TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Inhibition of active BACE1 (unknown origin)More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Inhibition of human recombinant BACE1 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 2 hrs by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibition of active BACE1 (unknown origin)More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Inhibition of human recombinant BACE1 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 2 hrs by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Inhibition of human recombinant BACE1 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 2 hrs by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Inhibition of human recombinant BACE1 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 2 hrs by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Inhibition of human recombinant BACE1 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 2 hrs by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 2(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Apparent inhibition of human recombinant BACE2 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 1 hr by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 2(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Apparent inhibition of human recombinant BACE2 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 1 hr by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Inhibition of pro-BACE1 (unknown origin)More data for this Ligand-Target Pair
TargetBeta-secretase 2(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Apparent inhibition of human recombinant BACE2 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 1 hr by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 2(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Apparent inhibition of human recombinant BACE2 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 1 hr by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetBeta-secretase 2(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Instituto De Biologia Experimental E Tecnol£Gica
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Apparent inhibition of human recombinant BACE2 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 1 hr by HPLC-FLU analysisMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataIC50: 5.75E+4nMAssay Description:Antagonist activity at Vibrio harveyi MM32 LuxP receptor assessed as decrease in receptor agonist DPD-induced bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataIC50: 1.60E+5nMAssay Description:Antagonist activity at Vibrio harveyi MM32 LuxP receptor assessed as decrease in receptor agonist DPD-induced bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataIC50: 1.69E+5nMAssay Description:Antagonist activity at Vibrio harveyi MM32 LuxP receptor assessed as decrease in receptor agonist DPD-induced bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 3.00E+4nMAssay Description:Agonist activity at Vibrio harveyi LuxP receptorMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 1.95E+4nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 650nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 2.65E+4nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 6.21E+3nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 1.16E+4nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 1.87E+3nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 3.00E+4nMAssay Description:Agonist activity at Vibrio harveyi LuxP receptorMore data for this Ligand-Target Pair
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Instituto De Tecnologia Qu£Mica E Biol£Gica
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair