Affinity DataKi: 0.600nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Reversible inhibition of wild-type human N-terminal GST-tagged EGFR cytoplasmic domain (669 to 1210 end amino acid residues) expressed in baculovirus...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Reversible inhibition of wild-type human N-terminal GST-tagged EGFR cytoplasmic domain (669 to 1210 end amino acid residues) expressed in baculovirus...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Binding affinity to 6xHis-taged MDM2 (unknown origin) expressed in Escherichia coli Gold (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Reversible inhibition of wild-type human N-terminal GST-tagged EGFR cytoplasmic domain (669 to 1210 end amino acid residues) expressed in baculovirus...More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:In vitro Binding affinity towards 5-hydroxytryptamine 3 receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 153nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 183nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 205nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 212nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of bovine brain MAOB using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:Inhibition of cloned isozyme, human carbonic anhydrase IIMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of bovine brain MAOB using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 569nMAssay Description:Inhibition of human LSD1/CoREST using histone H3 peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 680nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 690nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of bovine brain MAOA using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 1.18E+3nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of bovine brain MAOB using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of bovine brain MAOB using kynuramine as a substrate after 30 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 2.79E+3nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 2.93E+3nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 3.13E+3nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 3.26E+3nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 3.94E+3nMAssay Description:Inhibition of G9a (unknown origin) assessed as reduction in substrate methylation using histone H3 and SAM as substrate measured after 15 to 60 mins ...More data for this Ligand-Target Pair