Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 279 hits in this display
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 20nMAssay Description:Inhibition of [3H]- quinuclidinyl benzilate binding to human Muscarinic acetylcholine receptor M2 expressed in CHO cell membraneMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 20nMAssay Description:Inhibition of binding of [3H]quinuclidinyl benzilate to Muscarinic acetylcholine receptor M2 in rat cerebral cortical membranesMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 31nMAssay Description:Affinity versus [3H]oxotremorine M (agonist) binding to Muscarinic acetylcholine receptor M1 in Rat Cerebral Cortical Membranes, (Kd=0.75 nM)More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 37nMAssay Description:Binding affinity of [3H](R)-QNB binding to Muscarinic acetylcholine receptor M1 expressed in A9 L cell line in the presence of 300 uM GTP-gamma-SMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 210nMAssay Description:Binding affinity towards rat Nicotinic acetylcholine receptor alpha3-beta2 expressed in HEK293 cells using [3H]EB as radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 590nMAssay Description:Binding affinity towards rat Nicotinic acetylcholine receptor alpha4-beta2 expressed in HEK293 cells using [3H]EB as radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.10E+3nMAssay Description:Binding affinity towards rat Nicotinic acetylcholine receptor alpha4-beta4 expressed in HEK293 cells using [3H]EB as radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.23E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor transfected in CHO cells after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.23E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.30E+3nMAssay Description:Binding affinity of compound was determined towards human Muscarinic acetylcholine receptor M2 using [3H]-QNB radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.30E+3nMAssay Description:Binding affinity towards rat nicotinic acetylcholine receptor alpha2-beta2 expressed in HEK293 cells using [3H]EB as radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.60E+3nMAssay Description:Inhibition of binding of [3H]quinuclidinyl benzilate to Muscarinic acetylcholine receptor M4 in rat cerebral cortical membranesMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 4.30E+3nMAssay Description:Binding affinity of compound was determined towards human Muscarinic acetylcholine receptor M5 using [3H]-QNB radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 4.80E+3nMAssay Description:Binding affinity towards rat Nicotinic acetylcholine receptor alpha3-beta4 expressed in HEK293 cells using [3H]EB as radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 6.31E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 6.31E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor transfected in CHO cells after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 7.60E+3nMAssay Description:Binding affinity of compound was determined towards human Muscarinic acetylcholine receptor M4 using [3H]-QNB radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 8.20E+3nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 8.20E+3nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.20E+4nMAssay Description:Binding affinity of compound was determined towards human Muscarinic acetylcholine receptor M1 using [3H]-QNB radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.26E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.37E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.46E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.70E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.82E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.85E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.93E+4nMAssay Description:In brief, membranes from COS-7 cells expressing different Cys-substituted mutant M3R constructs were first treated with CuPhen (100 μM; 10 min a...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.95E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.97E+4nMAssay Description:In brief, membranes from COS-7 cells expressing different Cys-substituted mutant M3R constructs were first treated with CuPhen (100 μM; 10 min a...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.00E+4nMAssay Description:Binding affinity of compound was determined towards human Muscarinic acetylcholine receptor M3 using [3H]-QNB radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.04E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.20E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.38E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.46E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.79E+4nMAssay Description:In brief, membranes from COS-7 cells expressing different Cys-substituted mutant M3R constructs were first treated with CuPhen (100 μM; 10 min a...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 2.95E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 3.32E+4nMAssay Description:In brief, membranes from COS-7 cells expressing different Cys-substituted mutant M3R constructs were first treated with CuPhen (100 μM; 10 min a...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 3.80E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 3.80E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor transfected in CHO cells after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 4.13E+4nMpH: 7.4Assay Description:In brief, binding reactions containing ~10 μg of membrane protein per tube were carried out for 2 h (22 °C) in 1 ml of binding buffer containing...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 4.13E+4nMAssay Description:In brief, membranes from COS-7 cells expressing different Cys-substituted mutant M3R constructs were first treated with CuPhen (100 μM; 10 min a...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 4.37E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 4.37E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor transfected in CHO cells after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 6.92E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor transfected in CHO cells after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 6.92E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation countingMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Ki: 1.60E+5nMAssay Description:Binding activity to muscarinic acetylcholine receptor in rat heart, assayed using [3H]QNB as a radioligand in the presence of Gpp(NH)p.More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 6.70nMAssay Description:Binding affinity towards muscarinic receptor using [3H]cis-methyldioxolane (CMD) to label agonist sites in membrane preparations from rat neocortexMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 6.70nMAssay Description:Compound was evaluated for inhibition of [3H]cis-methyldioxolane binding to label agonist sites (RCMD) in rat neocortexMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 6.70nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 17nMAssay Description:Ability to displace [3H]cis--2-methyl-5-((dimethylamino)methyl)-1,3-di oxolane from muscarinic acetylcholine receptor in rat cortical tissue.More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 23nMAssay Description:In vitro binding affinity against Muscarinic acetylcholine receptor M1 from rat hippocampus, using [3H]-oxotremorine-M (Oxo-M) as radioligand.More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 130nMAssay Description:Inhibitory activity against [3H]quinuclidinyl Benzilate binding to Muscarinic acetylcholine receptor M2 in the absence of GTPMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 130nMAssay Description:Inhibition of binding of 0.1 nM [3H]quinuclidinyl benzilate to Muscarinic acetylcholine receptor M2 in rat cerebral cortical membranes of transfected...More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 230nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 1.38E+3nMAssay Description:In vitro binding affinity against muscarinic acetylcholine receptor M1 from rat hippocampus, using [3H]-pirenzepine (Pz) as radioligandMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 3.10E+3nMAssay Description:Inhibitory activity against [3H]quinuclidinyl Benzilate binding to Muscarinic acetylcholine receptor M2 in the presence of GTPMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
IC50: 1.89E+4nMAssay Description:Compound was evaluated for the displacement of the muscarinic QNB in rat heart homogenate containing the pharmacologic M2 receptor (M2-QNB heart)More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 700nMAssay Description:Compound was tested for its potency towards Muscarinic acetylcholine receptor M2 by inhibiting forskolin induced c-AMP formation in CHO-M2 cellsMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 4.60E+3nMAssay Description:Stimulation of phosphoinositol hydrolysis in the mouse fibroblast cell line A9L-M1 expressing Muscarinic acetylcholine receptor M1.More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 1.50E+4nMAssay Description:Agonist activity at human M3 receptor in HEK293 cells assessed as induction of calcium response by fluorescence assayMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 1.07E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 74nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M2 determined by receptor selection and amplification technology (R-SAT).More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 360nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 1.80E+3nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M3 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 75nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M4 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 6.10E+4nMAssay Description:Reversal of forskolin-stimulated accumulation of adenylate cyclase in transfected CHO cells, against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
EC50: 6.00E+4nMAssay Description:Reversal of forskolin-stimulated accumulation of adenylate cyclase in transfected CHO cells, against Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
BDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
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