BindingDB PrimarySearch_ki

Found 195 with Last Name = 'zahid' and Initial = 'h'

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584413(CHEMBL5084290)

IC50: 12nMAssay Description:Inhibition of His9-tagged BRD4-BD1 (unknown origin) using Ac-SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRKVLR-Peg-(Biot) as substrate incubated for 1 hr and m...More data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573200(CHEMBL4861491)

IC50: 36nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 51nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573201(CHEMBL4848701)

IC50: 56nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573197(CHEMBL4872300)

IC50: 67nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 72nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) by fluorescence anisotropy methodMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 77nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by fluorescence anisotropy methodMore data for this Ligand-Target Pair

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Bromodomain-containing protein 3(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: <80nMAssay Description:Inhibition of BRD3 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584414(CHEMBL5087797)

IC50: <92nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584418(CHEMBL5082732)

IC50: <92nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584393(CHEMBL5085236)

IC50: <92nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584400(CHEMBL5075050)

IC50: <92nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584412(CHEMBL5085224)

IC50: <92nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584403(CHEMBL5078890)

IC50: <92nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: <92nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 94nMAssay Description:Inhibition of BRD4 D2 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 3(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 96nMAssay Description:Inhibition of BRD3 D2 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584408(CHEMBL5086716)

IC50: 100nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584399(CHEMBL5089270)

IC50: 110nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584416(CHEMBL5090760)

IC50: 110nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 2(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 120nMAssay Description:Inhibition of BRD2 D2 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain testis-specific protein(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 120nMAssay Description:Inhibition of BRDT D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50582040(CHEMBL5083660)

IC50: 137nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by fluorescence anisotropy methodMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 2(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 140nMAssay Description:Inhibition of BRD2 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573198(CHEMBL4848138)

IC50: 170nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584395(CHEMBL5088918)

IC50: 190nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584392(CHEMBL5081513)

IC50: 200nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584393(CHEMBL5085236)

IC50: 200nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584398(CHEMBL5079869)

IC50: 200nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50234940(CHEMBL4101756)

IC50: 220nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573192(CHEMBL4850516)

IC50: 250nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584410(CHEMBL5082969)

IC50: 260nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584402(CHEMBL5087306)

IC50: 270nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 2(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584413(CHEMBL5084290)

IC50: 280nMAssay Description:Inhibition of BRD2-BD1 (unknown origin) measured by AlphaScreen assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573190(CHEMBL4866748)

IC50: 290nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584413(CHEMBL5084290)

IC50: 300nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584390(CHEMBL5085763)

IC50: 310nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573191(CHEMBL4870218)

IC50: 310nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584411(CHEMBL5084552)

IC50: 360nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573193(CHEMBL4848082)

IC50: 370nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573203(CHEMBL4863631)

IC50: 380nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584401(CHEMBL5091410)

IC50: 430nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584420(CHEMBL5079566)

IC50: 440nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584392(CHEMBL5081513)

IC50: 440nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584397(CHEMBL5080722)

IC50: 500nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573202(CHEMBL4877696)

IC50: 550nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584391(CHEMBL5085543)

IC50: 610nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by competitive fluorescence anisotropy assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50584390(CHEMBL5085763)

IC50: 640nMAssay Description:Inhibition of BRD4 D1 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair

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Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50573188(CHEMBL4850913)

IC50: 700nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair

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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL

PNG

BDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)

IC50: 720nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) by fluorescence anisotropy methodMore data for this Ligand-Target Pair

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3D Structure (crystal)

Displayed 1 to 50 (of 195 total ) | Next | Last >>

Filter my 195 hits

Targets 11▿
- Bromodomain-containing protein 4 125
- Nucleosome-remodeling factor subunit BPTF 32
- Bromodomain-containing protein 2 9
- Bromodomain-containing protein 3 8
- Mitogen-activated protein kinase 14 8
- Histone acetyltransferase KAT2B 4
- Bromodomain testis-specific protein 3
- Bromodomain-containing protein 9 3
- Histone acetyltransferase KAT2A 1
- Bromodomain-containing protein 7 1
- Chromatin remodeling regulator CECR2 1
- ...
Publications 4▿
- J Med Chem 64: 10497-10511 (2021) 76
- J Med Chem 65: 2342-2360 (2022) 65
- J Med Chem 64: 13902-13917 (2021) 47
- ACS Med Chem Lett 13: 1621-1627 (2022) 7
Institutions 1▿
- University Of Minnesota 195
Affinity: 0.24 to 1.2E+5 nM▿
- IC50 146
- Kd 49
- Affinity ≤ nM
Xtal structures: 21
Docked structures: 0
Catalog Cmpds: 14