pyridin-2-yl)-3-[2-(5-oxo-pyrazolo[1,5-...)
Affinity DataKi:  100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution L1001More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102277(1-(5-Bromo-pyridin-2-yl)-3-[2-(7,9-difluoro-4-oxo-...)
Affinity DataKi:  100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution L1001More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102275(1-(5-Bromo-pyridin-2-yl)-3-[2-(4-oxo-4H-pyrrolo[1,...)
Affinity DataKi:  100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution K103NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102267(1-(5-Bromo-pyridin-2-yl)-3-[2-(7-chloro-pyrrolo[1,...)
Affinity DataKi:  100nMAssay Description:Inhibition of HIV-1 Mutant HIV-1 RT enzymes containing the single amino acid substitution Y188LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082059(5-Ethyl-5-(3-fluoro-phenyl)-6-oxa-10b-aza-benzo[e]...)
Affinity DataKi:  100nMAssay Description:In vitro inhibitory activity against HIV-1 wild type reverse transcriptase (RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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