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Found 127 with Last Name = 'wikström' and Initial = 'hv'
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50123626((S)-6-[Propyl-(2-thiophen-2-yl-ethyl)-amino]-5,6,7...)
Affinity DataKi:  0.0600nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 expressed in CHO K1 cells was measured by its ability to displace [3H]- N-0437More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115642((+)-65-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro-2,...)
Affinity DataKi:  0.160nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2C receptor was determined using [3H]-mesulergineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115279(4-Propyl-3,4,4a,5,6,10b-hexahydro-2H-naphtho[1,2-b...)
Affinity DataKi:  0.210nMAssay Description:In vitro binding affinity at human Dopamine receptor D3 expressed in CHO K1 cells was measured by its ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115643((+/-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro...)
Affinity DataKi:  0.210nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2C receptor was determined using [3H]-mesulergineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115640((-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro-2...)
Affinity DataKi:  0.390nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2C receptor was determined using [3H]-mesulergineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115642((+)-65-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro-2,...)
Affinity DataKi:  0.550nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2A receptor was determined using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50054067((2R)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen...)
Affinity DataKi:  0.570nMAssay Description:In vitro binding affinity at human Dopamine receptor D3 expressed in CHO K1 cells was measured by its ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115643((+/-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro...)
Affinity DataKi:  0.700nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2A receptor was determined using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115640((-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro-2...)
Affinity DataKi:  0.75nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2A receptor was determined using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154716((-)-1-Methyl-4-(8-methylsulfanyl-10,11-dihydro-dib...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50098551((R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolid...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM31005(2-methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyraz...)
Affinity DataKi:  1.40nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2C receptor was determined using [3H]-mesulergineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM31005(2-methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyraz...)
Affinity DataKi:  1.5nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2A receptor was determined using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115644((+/-)-12-Methyl-1,2,3,4,9,13b-hexahydro-2,4a,5-tri...)
Affinity DataKi:  2nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2A receptor was determined using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115641((+/-)-7-2-Methyl-1,2,3,4,9,13b-hexahydro-2,4a-diaz...)
Affinity DataKi:  2nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2C receptor was determined using [3H]-mesulergineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50123627((S)-6-Dipropylamino-5,6,7,8-tetrahydro-naphthalene...)
Affinity DataKi:  2nMAssay Description:Binding affinity of compound for Dopamine receptor D2 using [3H]-N-0437More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50123627((S)-6-Dipropylamino-5,6,7,8-tetrahydro-naphthalene...)
Affinity DataKi:  3nMAssay Description:Binding affinity of compound for Dopamine receptor D1 using [3H]-SCH- 23390More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026553((+)-6-Dipropylamino-5,6,7,8-tetrahydro-naphthalene...)
Affinity DataKi:  3nMAssay Description:In vitro binding affinity of the compound towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50130279((R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidi...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50123626((S)-6-[Propyl-(2-thiophen-2-yl-ethyl)-amino]-5,6,7...)
Affinity DataKi:  4nMAssay Description:In vitro binding affinity at human Dopamine receptor D3 expressed in CHO K1 cells was measured by its ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154714((5R,6R)-5-Methyl-6-((R)-6-methyl-5,6,6a,7-tetrahyd...)
Affinity DataKi:  4nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115644((+/-)-12-Methyl-1,2,3,4,9,13b-hexahydro-2,4a,5-tri...)
Affinity DataKi:  5.5nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2C receptor was determined using [3H]-mesulergineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50123625((S)-6-[Propyl-(2-thiophen-2-yl-ethyl)-amino]-5,6,7...)
Affinity DataKi:  6nMAssay Description:Binding affinity of compound for Dopamine receptor D2 using [3H]-N-0437More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115279(4-Propyl-3,4,4a,5,6,10b-hexahydro-2H-naphtho[1,2-b...)
Affinity DataKi:  6.24nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 expressed in CHO K1 cells was measured by its ability to displace [3H]- N-0437More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50130278((R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-pyrr...)
Affinity DataKi:  10nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154706(CHEMBL187764 | N-Ethyl-N-[3-(6-methoxy-3,4-dihydro...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115283(2-Phenyl-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-naph...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity at human Dopamine receptor D3 expressed in CHO K1 cells was measured by its ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115641((+/-)-7-2-Methyl-1,2,3,4,9,13b-hexahydro-2,4a-diaz...)
Affinity DataKi:  12nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 2A receptor was determined using [3H]-ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50123626((S)-6-[Propyl-(2-thiophen-2-yl-ethyl)-amino]-5,6,7...)
Affinity DataKi:  15nMAssay Description:Binding affinity of compound for Dopamine receptor D2 using [3H]-N-0437More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115644((+/-)-12-Methyl-1,2,3,4,9,13b-hexahydro-2,4a,5-tri...)
Affinity DataKi: >18nMAssay Description:The binding affinity of the compound at the 5-hydroxytryptamine 1A receptor determined using [3H]-5-CTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154711(CHEMBL364124 | N-Ethyl-N-{3-[4-(2-methoxy-phenyl)-...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154712(CHEMBL184310 | N-Ethyl-4-methoxy-N-[3-(6-methoxy-3...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115282(CHEMBL103622 | Dipropyl-(4,5,6,7-tetrahydro-benzo[...)
Affinity DataKi:  20nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 expressed in CHO K1 cells was measured by its ability to displace [3H]- N-0437More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115644((+/-)-12-Methyl-1,2,3,4,9,13b-hexahydro-2,4a,5-tri...)
Affinity DataKi: >20nMAssay Description:The binding affinity of the compound at the Dopamine receptor D3 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115640((-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro-2...)
Affinity DataKi:  20nMAssay Description:The binding affinity of the compound at the Dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154707((1R,6S)-5-Methyl-6-((S)-6-methyl-5,6,6a,7-tetrahyd...)
Affinity DataKi:  21nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115644((+/-)-12-Methyl-1,2,3,4,9,13b-hexahydro-2,4a,5-tri...)
Affinity DataKi: >25nMAssay Description:The binding affinity of the compound at the Dopamine receptor D4 determined using [3H]-YM-09151-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115275(CHEMBL103857 | Dipropyl-(4,5,6,7-tetrahydro-benzo[...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 expressed in CHO K1 cells was measured by its ability to displace [3H]- N-0437More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115275(CHEMBL103857 | Dipropyl-(4,5,6,7-tetrahydro-benzo[...)
Affinity DataKi:  28nMAssay Description:In vitro binding affinity at human Dopamine receptor D3 expressed in CHO K1 cells was measured by its ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115643((+/-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro...)
Affinity DataKi:  28nMAssay Description:The binding affinity of the compound at the Dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50054067((2R)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen...)
Affinity DataKi:  34nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 expressed in CHO K1 cells was measured by its ability to displace [3H]- N-0437More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115282(CHEMBL103622 | Dipropyl-(4,5,6,7-tetrahydro-benzo[...)
Affinity DataKi:  40nMAssay Description:In vitro binding affinity at human Dopamine receptor D3 expressed in CHO K1 cells was measured by its ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115640((-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro-2...)
Affinity DataKi:  47nMAssay Description:The binding affinity of the compound at the Dopamine receptor D4 determined using [3H]-YM-09151-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154718(CHEMBL185762 | N-{3-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  52nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154710(CHEMBL188876 | N-Ethyl-N-[3-(6-methoxy-3,4-dihydro...)
Affinity DataKi:  54nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50115280(CHEMBL103912 | Dipropyl-(4,5,6,7-tetrahydro-benzo[...)
Affinity DataKi:  60nMAssay Description:In vitro binding affinity at human Dopamine receptor D3 expressed in CHO K1 cells was measured by its ability to displace [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM31005(2-methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyraz...)
Affinity DataKi:  70nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 3 receptor was determined using [3H]-LY-278,584More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154708(CHEMBL364795 | N-[3-(6-Methoxy-3,4-dihydro-1H-isoq...)
Affinity DataKi:  75nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
State University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50154703(CHEMBL187088 | N-{2-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  75nMAssay Description:Binding affinity towards rat 5-HT7 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University Center For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50115640((-)-6 5-Methoxy-2-methyl-1,2,3,4,9,13b-hexahydro-2...)
Affinity DataKi:  80nMAssay Description:The binding affinity of the compound at 5-hydroxytryptamine 1D receptor was determined using [3H]-5-CTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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