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Found 64 with Last Name = 'yoshioka' and Initial = 'y'
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13152((2S)-1-[(2S)-2-[(2S)-2-aminobutanamido]-3-methylbu...)
Affinity DataKi:  24nM ΔG°:  -43.1kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13151((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  28nM ΔG°:  -42.7kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13155((2S)-1-[(2S)-2-[(2S)-2-aminobutanamido]-3-methylbu...)
Affinity DataKi:  81nM ΔG°:  -40.1kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13150((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  150nM ΔG°:  -38.6kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13148((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  180nM ΔG°:  -38.1kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13147((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  220nM ΔG°:  -37.6kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13142((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  290nM ΔG°:  -36.9kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  930nMAssay Description:Binding affinity to recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  1.07E+3nMAssay Description:Binding affinity to full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13153((2S)-2-amino-N-[(2S)-3-methyl-1-oxo-1-[(2R)-2-(3-p...)
Affinity DataKi:  1.20E+3nM ΔG°:  -33.5kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13146((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  1.27E+3nM ΔG°:  -33.3kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13156((2S)-1-[(2S)-2-[(2S)-2-amino-3-methylbutanamido]-3...)
Affinity DataKi:  4.15E+3nM ΔG°:  -30.4kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13145((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  4.41E+3nM ΔG°:  -30.3kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13149((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  4.90E+3nM ΔG°:  -30.0kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  1.25E+4nMAssay Description:Competitive inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13143((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  1.34E+4nM ΔG°:  -27.5kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13144((2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]-3-methylb...)
Affinity DataKi:  2.45E+4nM ΔG°:  -26.1kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13157((2S)-1-[(2S)-2-[(2S)-2-aminopentanamido]-3-methylb...)
Affinity DataKi:  5.40E+4nM ΔG°:  -24.1kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Michigan

LigandPNGBDBM13154((2S)-1-[(2S)-2-(2-aminoacetamido)-3-methylbutanoyl...)
Affinity DataKi:  6.80E+4nM ΔG°:  -23.5kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  75nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50367841(CHEMBL1788193)
Affinity DataIC50:  84nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50405738(CHEMBL2093039)
Affinity DataIC50:  91nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020324(4-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  92nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020321(2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  94nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020318(2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  96nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020337(4-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  100nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020328(2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  110nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020325(2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020340(2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  410nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020327(2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-prop...)
Affinity DataIC50:  670nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020332(CHEMBL158254 | {2-[(2-Acetoxy-3-octadecyloxy-propo...)
Affinity DataIC50:  880nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020330(1-{2-[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-pr...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020329(CHEMBL158489 | {2-[Acetyl-(2-methoxy-3-octadecylca...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 4(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human USP4 using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536673(CHEMBL4587307)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020333(CHEMBL160653 | {2-[Butyryl-(2-methoxy-3-octadecylc...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536673(CHEMBL4587307)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536672(CHEMBL2012939)
Affinity DataIC50:  2.71E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of UCH-L1 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of USP5 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable ubiquitin carboxyl-terminal hydrolase FAF-X(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of USP9x in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536672(CHEMBL2012939)
Affinity DataIC50:  3.76E+3nMAssay Description:Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50536674(CHEMBL4593579)
Affinity DataIC50:  3.79E+3nMAssay Description:Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437694(CHEMBL1410015)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human USP14More data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020319(1-{2-[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-pr...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020320(CHEMBL160910 | {2-[(2-Methoxy-3-octadecylcarbamoyl...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50020322(CHEMBL350437 | {2-[Butyryl-(2-methoxy-3-octadecylc...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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