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Found 2134 with Last Name = 'white' and Initial = 's'
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | GWTLNSAGYLLGPQQFFGLM-CONH2 | Galani...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307256(CHEMBL604373 | GWTLNSAGYLLGPrPKPQQwFwLL-CONH2 | Ga...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307255(CHEMBL592413 | GWTLNSAGYLLGPRHYINLITRQRY-CONH2)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273353((S)-1-(2-((S)-2-((S)-2-((S)-2-(2-((S)-2-((S)-2-((S...)
Affinity DataKi:  0.400nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293023((Sar)WTLNSAGYLLGPKKKK | CHEMBL508036)
Affinity DataKi:  0.400nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataKi:  0.430nMAssay Description:Antagonist activity at human P2Y14 expressed in CHO cells assessed as inhibition of forskolin-induced increase of cAMP accumulation incubated for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293024((Sar)WTLNSAGYLLGPKK(Lys-MPEG4)K | CHEMBL505299)
Affinity DataKi:  0.5nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273351(CHEMBL508083 | GWTLNSAGYLLGPHAV-NH2)
Affinity DataKi:  0.5nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307256(CHEMBL604373 | GWTLNSAGYLLGPrPKPQQwFwLL-CONH2 | Ga...)
Affinity DataKi:  0.600nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293030((Sar)WTLNSAGYLLGPKK(Lys-octanoyl)K | CHEMBL503900)
Affinity DataKi:  0.700nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214688(1-{4-[(1R)-2-(amino-3-methylbutyl)-6-fluorophenyl]...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214682(1-{4-[(1S)-2-(1-amino-3-methylbutyl)-4-trifluorome...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  0.900nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273359(CHEMBL526500)
Affinity DataKi:  0.900nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214704(1-{4-[(1S)-2-(amino-3-methylbutyl)-4-fluorophenyl]...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | GWTLNSAGYLLGPQQFFGLM-CONH2 | Galani...)
Affinity DataKi:  1.10nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293029((Sar)WTLNSAGYLLGPKK(Lys-decanoyl)K | CHEMBL460706)
Affinity DataKi:  1.30nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307255(CHEMBL592413 | GWTLNSAGYLLGPRHYINLITRQRY-CONH2)
Affinity DataKi:  1.40nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293028((Sar)WTLNSAGYLLGPKK(Lys-lauroyl)K | CHEMBL507733)
Affinity DataKi:  1.40nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  1.5nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307252(CHEMBL578710 | WTLNSAGYLL-CONH2)
Affinity DataKi:  1.70nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50198702((E)-3-((6-methylpyridin-2-yl)ethynyl)cyclohex-2-en...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]ABP688 from human mGluR5 receptor expressed in L (tk-) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307258(CHEMBL578317 | [N-Ac,des-Sar]Gal-B2)
Affinity DataKi:  1.70nMAssay Description:Displacement of Eu-labeled galanin from human GalR1 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  1.80nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214689(1-{4-[(1S)-2-(1-amino-3-methylbutyl)-4-trifluorome...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50198702((E)-3-((6-methylpyridin-2-yl)ethynyl)cyclohex-2-en...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]ABP688 from mGluR5 in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214695(1-{4-[(1S)-2-(1-amino-3-methylbutyl)-4-trifluorome...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273354(CHEMBL525755)
Affinity DataKi:  1.90nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052588((2E,4E,6Z)-7-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]-Targretin binding to Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052588((2E,4E,6Z)-7-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]-Targretin binding to Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214703(1-{4-[(1R)-2-(amino-3-methylbutyl)-6-fluorophenyl]...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214679(1-{4-[(1S)-2-(amino-3-methylbutyl)-6-trifluorometh...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293027((Sar)WTLNSAGYLLGPKK(Lys-myristoyl)K | CHEMBL524678)
Affinity DataKi:  2.60nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273360((S)-N-((S)-6-amino-1-((S)-6-amino-1-((S)-1-((S)-1,...)
Affinity DataKi:  2.80nMAssay Description:Displacement of Eu-labeled galanin from human GalR1 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273362(CHEMBL505336)
Affinity DataKi:  3.30nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214691(1-{4-[(1S)-2-(1-amino-3-methylbutyl)-6-trifluorome...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214700(1-{4-[(1S)-2-(1-amino-3-methylbutyl)-6-fluoropheny...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50273355(CHEMBL525023)
Affinity DataKi:  3.5nMAssay Description:Displacement of europium-labeled galanin from human GalR1 expressed in HEK293 EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307250(CHEMBL578514 | GalB2)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50307250(CHEMBL578514 | GalB2)
Affinity DataKi:  3.5nMAssay Description:Displacement of Eu-labeled galanin from human GalR1 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293026((Sar)WTLNSAGYLLGPKK(Lys-palmitoyl)K | CHEMBL507353)
Affinity DataKi:  3.5nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50198702((E)-3-((6-methylpyridin-2-yl)ethynyl)cyclohex-2-en...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]M-MPEP from human mGluR5 receptor expressed in L (tk-) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052588((2E,4E,6Z)-7-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]-Targretin binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50293025((Sar)WTLNSAGYLLGPKK(Lys-stearoyl)K | CHEMBL450827)
Affinity DataKi:  4nMAssay Description:Displacement of europium labeled galanin from human recombinant GalR1 receptor by time-resolved fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052590((2E,4E,6Z)-7-(3-Ethoxy-5,5,8,8-tetramethyl-5,6,7,8...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]-Targretin binding to Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214696(1-((R)-1-(4-(2-((S)-1-amino-3-methylbutyl)-4-(trif...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214681(1-[(R)-2-{4-[(1S)-2-(1-amino-3-methylbutyl)-4-trif...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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