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Found 89 with Last Name = 'taramelli' and Initial = 'd'
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50323737(CHEMBL1213687 | N-((2S)-1-((2S)-6-amino-1-(4-(6-me...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of Plasmodium falciparum PLM2 using Lys-Glu-Phe-Val-Phe-NPhe-Ala-Leu-Lys as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200018((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  1nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50390636(CHEMBL2069615)
Affinity DataKi:  1.30nMAssay Description:Inhibition of Plasmodium falciparum PLM2 using Lys-Glu-Phe-Val-Phe-NPhe-Ala-Leu-Lys as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50390637(CHEMBL2069616)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Plasmodium falciparum PLM2 using Lys-Glu-Phe-Val-Phe-NPhe-Ala-Leu-Lys as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50390633(CHEMBL2069612)
Affinity DataKi:  2.30nMAssay Description:Inhibition of Plasmodium falciparum PLM2 using Lys-Glu-Phe-Val-Phe-NPhe-Ala-Leu-Lys as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50390635(CHEMBL2069614)
Affinity DataKi:  2.60nMAssay Description:Inhibition of Plasmodium falciparum PLM2 using Lys-Glu-Phe-Val-Phe-NPhe-Ala-Leu-Lys as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50390634(CHEMBL2069613)
Affinity DataKi:  3.80nMAssay Description:Inhibition of Plasmodium falciparum PLM2 using Lys-Glu-Phe-Val-Phe-NPhe-Ala-Leu-Lys as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200018((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200015((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  9.90nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200020((3S,4S)-4-((2S,3S)-2-(4-(4-((4-(6-methoxyquinolin-...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200015((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200019((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200017((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-amino-1-...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200021((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-(1-(4-(6-methoxyqu...)
Affinity DataKi:  12nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200019((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  17nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200014((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  26nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200017((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-amino-1-...)
Affinity DataKi:  33nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200023((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  58nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50146527((3S,4S)-N-butyl-3-hydroxy-6-methyl-4-((2S,3S)-3-me...)
Affinity DataKi:  59nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200014((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  74nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200020((3S,4S)-4-((2S,3S)-2-(4-(4-((4-(6-methoxyquinolin-...)
Affinity DataKi:  81nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200023((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  103nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50146524((S)-3-(S)-Hydroxy-4-{(S)-3-methyl-2-[2-(naphthalen...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50223627(CHEMBL3215350)
Affinity DataKi:  180nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200016((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-(tert-bu...)
Affinity DataKi:  230nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50200016((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-(tert-bu...)
Affinity DataKi:  403nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50146527((3S,4S)-N-butyl-3-hydroxy-6-methyl-4-((2S,3S)-3-me...)
Affinity DataKi:  727nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200021((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-(1-(4-(6-methoxyqu...)
Affinity DataKi:  765nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50343187(CHEMBL1773155 | N,N'-Bis(3-aminopropyl)-3,9-dimeth...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of clostridium botulinum Botulinum neurotoxin type A light chain at 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBotulinum neurotoxin type A(Clostridium botulinum)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50343188(CHEMBL1773156 | N,N'-Bis(2-aminoethyl)-3,9-dimethy...)
Affinity DataKi:  8.70E+3nMAssay Description:Inhibition of clostridium botulinum Botulinum neurotoxin type A light chain at 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50366912(CHEMBL1790774)
Affinity DataIC50:  0.590nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50366909(CHEMBL1790773)
Affinity DataIC50:  1.5nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50366908(CHEMBL1790772)
Affinity DataIC50:  9.60nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50399931(CHEMBL2181207)
Affinity DataIC50:  22nMAssay Description:Inhibition of human ERG expressed in rat after 2 to 3 days by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50146530((S)-2-[4-(4-{(S)-1-[(S)-1-((S)-2-Butylcarbamoyl-1-...)
Affinity DataIC50:  123nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50366910(CHEMBL1790776)
Affinity DataIC50:  135nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50390633(CHEMBL2069612)
Affinity DataIC50:  220nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50247629(CHEMBL453384 | N-(3-((tert-butylamino)methyl)-4-fl...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50390635(CHEMBL2069614)
Affinity DataIC50:  300nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50366911(CHEMBL1790775)
Affinity DataIC50:  396nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50390634(CHEMBL2069613)
Affinity DataIC50:  540nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Universit£

Curated by ChEMBL
LigandPNGBDBM50146528(6-Amino-2-(S)-amino-hexanoic acid [4-(6-methoxy-qu...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  2.67E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch plate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytochrome P450 2C8(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50041457(4-[(7-chloroquinolin-4-yl)amino]-2-[(diethylamino)...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human CYP2C8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

LigandPNGBDBM50462274(CHEMBL4246869)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of CaV1.2 channel in rat tail artery myocytes assessed as reduction in Ba2+ current at -50 mV holding potential by whole-cell patch-clamp ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50142038(CHEMBL3758349)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch plate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50142039(CHEMBL3758840)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch plate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50041457(4-[(7-chloroquinolin-4-yl)amino]-2-[(diethylamino)...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50056190(4-(7-Chloro-quinolin-4-ylamino)-2-ethylaminomethyl...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Liverpool

Curated by ChEMBL
LigandPNGBDBM50134931(5-(7-Chloro-quinolin-4-ylamino)-2-diethylaminometh...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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