TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetMultidrug and toxin extrusion protein 1(Mus musculus)
Riken Center For Life Science Technologies
Curated by ChEMBL
Riken Center For Life Science Technologies
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Inhibition of mouse Mate1 transfected in HEK293 cells assessed as uptake of [14C]-TEA preincubated for 15 mins by liquid scintillation counting analy...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 238nMAssay Description:TP_TRANSPORTER: inhibition of Cerivastatin uptake in OATP2-expressing MDCKII cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 580nMAssay Description:TP_TRANSPORTER: inhibition of Taurocholate uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 910nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.01E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.03E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.46E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.62E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.91E+3nMAssay Description:TP_TRANSPORTER: inhibition of SN-38 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.96E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1C1(Mus musculus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 2.15E+3nMAssay Description:TP_TRANSPORTER: inhibition of L-T4 uptake in Oatp14-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 2.18E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 3(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.74E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Oat1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 2.87E+3nMAssay Description:TP_TRANSPORTER: inhibition of SN-38 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
Affinity DataKi: 3.09E+3nMAssay Description:TP_TRANSPORTER: inhibition of Pravastatin uptake in Oat3-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(Mus musculus)
Riken Center For Life Science Technologies
Curated by ChEMBL
Riken Center For Life Science Technologies
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Inhibition of mouse Oct1 transfected in HEK293 cells assessed as uptake of [14C]-TEA preincubated for 15 mins by liquid scintillation counting analys...More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 3.81E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 3.84E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
Affinity DataKi: 4.43E+3nMAssay Description:TP_TRANSPORTER: inhibition of PCG uptake in Oat3-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetABC-type glutathione-S-conjugate transporter(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 5.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in membrane vesicle from MRP3-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 7.95E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 8.32E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
Affinity DataKi: 9.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of PCG uptake in OAT3-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 9.27E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Rattus norvegicus)
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair