Compound (290)
Article Title (2)
Article Author (139)
BDBM50015082 Ser-Asn-CH=CH-Val-Phe-Ala-NH-Bzl CHEMBL367080
Ser-Asn-Val-CH=CH-Phe-Ala-O-Bzl CHEMBL366854 BDBM50015062
BDBM31887 Ch 80 BMS181156
BDBM50525572 CHEMBL1743245 CH-223191
US10106501, Example CH BDBM293207
BDBM483514 US10927076, Compound Table2.CH(OH)CH3
US10774085, Example 11 US8865698, 11 US10047097, 11 US11267818, Example 11 BDBM136594 US10005783, 11 US9676783, 11
US10968213, Example 11 US9920047, 11 US10053456, 11 US9487511, 11 US10414761, Example 11 BDBM256632 US9718814, 11
US10765676, Example 11 US9763943, 11 BDBM249321 US10300060, Example 11 US9993479, 11 US9463192, 11
BDBM143188 US9994576, 11 US9266895, 11 US11040980, Example 11 US8940744, 11
US9227975, 11 US10011604, 11 BDBM200583 US10590139, Example 11 US9795611, 11
US10967060, Example 11 US20240173303, Example 11 US9320732, 11 BDBM223009 US11207302, Example 11 US9789094, 11 US10034939, Example 11
US9102686, 11 BDBM174780 US9540388, 11 US10053462, 11
US9695149, 11 US8952177, 11 US9089569, 11 BDBM145657
US9820989, 11 US9388176, 11 BDBM139551 US8889870, 11
US10028934, Compound 11 US10478423, Cpd. 11 US9408850, 11 US9597317, 11 BDBM239017
US9694016, 11 US10709712, Example 11 US9242969, 11 BDBM202666 US10245267, Example 11
US9802939, 11 US8940720, 11 BDBM142860 US10487086, Example 11 US11136327, Example 11
BDBM161226 US10087143, Compound 11 US11673864, Compound 11 US9051270, 11 US10738009, Compound 11 US9758483, Compound 11
BDBM164817 US10604504, Example 11 US11623921, Example 11 US9688629, 11 US9920031, Example 11 US9802915, Example 11
US9586962, Example 11 US11059828, Example 11 US11667644, Example 11 USRE48841, Example 11 BDBM118358 US8653263, 11
BDBM391513 US10472358, Example 11 US10781209, Example 11 US11059821, Example 11 US11702416, Example 11 US12227502, Example 11 US9957268, Example 11
US10526330, Example 11 BDBM292114 US11299492, Example 11 US10100049, Example 11 US10183942, Example 11 US11718616, Example 11 US10913740, Example 11
BDBM257473 US9493441, 11-11
11 BDBM50598559 Compound 11 AFTOBETIN ANCA11 ANCA-11
BDBM150337 US8987249, 11 US10238633, Example 11 US9713606, 11
BDBM150704 US9526727, 11 US8981112, 11 US9949975, Example 11
US10092556, Example 11 BDBM155567 US9012475, 11 US9346787, 11
US10640503, Example 11 US10047086, 11 BDBM103897 US9695168, 11
US9227969, 11 US9629836, 11 US10011599, Example 11 BDBM200383
US9708313, 11 US9181249, 11 US10077266, Example 11 BDBM190900
US10632171, Peptide No. 11 US10179804, Example 11 BDBM135626 US8846601, 11 US9458201, 11
US10941151, Compound 11 BDBM251913 US9475814, 11 US10683295, Compound 11 US10065961, Compound 11
US11512066, Example 11 US10167273, Example 11 BDBM250532 US10544126, Example 11 US9475795, 11
US11673868, Example 11 US11180460, Example 11 US10457647, Example 11 US9512084, 11 BDBM259412
US20240043404, Example 11 US11369599, Compound 11 US9174982, 11 BDBM189465 US10213433, Compound 11
US9314464, 11 US10568884, Cpd 11 USRE49556, Compound 11 US9593100, Compound 11 BDBM221690
US9796729, 11 BDBM321144 US10174049, Example 11 US10385066, Example 11 US9738658, Example 11
US10035797, Compound 11 US11560377, Compound 11 BDBM279672 US9630965, Compound 11 US10428068, Compound 11 US10844056, Compound 11
US10689414, Compound 11 US10717764, Compound 11 US11021515, Compound 11 BDBM363519 US9850277, Compound 11 US10640534, Compound 11
US10881652, Example 11 US10441581, Example 11 US10172845, Example 11 US11648243, Example 11 BDBM304995 US10144734, Example 11
US9802924, Entry 11 BDBM352207 US10287274, Entry 11 US10239868, Entry 11 US10676464, Entry 11 US20240425487, Entry 11
US9422299, 11 US20240199618, Compound 11 US10836768, Cpd no 11 BDBM50112245 US9987274, Compound 11 US10030025, Compound 11 US11731974, Compound 11 CHEMBL3608741
CHEMBL386023 BDBM50159394 Des-AA1,2,5-[D-Trp8,IAmp9]SRIF CH-275
US11583516, Cmpd ID 4175CH US11096924, DASH-inhibitors 4175 CH BDBM514516
BDBM103746 US8551978, I-11 US9572802, Compound I-11 US9394275, I-11 US8816088, I-11 US9682957, I-11
BDBM340019 US11541059, Compound 11 US10329299, Compound 11 US9775844, Compound 11 US10675286, Compound 11
BDBM370361 US10233189, Example 11 US10787457, Example 11 US11014930, Example 11 US11236096, Example 11
US11161855, Example 11 US10370387, Example 11 US9777017, Example 11 BDBM344027 US9908895, Example 11
US11535614, Compound 11 BDBM317858 US9624217, Compound 11 US10807980, Compound 11 US10399976, Compound 11
US11608338, Example 11 US10745399, Example 11 BDBM418443 US10975075, Example 11 US10457677, Example 11
US11634410, Example 11 US10787438, Example 11 US10174007, Example 11 US10988463, Example 11 BDBM319592
US9675614, 11 BDBM176830 US10391089, Compound 11 US10980794, Cmpd No 11 US10307413, Compound 11
US9796724, Example 11 US10251889, Example 11 US9782415, Example 11 BDBM344302 US10758542, Example 11
US9975907, Example 11 US10829502, Example 11 BDBM394292 US10428087, Example 11 US11401280, Example 11
US9981975, Example 11 US10844069, Example 11 BDBM396949 US10442810, Example 11 US11591338, Example 11
BDBM153694 US9610299, Example 11 US10507215, Compound 11 US9000015, 11
BDBM155365 US10918640, Example 11 US10383871, Example 11 US9006269, 11
BDBM173259 US9604982, Example 11 US9096596, 11 US10323032, Example 11
BDBM185195 US10011588, Example 11 US9156829, 11 US10689373, Example 11
BDBM207566 US9617273, Example 11 US10501467, Example 11 US9260440, 11
BDBM241169 US10479788, Example 11 US9409907, 11 US11046688, Example 11
BDBM246106 US10183932, Example 11 US9822102, Example 11 US9434690, 11
BDBM265047 US9718793, 11 US11234987, Example 11 US10413550, Example 11
Method #11 US11607396, Example 11 US11071721, Example 11 BDBM508766
US10023562, Example 11 US10544133, Example 11 BDBM283817 US9657009, 11
US10080750, Compound 11 BDBM224334 US9662330, Compound 11 US9321760, 11
US10112931, Example 11 US9434719, 11 US9688672, Example 11 BDBM247488
US10125133, Example 11 US10968221, Example 11 BDBM103884 US9695167, 11
US10329256, Example 11 US9487512, 11 US9944601, Example 11 BDBM256466
US10329300, Example 11 US11696917, Example 11 BDBM376917 US9920060, 11
US10501411, Example 11 US11697636, Example 11 US9452980, 11 BDBM250101
US10683287, Example 11 US10035794, Example 11 BDBM116236 US8637508, 11
US11254644, Compound 11 US10513499, Compound 11 US9708272, 11 BDBM261588
US8551988, 11 US10736881, Compound 11 BDBM103541 US10201527, Compound 11
US9447106, 11 US10005782, Compound 11 US9556188, Compound 11 BDBM249884
US9527851, example 11 US9527851, 11 US10428074, Example 11 BDBM260455
US9540373, 11 US9879026, Example 11 BDBM201022 USRE47636, Example 11
US9744173, Example 11 BDBM223324 US9605007, Example 11 US9315520, 11
US9884878, Compound 11 US9745328, Compound 11 US9079866, 11 BDBM168638
US9918985, Example 11 US8865911, 11 US10231967, Example 11 BDBM136921
US10765676, Example 23-11 US9463192, 23-11 BDBM249354 US9763943, 23-11 US10300060, Example 23-11 US9993479, 23-11
BDBM110543 US8614234, 11 US9725433, 11
BDBM119328 US8673906, 11 US9718800, 11
BDBM125050 US8772511, 11 US9714242, 11
BDBM156388 US9248140, 11 US9018381, 11
BDBM160344 US9040714, 11 US9693992, 11
BDBM160597 US9045468, 11(+) US9045468, 11(-)
BDBM164978 US9682971, 11 US9067917, 11
BDBM185601 US9493431, 11 US9156856, 11
BDBM234458 US9353084, 11 US10004738, 11
BDBM254928 US9499542, 11 US9675594, 11
BDBM504390 US11040970, Compound 11-11
US10016420, 11 BDBM209590 US9273011, 11
US10047092, 11 US9040534, 11 BDBM160070
US10047103, 11 US9688695, 11 BDBM175978
US10080744, Example 11/11 BDBM285800
US10759813, Example 11-11 BDBM459244
US8541408, 11 BDBM100988 US8507479, 11
US8613914, 11 US9206232, 11 BDBM110243
US8921389, 11 US9695170 11 BDBM141555
US8952157, 11 BDBM144829 US9303025, 11
US8987335, 11 BDBM151610 US9555024, 11
US9024044, 11 US9227949, 11 BDBM158083
US9034899, 11 BDBM159329 US9604960, 11
US9073869, 11 BDBM138500 US8877775, 11
US9120752, 11 BDBM176468 US9765029, 11
US9120769, 11 BDBM177587 US9663470, 11
US9169243, 11 US9908875, 11 BDBM187363
US9259470, 11 US8697715, 11 BDBM120090
US9290459, 11 BDBM211759 US9670166, 11
US9365529, 11 US8633196, 11 BDBM113583
US9597333, 11 US9475775, 11 BDBM254744
US9611251, 11 US9115117, 11 BDBM175109
US9630945, 11 US9409895, 11 BDBM241100
US9694018, 11 BDBM77080 US10093697, 11.
US9732066, 11 BDBM197412 US9216968, 11
US9822074, 11 BDBM235188 US9365558, 11
US9918969, 11 US9475809, 11 BDBM251899
US10980815, Ex. No. 11 US9663526, Example 11 US10463675, Example 11 US11197867, Example 11 BDBM329928
US10053465, 11 US11992490, Compound 11 US11084822, Example 11 US11304949, Compound 11 US10479803, Example 11 US10065963, Compound 11 US11957661, Compound 11 US20240307353, Compound 11 US10519163, Example 11 US11324749, Comp. No. 11 US20240058343, Compound 11 US11406640, Comp. No. 11 US10675284, Example 11 US11136326, Example 11 US10336759, # 11 {trans-3-(4-{[4-[(3- hydroxyazetidin-1- yl)methyl]-6- (trifluoromethyl) pyridin-2- yl]oxy}piperidin-1- yl)-1-[4-(7H- pyrrolo[2,3- d]pyrimidin-4-yl)- 1H-pyrazol-1- yl]cydobutyl} acetonitrile US10125150, Example 11 US12268667, Compound 11 US11130767, # 11 US12226418, Example 11 US11918581, Compound 11 US11596632, Comp. No. 11 US9732097, Example 11 BDBM246872
US9951048, Compound 11 US10544128, Compound 11 US11548872, Compound 11 US20230286945, Compound 11 US10604514, Compound 9 US10106527, Compound 11 BDBM293425
BDBM244402 US9428502, 11 US20250017938, Compound 002-11 US10226449, cpd 11
BDBM281485 US9586949, Example 11 US10022387, Example 11 US10596184, Example 11
BDBM314698 US10513522, Example 11 US11214573, Example 11 US9611269, Example 11
BDBM331879 US10927120, Compound 11 US10189849, Compound 11 US9957276, Compound 11
BDBM458537 US12180213, Example 11 US10745401, Example 11 US11466007, Example 11
US10077273, Compound 11 US10584132, Compound 11 BDBM285663 US10934305, Compound 11
US10266491, Example 11 US11053197, Example 11 BDBM377343 US10676434, Example 11
US10392376, Example 11 BDBM411438 US10800769, Example 11 US11434233, Example 11
US10442803, Example 11 BDBM343412 US11091484, Example 11 US9777003, Example 11
US10675268, Example 11 US9789082, Example 11 US10166214, Example 11 BDBM311875
US10793579, Example 11 BDBM402861 US10329302, Example 11 US11702424, Example 11
US10800783, Example 11 US10233188, Example 11 US11396512, Example 11 BDBM370122
US10875867, Example 11 US10023575, Example 11 US10479794, Example 11 BDBM284720
US10934296, Example 11 US10239883, Example 11 US9758524, Example 11 BDBM340084
US11130754, Example 11 US12139484, Example 11 BDBM303827 US10138241, Example 11
US11236095, Example 11 US9492453, 11 BDBM50427336 CHEMBL2325992 US10654855, Example 11
US11332464, Compound 11 BDBM397440 US10676470, Compound 11 US9988375, Compound 11
US11479538, Example 11 BDBM211296 US10093650, Example 11 US10329273, Example 11
US11547695, Compound 11 US10517849, Compound 11 US11013718, Compound 11 BDBM424915
US11608330, Example 11 US10995088, Example 11 US10807974, Example 11 BDBM468988
US11701371, Compound 11 US11707471, Compound 11 BDBM608786 US20230277570, Compound 11
US9745310, Example 11 US11046702, Example 11 BDBM292156 US10100057, Example 11
BDBM50194237 CHEMBL377960 H-Dmt-Tic-NH-CH[(CH2)4-NH2]-Bid
Des-AA1,5-[Tyr2,D-Trp8,IAmp9]SRIF CH-288 BDBM50159431 CHEMBL411002
H-Dmt-Tic-NH-(R)CH(CH2-COOH)-Bid CHEMBL444197 BDBM50272229
BDBM111159 US10556908, Example 11 US9695180, 11
BDBM145232 US8952169, 11 US9771376, Example 11
BDBM166925 US9073876, 11 US9732093, Compound 11
BDBM181168 US9783501, Compound 11 US9139529, 11
BDBM200749 US9233108, 11 US9757383, Example 11
BDBM232930 US9346839, 11 US9738668, Compound 11
BDBM236780 US9388149, 11 US9580412, Example 11
BDBM239111 US9403810, 11 US10195181, Example 11
BDBM258537 US10633384, Example 11 US9493486, 11
BDBM260825 US9540323, 11 US9540323, example 11
BDBM308060 US9650366, 11 US10011593, Ex. 11
BDBM323622 US10188653, Example 11 US9789110, 11
BDBM578768 US11479550, Example 11-11(2)
Method #11 US10947226, Example 11 BDBM486464
US10000475, Compound 11 BDBM177782 US9120786, 11
US10017516, Compound 11 BDBM143311 US9682983, 11
US10023561, Example 11 BDBM148454 US9682965, 11
US10188642, Example 11 US9334286, 11 BDBM230885
US10195186, Example 11 US9682967, 11 BDBM159123
US10233178, Example 11 BDBM261744 US9708309, 11
US10280160, Example 11. BDBM160519 US9682969, 11
US10336717, Compound 11 BDBM113233 US8633212, 11
US20240025908, Example 11 BDBM647643 T-11
US9051313, 11 BDBM162320 US10307427, Compound 11
US9073922, 11 US9796708, Example 11 BDBM167527
US9163003, 11 USRE46942, Example 11 BDBM185803
US9200016, 11 BDBM194329 US9902710, Compound 11
US9221828, 11 BDBM50043873 US9174993, 11 CHEMBL3356059
US9346815, 11 US9604984, Example 11 BDBM232465
US9422293, 11 US9738649, Example 11 BDBM244806
US9464060, 11 US10100018, Example 11 BDBM251675
US9505745, 11 BDBM259334 US9790212, Example 11
US9512114, 11 BDBM259451 US9657007, Example 11
US9611222, Example 11 BDBM162392 US9056832, 11
US9650377, Example 11 US8853203, 11 BDBM135957
US9656968, Compound 11 US9163008, 11 BDBM185922
US9682966, 11 BDBM155024 US10118915, Compound 11
US9718820, Compound 11 US9409915, 11 BDBM241619
US9738632, Example 11 US8916600, 11 BDBM141377
US9744252, Example 11 US9345793, 11 BDBM228630
US9771375, Example 11 BDBM130548 US8822447, 11
US9896444, Example 11 BDBM230757 US9340537, 11
US9902741, Example 11 US9718822, 11 BDBM267419
US9951071, Example 11 BDBM241379 US9409908, 11
BDBM445673 US10683309, Example 11 Ex. 11/KM-06-91/(I-11)
US11123311, Compound 11 US10377744, Compound No. 11 BDBM408990 US11723929, Compound 11
US11230523, Compound 11 US11648234, Compound 11 BDBM50529667 US10806720, Compound 11 CHEMBL4444904
US11247972, Compound 11 BDBM50389685 US10544104, Compound 11 CHEMBL2070052 US9765037, Compound 11
US8614253, 3-11 US9963434, Compound 3-11 US9241942, 3-11 BDBM110980
US10774052, Compound I-11 BDBM88648 US10618902, Compound I-11 US10189794, Compound I-11 US9695132, I-11
US10793564, Compound 11 US20230293519, Compound 16 US20230271960, Compound 11 US11419869, Compound 11 BDBM465222 US11560376, Compound 11
BDBM277475 US11780852, Example 2-11 US12358931, Example 2-11 US10947254, Example 2-11 US10072026, Example 2-11
BDBM277520 US10947254, Example 4-11 US12358931, Example 4-11 US10072026, Example 4-11 US11780852, Example 4-11
US10072026, Example 6-11 BDBM277592 US10947254, Example 6-11 US12358931, Example 6-11 US11780852, Example 6-11
US12358931, Example 1-11 BDBM277417 US10072026, Example 1-11 US10947254, Example 1-11 US11780852, Example 1-11
US9987276, Compound I-11 US11351168, Compound I-11 BDBM397293 US10828300, Compound I-11 US10596172, Compound I-11
US10179769, Example 11 3-{[4-(propan-2-yloxy)benzyl]amino}pyridine-4-carboxylic acid BDBM314107 US10807956, Example 11 US11214542, Example 11 US9828343, Example 11 US11639333, Example 11 US9611221, Example 11 US9725441, Example 11
BDBM209470 US10328074, Example III-11 US9266891, III-11 US11077107, Example III-11
US10392392, Example 8-11 US10047093, 8-11 BDBM228294 US10875864, EX. 8-11
US10434101, Compound I-11 BDBM149411 US8975249, I-11 US11096942, Compound I-11
US9238629, I-11 US9765038, Compound I-11 US10081606, Compound I-11 BDBM202379
BDBM50194238 CHEMBL386309 H-Dmt-Tic-NH-CH[(CH2)4-NH-Z]-Bid
Benzyoxycarbonyl-Asn-Phe-[S]-[CH(OH)CH2N]Pro-Otert-butyl BDBM50010502 CHEMBL115292
CHEMBL268205 Des-AA1,2,5-[D-Trp8,IAmp9,Tyr11]SRIF [Tyr11]CH-275 BDBM50159420
H-Dmt-Tic-NH-CH[(CH2)4-NH-Ac]-Bid CHEMBL378082 BDBM50194242
BDBM111436 US8614253, 42-11 US9241942, 42-11
BDBM147507 US8962608, 11-5 US8962608, 11-3
BDBM232962 US9353113, 11(12) US9862721, 11(12)
BDBM232963 US9353113, 11(24) US9862721, 11(24)
BDBM261488 US10011568, Ex. No. 11 US9708266, 11
BDBM289101 US11014909, Example 11 US9107923, 11 BDBM160922
BDBM303502 US10875852, Example 11 US10138229, Example 11
BDBM345834 US10202365, Compound 11 US10774070, Compound 11
BDBM360324 US9828348, Compound 11 US9975858, Compound 11
BDBM362444 US9834564, Compound 11 US10562916, Compound 11
BDBM364329 US10570156, Compound 11 US9856274, Compound 11
BDBM375945 US9914735, Example 11 US10947243, Example 11
BDBM377029 US10259818, Example 11 US9944646, Example 11
BDBM382195 US10273259, Example 11 US10711020, Example 11
BDBM393700 US10597367, Example 11 US9969726, Example 11
BDBM397939 US10604536, Compound 11 US9994590, Compound 11
BDBM410194 US11059827, Compound 11 US10370379, Compound 11
BDBM412272 US10399945, Example 11 US10927079, Compound 11
BDBM421420 US10995073, Example 11 US10508086, Example 11
BDBM434089 US11008308, Example 11 US10562891, Example 11
BDBM448069 US11319326, Compound 11 US10689390, Compound 11
BDBM448207 US10689401, EX 11 US11008338, Example 11
BDBM448538 US10696655, Example 11 US11168070, Example 11
BDBM450247 US11117861, Example 11 US10676431, Example 11
BDBM461303 US10774065, Example 11 US11401259, Example 11
BDBM461305 US11427560, Example 11 US10774068, Example 11
BDBM466555 US11014905, Example 11 US10800755, Example 11
BDBM466692 US11731958, Example 11 US10800761, Example 11
BDBM470586 US11369605, Example 11 US10815241, Example 11
BDBM50427476 US10308662, Compound 11 US9505780, 11 CHEMBL2322247
BDBM536104 US11891388, Example 11 US11242343, Example 11
BDBM578169 US11478474, Compound 11 US12070457, Compound 11
BDBM97380 Orexin receptor antagonist 11 US20130102619, 11
US10071974, Example 11 BDBM275900 US10577336, Example 11
US10155002, Compound 11 BDBM514152 US9090562, 11 BDBM172007
US10221195, Example 11 BDBM275069 US9879032, Example 11
US10259811, Example 11 US10072001, Example 11 BDBM276825
US10287278, Example 11 US10647706, Example 11 BDBM385549
US10336721, Example 11 US10968198, Example 11 BDBM403755
US10351575, Example 11 BDBM406057 US10889589, EX. # 11
US10399989, Example 11 BDBM412795 US10611766, Example 11
US10584135, Example 11 US10273244, Example 11 BDBM382179
US10590114, No. 11 US11111235, No. 11 BDBM436219
US10597366, Compound 11 US9896418, Compound 11 BDBM372972
US10632122, Example 11 US10307425, Example 11 BDBM416545
US10702498, Compound 11 BDBM449090 US11484525, Compound 11
US10793567, Compound 11 US11225479, Compound 11 BDBM465376
US10800739, Compound (11) BDBM466534 US11420940, cpd (11)
US10807986, Example 11 BDBM469360 US11046696, Compound 11
US10822345, Ex 11 US10399991, Example 11 BDBM412894
US10851080, Example 11 BDBM373063 US9896435, Example 11
US10888567, Compound 11 US20250186410, Compound 11 BDBM477116
US10934288, Example 11 BDBM414593 US10435405, Example 11
US11001561, Compound 11 BDBM497015 US11702392, Compound 11
US11001583, Compound 11 BDBM329655 US9663515, Compound 11
US11014911, Example 11 BDBM498183 US11718603, Example 11
US11014929, Example 11 US11542265, Example 11 BDBM498971
US11168090, Example 11 US11851434, Example 11 BDBM524569
US11352361, Example 11 US11680068, Example 11 BDBM557352
US11390631, Example 11 BDBM561469 US12268694, Example 11
US11414404, Ex. # 11 US11634409, Example 11 BDBM565134
US11504381, Compound 11 US11548866, Compound 11 BDBM581328
US11591316, Compound 11 US9932325, Example 11 BDBM384307
US11655249, Example 11 BDBM500330 US11021478, Example 11
US11691950, Example 11 BDBM511467 US11059789, Example 11
US11911372, Example 11 BDBM653590 US20240277683, Example 11
US12195427, Compound 11 US11584714, Compound 11 BDBM594031
US20240300954, Entry 11 US10961249, Entry 11 BDBM489600
US20240327430, Example 11 BDBM699172 US12145945, Example 11
US20250066388, Example 11 BDBM669469 US11964990, Example 11
US8614253, 26-11 BDBM111224 US9241942, 26-11
US8614253, 43-11 BDBM111251 US9241942, 27-11
US8871790, 11 BDBM136959 US20250017938, Compound 001-11
US8962608, 11-10 US8962608, 11-9 BDBM147513
US9241942, 29-11 US8614253, 29-11 BDBM111351
US9624228, Example 11 US10301317, Example 11 BDBM318055
US9745291, Compound 11 BDBM336965 US9765068, Compound 11
US9833448, Example 11 US10272077, Example 11 BDBM362173
Pierce, AC; ter Haar, E; Binch, HM; Kay, DP; Patel, SR; Li, P CH...O and CH...N hydrogen bonds in ligand design: a novel quinazolin-4-ylthiazol-2-ylamine protein kinase inhibitor. J Med Chem 48: 1278 -81 (2005)
Herrero, S; Suarez-Gea, M; Gonzalez-Muniz, R; Garcia-Lopez, M; Herranz, R; Ballaz, S; Barber, A; Fortuno, A; Del Rio, J Pseudopeptide CCK-4 analogues incorporating the [CH(CN)NH] peptide bond surrogate Bioorg Med Chem Lett 7: 855 -860 (1997)
van Niel, MB; Wilson, K; Adkins, CH; Atack, JR; Castro, JL; Clarke, DE; Fletcher, S; Gerhard, U; Mackey, MM; Malpas, S; Maubach, K; Newman, R; O'Connor, D; Pillai, GV; Simpson, PB; Thomas, SR; MacLeod, AM J Med Chem 48: 6004 -11 (2005)
Chung, SC; Jang, KH; Park, J; Ahn, CH; Shin, J; Oh, KB Bioorg Med Chem Lett 21: 1958 -61 (2011)
Pippione, AC; Sainas, S; Goyal, P; Fritzson, I; Cassiano, GC; Giraudo, A; Giorgis, M; Tavella, TA; Bagnati, R; Rolando, B; Caing-Carlsson, R; Costa, FTM; Andrade, CH; Al-Karadaghi, S; Boschi, D; Friemann, R; Lolli, ML Eur J Med Chem 163: 266 -280 (2019)
Bromberg, KD; Mitchell, TR; Upadhyay, AK; Jakob, CG; Jhala, MA; Comess, KM; Lasko, LM; Li, C; Tuzon, CT; Dai, Y; Li, F; Eram, MS; Nuber, A; Soni, NB; Manaves, V; Algire, MA; Sweis, RF; Torrent, M; Schotta, G; Sun, C; Michaelides, MR; Shoemaker, AR; Arrowsmith, CH; Brown, PJ; Santhakumar, V; Martin, A; Rice, JC; Chiang, GG; Vedadi, M; Barsyte-Lovejoy, D; Pappano, WN Nat Chem Biol 13: 317 -324 (2017)
Belvisi, MG; Bundschuh, DS; Stoeck, M; Wicks, S; Underwood, S; Battram, CH; Haddad, el-B; Webber, SE; Foster, ML J Pharmacol Exp Ther 314: 568 -74 (2005)
Foloppe, N; Allen, NH; Bentley, CH; Brooks, TD; Kennett, G; Knight, AR; Leonardi, S; Misra, A; Monck, NJ; Sellwood, DM Bioorg Med Chem Lett 18: 1199 -206 (2008)
Stehouwer, JS; Bourke, CH; Owens, MJ; Voll, RJ; Kilts, CD; Goodman, MM Bioorg Med Chem Lett 25: 5111 -4 (2015)
JEONG, J; SHIN, HK; AHN, SJ; LIM, HJ; SONG, JS; KIM, SH; CHAE, CH; KIM, EH; CHOI, JH; LIM, JS; JANG, ES; SONG, JW; KIM, DH US Patent US20250145625 (2025)
Self, CR; Barber, WE; Machin, PJ; Osbond, JM; Smithen, CE; Tong, BP; Wickens, JC; Bloxham, DP; Bradshaw, D; Cashin, CH J Med Chem 34: 772 -7 (1991)
Yun, CS; Kim, HR; Cho, SY; Jung, HJ; Lee, K; Chae, CH; Lee, CO; Park, CH; Kim, P; Hwang, JY; Ha, JD; Ahn, SJ US Patent US10053458 (2018)
Mahindroo, N; Huang, CF; Peng, YH; Wang, CC; Liao, CC; Lien, TW; Chittimalla, SK; Huang, WJ; Chai, CH; Prakash, E; Chen, CP; Hsu, TA; Peng, CH; Lu, IL; Lee, LH; Chang, YW; Chen, WC; Chou, YC; Chen, CT; Goparaju, CM; Chen, YS; Lan, SJ; Yu, MC; Chen, X; Chao, YS; Wu, SY; Hsieh, HP J Med Chem 48: 8194 -208 (2005)
Chern, JW; Tao, PL; Yen, MH; Lu, GY; Shiau, CY; Lai, YJ; Chien, SL; Chan, CH J Med Chem 36: 2196 -207 (1993)
Rodgers, JD; Johnson, BL; Wang, H; Erickson-Viitanen, S; Klabe, RM; Bacheler, L; Cordova, BC; Chang, CH Bioorg Med Chem Lett 8: 715 -20 (1999)
Shi, LS; Chao, CH; Shen, DY; Chan, HH; Chen, CH; Liao, YR; Wu, SJ; Leu, YL; Shen, YC; Kuo, YH; Lee, EJ; Qian, K; Wu, TS; Lee, KH Bioorg Med Chem 19: 677 -83 (2011)
Goey, AK; Chau, CH; Sissung, TM; Cook, KM; Venzon, DJ; Castro, A; Ransom, TR; Henrich, CJ; McKee, TC; McMahon, JB; Grkovic, T; Cadelis, MM; Copp, BR; Gustafson, KR; Figg, WD J Nat Prod 79: 1267 -75 (2016)
Lin, SY; Chang Hsu, Y; Peng, YH; Ke, YY; Lin, WH; Sun, HY; Shiao, HY; Kuo, FM; Chen, PY; Lien, TW; Chen, CH; Chu, CY; Wang, SY; Yeh, KC; Chen, CP; Hsu, TA; Wu, SY; Yeh, TK; Chen, CT; Hsieh, HP J Med Chem 62: 10108 -10123 (2019)
Yu, Z; Fong, WP; Cheng, CH Drug Metab Dispos 35: 981 -6 (2007)
Tsai, TY; Hsu, T; Chen, CT; Cheng, JH; Yeh, TK; Chen, X; Huang, CY; Chang, CN; Yeh, KC; Hsieh, SH; Chien, CH; Chang, YW; Huang, CH; Huang, YW; Huang, CL; Wu, SH; Wang, MH; Lu, CT; Chao, YS; Jiaang, WT Bioorg Med Chem 17: 2388 -99 (2009)
Li, MC; Lai, YL; Kuo, PH; Reddy, JS; Chen, CM; Manimala, J; Wang, PC; Wu, MS; Chang, CY; Yang, CM; Lin, CY; Huang, YC; Chiu, CH; Chang, L; Lin, WH; Yeh, TK; Yen, WC; Hsieh, HP J Med Chem 67: 10906 -10927
Scott, SA; Spencer, CT; O'Reilly, MC; Brown, KA; Lavieri, RR; Cho, CH; Jung, DI; Larock, RC; Brown, HA; Lindsley, CW ACS Chem Biol 10: 421 -32 (2015)
Choi, CH; Kim, JH; Kim, SH Biochem Biophys Res Commun 320: 672 -9 (2004)
Chou, CH; Gong, CL; Chao, CC; Lin, CH; Kwan, CY; Hsieh, CL; Leung, YM J Nat Prod 72: 830 -4 (2010)
Chu, CH; Wang, LY; Hsu, KC; Chen, CC; Cheng, HH; Wang, SM; Wu, CM; Chen, TJ; Li, LT; Liu, R; Hung, CL; Yang, JM; Kung, HJ; Wang, WC J Med Chem 57: 5975 -85 (2014)
Liu, B; Croy, CH; Hitchcock, SA; Allen, JR; Rao, Z; Evans, D; Bures, MG; McKinzie, DL; Watt, ML; Stuart Gregory, G; Hansen, MM; Hoogestraat, PJ; Jamison, JA; Okha-Mokube, FM; Stratford, RE; Turner, W; Bymaster, F; Felder, CC Bioorg Med Chem Lett 25: 4158 -63 (2015)
Suman, P; Murthy, TR; Rajkumar, K; Srikanth, D; Dayakar, Ch; Kishor, C; Addlagatta, A; Kalivendi, SV; Raju, BC Eur J Med Chem 90: 603 -19 (2015)
Dreas, A; Kucwaj-Brysz, K; Pyziak, K; Kulesza, U; Wincza, E; Fabritius, CH; Michalik, K; Gabor-Worwa, E; Gołas, A; Milik, M; Masiejczyk, M; Majewska, E; Pyśniak, K; Wójcik-Trechcińska, U; Sandowska-Markiewicz, Z; Brzózka, K; Ostrowski, J; Rzymski, T; Mikula, M Eur J Med Chem 213: (2021)
Fournet, A; Inchausti, A; Yaluff, G; Rojas De Arias, A; Guinaudeau, H; Bruneton, J; Breidenbach, MA; Karplus, PA; Faerman, CH J Enzym Inhib 13: 1 -9 (1998)
Chorvat, RJ; Bakthavatchalam, R; Beck, JP; Gilligan, PJ; Wilde, RG; Cocuzza, AJ; Hobbs, FW; Cheeseman, RS; Curry, M; Rescinito, JP; Krenitsky, P; Chidester, D; Yarem, JA; Klaczkiewicz, JD; Hodge, CN; Aldrich, PE; Wasserman, ZR; Fernandez, CH; Zaczek, R; Fitzgerald, LW; Huang, SM; Shen, HL; Wong, YN; Chien, BM; Arvanitis, A J Med Chem 42: 833 -48 (1999)
Wehn, PM; Harrington, PE; Carlson, TJ; Davis, J; Deprez, P; Fotsch, CH; Grillo, MP; Lu, JY; Morony, S; Pattabiraman, K; Poon, SF; Reagan, JD; St Jean, DJ; Temal, T; Wang, M; Yang, Y; Henley, C; Lively, SE Bioorg Med Chem Lett 23: 6625 -8 (2013)
Borsari, C; Jiménez-Antón, MD; Eick, J; Bifeld, E; Torrado, JJ; Olías-Molero, AI; Corral, MJ; Santarem, N; Baptista, C; Severi, L; Gul, S; Wolf, M; Kuzikov, M; Ellinger, B; Reinshagen, J; Witt, G; Linciano, P; Tait, A; Costantino, L; Luciani, R; Tejera Nevado, P; Zander-Dinse, D; Franco, CH; Ferrari, S; Moraes, CB; Cordeiro-da-Silva, A; Ponterini, G; Clos, J; Alunda, JM; Costi, MP Eur J Med Chem 183: (2019)
Stoermer, MJ; Chappell, KJ; Liebscher, S; Jensen, CM; Gan, CH; Gupta, PK; Xu, WJ; Young, PR; Fairlie, DP J Med Chem 51: 5714 -21 (2008)
Maolanon, AR; Villadsen, JS; Christensen, NJ; Hoeck, C; Friis, T; Harris, P; Gotfredsen, CH; Fristrup, P; Olsen, CA J Med Chem 57: 9644 -57 (2014)
Francis, S; Croft, D; Schüttelkopf, AW; Parry, C; Pugliese, A; Cameron, K; Claydon, S; Drysdale, M; Gardner, C; Gohlke, A; Goodwin, G; Gray, CH; Konczal, J; McDonald, L; Mezna, M; Pannifer, A; Paul, NR; Machesky, L; McKinnon, H; Bower, J Bioorg Med Chem Lett 29: 1023 -1029 (2019)
Charifson, PS; Grillot, AL; Grossman, TH; Parsons, JD; Badia, M; Bellon, S; Deininger, DD; Drumm, JE; Gross, CH; LeTiran, A; Liao, Y; Mani, N; Nicolau, DP; Perola, E; Ronkin, S; Shannon, D; Swenson, LL; Tang, Q; Tessier, PR; Tian, SK; Trudeau, M; Wang, T; Wei, Y; Zhang, H; Stamos, D J Med Chem 51: 5243 -63 (2008)
Zhou, J; Yu, LZ; Fan, YL; Guo, CH; Lv, XM; Zhou, ZY; Huang, HD; Miao, DD; Zhang, SP; Li, XY; Zhao, PP; Liu, XP; Hu, WH; Zhang, C Eur J Med Chem 245: (2023)
Coumar, MS; Chang, CN; Chen, CT; Chen, X; Chien, CH; Tsai, TY; Cheng, JH; Wu, HY; Han, CH; Wu, SH; Huang, YW; Hsu, T; Hsu, LJ; Chao, YS; Hsieh, HP; Jiaang, WT Bioorg Med Chem Lett 17: 1274 -9 (2007)
Sun, T; Zhen, T; Harakandi, CH; Wang, L; Guo, H; Chen, Y; Sun, H Eur J Med Chem 275:
Heathcock, CH; Hadley, CR; Rosen, T; Theisen, PD; Hecker, SJ J Med Chem 30: 1858 -73 (1987)
Davis, PD; Elliott, LH; Harris, W; Hill, CH; Hurst, SA; Keech, E; Kumar, MK; Lawton, G; Nixon, JS; Wilkinson, SE J Med Chem 35: 994 -1001 (1992)
Hyup, YH; Kwan, JK; Kang, SH; Noh, MS; Ha, JY; Kyu, JK; Min, KM; Hoon, CH; Chung, S Bioorg Med Chem Lett 13: 413 -7 (2003)
Hsiao, SH; Lu, YJ; Yang, CC; Tuo, WC; Li, YQ; Huang, YH; Hsieh, CH; Hung, TH; Wu, CP J Nat Prod 79: 2135 -42 (2016)
Qiao, JX; Hu, CH; Thibeault, C US Patent US9120798 (2015)
Chen, CS; Tan, CM; Huang, CH; Chang, LC; Wang, JP; Cheng, FC; Chern, JW Bioorg Med Chem 18: 597 -604 (2010)
Zhang, ML; Irwin, D; Li, XN; Sauriol, F; Shi, XW; Wang, YF; Huo, CH; Li, LG; Gu, YC; Shi, QW J Nat Prod 75: 2076 -81 (2012)
Wu, Y; Karna, S; Choi, CH; Tong, M; Tai, HH; Na, DH; Jang, CH; Cho, H J Med Chem 54: 5260 -4 (2011)
Kim, SH; Anilkumar, GN; Zawacki, LG; Zeng, Q; Yang, DY; Shao, Y; Dong, G; Xu, X; Yu, W; Jiang, Y; Jenh, CH; Hall, JW; Carroll, CD; Hobbs, DW; Baldwin, JJ; McGuinness, BF; Rosenblum, SB; Kozlowski, JA; Shankar, BB; Shih, NY Bioorg Med Chem Lett 21: 6982 -6 (2011)
Krall, J; Bavo, F; Falk-Petersen, CB; Jensen, CH; Nielsen, JO; Tian, Y; Anglani, V; Kongstad, KT; Piilgaard, L; Nielsen, B; Gloriam, DE; Kehler, J; Jensen, AA; Harpsøe, K; Wellendorph, P; Frølund, B J Med Chem 62: 2798 -2813 (2019)
Guo, T; Adang, AE; Dong, G; Fitzpatrick, D; Geng, P; Ho, KK; Jibilian, CH; Kultgen, SG; Liu, R; McDonald, E; Saionz, KW; Valenzano, KJ; van Straten, NC; Xie, D; Webb, ML Bioorg Med Chem Lett 14: 1717 -20 (2004)
Meng, YQ; Ren, J; Sun, JX; Guo, FY; Min, JZ; Nan, JX; Quan, JS; Lian, LH; Jin, CH Eur J Med Chem 269:
Vougogiannopoulou, K; Ferandin, Y; Bettayeb, K; Myrianthopoulos, V; Lozach, O; Fan, Y; Johnson, CH; Magiatis, P; Skaltsounis, AL; Mikros, E; Meijer, L J Med Chem 51: 6421 -31 (2008)
Barrett, DG; Boncek, VM; Catalano, JG; Deaton, DN; Hassell, AM; Jurgensen, CH; Long, ST; McFadyen, RB; Miller, AB; Miller, LR; Payne, JA; Ray, JA; Samano, V; Shewchuk, LM; Tavares, FX; Wells-Knecht, KJ; Willard, DH; Wright, LL; Zhou, HQ Bioorg Med Chem Lett 15: 3540 -6 (2005)
Esbenshade, TA; Krueger, KM; Miller, TR; Kang, CH; Denny, LI; Witte, DG; Yao, BB; Fox, GB; Faghih, R; Bennani, YL; Williams, M; Hancock, AA J Pharmacol Exp Ther 305: 887 -96 (2003)
Jagoda, E; Contoreggi, C; Lee, MJ; Kao, CH; Szajek, LP; Listwak, S; Gold, P; Chrousos, G; Greiner, E; Kim, BM; Jacobson, AE; Rice, KC; Eckelman, W J Med Chem 46: 3559 -62 (2003)
Mayer, SC; Banker, AL; Boschelli, F; Di, L; Johnson, M; Kenny, CH; Krishnamurthy, G; Kutterer, K; Moy, F; Petusky, S; Ravi, M; Tkach, D; Tsou, HR; Xu, W Bioorg Med Chem Lett 18: 3641 -5 (2008)
Kwon, SW; Kang, SK; Lee, JH; Bok, JH; Kim, CH; Dal Rhee, S; Jung, WH; Kim, HY; Bae, MA; Song, JS; Ha, DC; Cheon, HG; Kim, KY; Ahn, JH Bioorg Med Chem Lett 21: 435 -9 (2010)
Li, HY; Wang, Y; Heap, CR; King, CH; Mundla, SR; Voss, M; Clawson, DK; Yan, L; Campbell, RM; Anderson, BD; Wagner, JR; Britt, K; Lu, KX; McMillen, WT; Yingling, JM J Med Chem 49: 2138 -42 (2006)
Khanwelkar, RR; Chen, GS; Wang, HC; Yu, CW; Huang, CH; Lee, O; Chen, CH; Hwang, CS; Ko, CH; Chou, NT; Lin, MW; Wang, LM; Chen, YC; Hseu, TH; Chang, CN; Hsu, HC; Lin, HC; Shih, YC; Chou, SH; Tseng, HW; Liu, CP; Tu, CM; Hu, TL; Tsai, YJ; Chern, JW Bioorg Med Chem 18: 4674 -86 (2011)
Kruse, CH; Holden, KG; Offen, PH; Pritchard, ML; Feild, JA; Rieman, DJ; Bender, PE; Ferguson, B; Greig, RG; Poste, G J Med Chem 31: 1768 -72 (1988)
Kuo, CH; Robichaud, AJ; Rew, DJ; Bergstrom, JD; Berger, GD Bioorg Med Chem Lett 4: 1591 -1594 (1994)
Hsueh, WY; Lee, YE; Huang, MS; Lai, CH; Gao, YS; Lin, JC; Chen, YF; Chang, CL; Chou, SY; Chen, SF; Lu, YY; Chang, LH; Lin, SF; Lin, YH; Hsu, PC; Wei, WY; Huang, YC; Kao, YF; Teng, LW; Liu, HH; Chen, YC; Yuan, TT; Chan, YW; Huang, PH; Chao, YT; Huang, SY; Jian, BH; Huang, HY; Yang, SC; Lo, TH; Huang, GR; Wang, SY; Lin, HS; Chuang, SH; Huang, JJ J Med Chem 64: 1435 -1453 (2021)
Brown, BS; Keddy, R; Perner, RJ; DiDomenico, S; Koenig, JR; Jinkerson, TK; Hannick, SM; McDonald, HA; Bianchi, BR; Honore, P; Puttfarcken, PS; Moreland, RB; Marsh, KC; Faltynek, CR; Lee, CH Bioorg Med Chem Lett 20: 3291 -4 (2010)
Yang, GJ; Wu, J; Miao, L; Zhu, MH; Zhou, QJ; Lu, XJ; Lu, JF; Leung, CH; Ma, DL; Chen, J Eur J Med Chem 226: (2021)
Levenson, CH; Meyer, RB J Med Chem 27: 228 -32 (1984)
Zablocki, JA; Elzein, E; Li, X; Koltun, DO; Parkhill, EQ; Kobayashi, T; Martinez, R; Corkey, B; Jiang, H; Perry, T; Kalla, R; Notte, GT; Saunders, O; Graupe, M; Lu, Y; Venkataramani, C; Guerrero, J; Perry, J; Osier, M; Strickley, R; Liu, G; Wang, WQ; Hu, L; Li, XJ; El-Bizri, N; Hirakawa, R; Kahlig, K; Xie, C; Li, CH; Dhalla, AK; Rajamani, S; Mollova, N; Soohoo, D; Lepist, EI; Murray, B; Rhodes, G; Belardinelli, L; Desai, MC J Med Chem 59: 9005 -9017 (2016)
Chung, KH; Lim, CH; Lee, DR; Jin, C; Chi, DY Bioorg Med Chem Lett 11: 3077 -80 (2001)
Das, A; Adak, AK; Ponnapalli, K; Lin, CH; Hsu, KC; Yang, JM; Hsu, TA; Lin, CC Eur J Med Chem 123: 397 -406 (2016)
Shi, L; Yang, Y; Li, ZL; Zhu, ZW; Liu, CH; Zhu, HL Bioorg Med Chem 18: 1659 -64 (2010)
Lin, CS; Lu, CH; Lin, TH; Kiu, YT; Kan, JY; Chang, YJ; Hung, PY; Koval'skaya, AV; Tsypyshev, DO; Tsypysheva, IP; Lin, CW Bioorg Med Chem Lett 99:
Chang, CC; Cao, S; Kang, S; Kai, L; Tian, X; Pandey, P; Dunne, SF; Luan, CH; Surmeier, DJ; Silverman, RB Bioorg Med Chem 18: 3147 -58 (2010)
YOO, JH; IM, S; LEE, KH; KIM, DH; OH, EH; LEE, DY; JUNG, KM; KWAK, DJ; KIM, SY; KIM, YR; MIN, CH US Patent US20250051275 (2025)
Trani, G; Barker, JJ; Bromidge, SM; Brookfield, FA; Burch, JD; Chen, Y; Eigenbrot, C; Heifetz, A; Ismaili, MH; Johnson, A; Krülle, TM; MacKinnon, CH; Maghames, R; McEwan, PA; Montalbetti, CA; Ortwine, DF; Pérez-Fuertes, Y; Vaidya, DG; Wang, X; Zarrin, AA; Pei, Z Bioorg Med Chem Lett 24: 5818 -23 (2014)
Blackie, JA; Bloomer, JC; Brown, MJ; Cheng, HY; Hammond, B; Hickey, DM; Ife, RJ; Leach, CA; Lewis, VA; Macphee, CH; Milliner, KJ; Moores, KE; Pinto, IL; Smith, SA; Stansfield, IG; Stanway, SJ; Taylor, MA; Theobald, CJ Bioorg Med Chem Lett 13: 1067 -70 (2003)
Baldwin, J; Michnoff, CH; Malmquist, NA; White, J; Roth, MG; Rathod, PK; Phillips, MA J Biol Chem 280: 21847 -53 (2005)
Mazurov, AA; Kombo, DC; Hauser, TA; Miao, L; Dull, G; Genus, JF; Fedorov, NB; Benson, L; Sidach, S; Xiao, Y; Hammond, PS; James, JW; Miller, CH; Yohannes, D J Med Chem 55: 9793 -809 (2012)
Sauerberg, P; Olesen, PH; Nielsen, S; Treppendahl, S; Sheardown, MJ; Honoré, T; Mitch, CH; Ward, JS; Pike, AJ; Bymaster, FP J Med Chem 35: 2274 -83 (1992)
Verga, D; N'Guyen, CH; Dakir, M; Coll, JL; Teulade-Fichou, MP; Molla, A J Med Chem 61: 10502 -10518 (2018)
Tibon, NS; Ng, CH; Cheong, SL Eur J Med Chem 188: (2020)
Pontikis, R; Dollé, V; Guillaumel, J; Dechaux, E; Note, R; Nguyen, CH; Legraverend, M; Bisagni, E; Aubertin, AM; Grierson, DS; Monneret, C J Med Chem 43: 1927 -39 (2000)
James, ML; Shen, B; Zavaleta, CL; Nielsen, CH; Mesangeau, C; Vuppala, PK; Chan, C; Avery, BA; Fishback, JA; Matsumoto, RR; Gambhir, SS; McCurdy, CR; Chin, FT J Med Chem 55: 8272 -82 (2012)
Mersal, KI; Abdel-Maksoud, MS; Ali, EMH; Ammar, UM; Zaraei, SO; Haque, MM; Das, T; Hassan, NF; Kim, EE; Lee, JS; Park, H; Lee, KH; El-Gamal, MI; Kim, HK; Ibrahim, TM; Oh, CH Eur J Med Chem 261:
Kiesewetter, DO; Lee, J; Lang, L; Park, SG; Paik, CH; Eckelman, WC J Med Chem 38: 5 -8 (1995)
Sharma, R; Chatterjee, E; Mathew, J; Sharma, S; Rao, NV; Pan, CH; Lee, SB; Dhingra, A; Grewal, AS; Liou, JP; Guru, SK; Nepali, K Eur J Med Chem 240: (2022)
Achary, R; Mathi, GR; Lee, DH; Yun, CS; Lee, CO; Kim, HR; Park, CH; Kim, P; Hwang, JY Bioorg Med Chem Lett 27: 2185 -2191 (2017)
Owen, CP; Dhanani, S; Patel, CH; Shahid, I; Ahmed, S Bioorg Med Chem Lett 16: 4011 -5 (2006)
Mahindroo, N; Huang, CF; Peng, YH; Wang, CC; Liao, CC; Lien, TW; Chittimalla, SK; Huang, WJ; Chai, CH; Prakash, E; Chen, CP; Hsu, TA; Peng, CH; Lu, IL; Lee, LH; Chang, YW; Chen, WC; Chou, YC; Chen, CT; Goparaju, CM; Chen, YS; Lan, SJ; Yu, MC; Chen, X; Chao, YS; Wu, SY; Hsieh, HP J Med Chem 48: 8194 -208 (2005)
Bremer, PT; Adler, M; Phung, CH; Singh, AK; Janda, KD J Med Chem 60: 338 -348 (2017)
Sweetnam, PM; Caldwell, L; Lancaster, J; Jr., CB; McMillan, B; Kinnier, WJ; Price, CH J Nat Prod 56: 441 -455 (1993)
Pissot-Soldermann, C; Gerspacher, M; Furet, P; Gaul, C; Holzer, P; McCarthy, C; Radimerski, T; Regnier, CH; Baffert, F; Drueckes, P; Tavares, GA; Vangrevelinghe, E; Blasco, F; Ottaviani, G; Ossola, F; Scesa, J; Reetz, J Bioorg Med Chem Lett 20: 2609 -13 (2010)
Hardcastle, IR; Liu, J; Valeur, E; Watson, A; Ahmed, SU; Blackburn, TJ; Bennaceur, K; Clegg, W; Drummond, C; Endicott, JA; Golding, BT; Griffin, RJ; Gruber, J; Haggerty, K; Harrington, RW; Hutton, C; Kemp, S; Lu, X; McDonnell, JM; Newell, DR; Noble, ME; Payne, SL; Revill, CH; Riedinger, C; Xu, Q; Lunec, J J Med Chem 54: 1233 -43 (2011)
Kolluri, R; Tegley, CM; Zhu, L; Brown, SP; Reynolds, CH; Tasker, AS; Grice, CA US Patent US11629136 (2023)
Bashore, FM; Min, SM; Chen, X; Howell, S; Rinderle, CH; Morel, G; Silvaroli, JA; Wells, CI; Bunnell, BA; Drewry, DH; Pabla, NS; Ultanir, SK; Bullock, AN; Axtman, AD ACS Med Chem Lett 15: 1325 -1333
Childers, WE; Silverton, JV; Kellis, JT; Vickery, LE; Robinson, CH J Med Chem 34: 1344 -9 (1991)
Song, X; Chen, W; Lin, L; Ruiz, CH; Cameron, MD; Duckett, DR; Kamenecka, TM Bioorg Med Chem Lett 21: 7072 -5 (2011)
Yoon, J; Choi, H; Lee, HJ; Ryu, CH; Park, HG; Suh, YG; Oh, U; Jeong, YS; Choi, JK; Park, YH; Kim, HD Bioorg Med Chem Lett 13: 1549 -52 (2003)
Quancard, J; Simic, O; Pissot Soldermann, C; Aichholz, R; Blatter, M; Renatus, M; Erbel, P; Melkko, S; Endres, R; Sorge, M; Kieffer, L; Wagner, T; Beltz, K; Mcsheehy, P; Wartmann, M; Régnier, CH; Calzascia, T; Radimerski, T; Bigaud, M; Weiss, A; Bornancin, F; Schlapbach, A J Med Chem 63: 14594 -14608 (2020)
Chen, D; Misra, M; Sower, L; Peterson, JW; Kellogg, GE; Schein, CH Bioorg Med Chem 16: 7225 -33 (2008)
Ashton, TD; Aumann, KM; Baker, SP; Schiesser, CH; Scammells, PJ Bioorg Med Chem Lett 17: 6779 -84 (2007)
Alnabulsi, S; Hussein, B; Santina, E; Alsalahat, I; Kadirvel, M; Magwaza, RN; Bryce, RA; Schwalbe, CH; Baldwin, AG; Russo, I; Stratford, IJ; Freeman, S Bioorg Med Chem Lett 28: 1292 -1297 (2018)
Yu, WC; Yeh, TY; Ye, CH; Chong, PCT; Ho, YH; So, DK; Yap, KY; Peng, GR; Shao, CH; Jagtap, AD; Chern, JW; Lin, CS; Lin, SP; Lin, SL; Yu, SH; Yu, CW J Med Chem 66: 10528 -10557 (2023)
Agniswamy, J; Louis, JM; Shen, CH; Yashchuk, S; Ghosh, AK; Weber, IT J Med Chem 58: 5088 -95 (2015)
Rosowsky, A; Forsch, RA; Sibley, CH; Inderlied, CB; Queener, SF J Med Chem 47: 1475 -86 (2004)
Yang, SH; Song, CH; Van, HT; Park, E; Khadka, DB; Gong, EY; Lee, K; Cho, WJ J Med Chem 56: 3414 -8 (2013)
Larsen, SD; Spilman, CH; Bell, FP; Dinh, DM; Martinborough, E; Wilson, GJ J Med Chem 34: 1721 -7 (1991)
Ahmad, S; Phillips, RS; Stammer, CH J Med Chem 35: 1410 -7 (1992)
Fong, J; Yuan, M; Jakobsen, TH; Mortensen, KT; Delos Santos, MM; Chua, SL; Yang, L; Tan, CH; Nielsen, TE; Givskov, M J Med Chem 60: 215 -227 (2017)
Shao, A; Kang, CW; Tang, CH; Cain, CF; Xu, Q; Phoumyvong, CM; Del Valle, JR; Hu, CC J Med Chem 62: 5404 -5413 (2019)
Turner, LD; Trinh, CH; Hubball, RA; Orritt, KM; Lin, CC; Burns, JE; Knowles, MA; Fishwick, CWG J Med Chem 65: 1481 -1504 (2022)
Chi, YH; Yeh, TK; Ke, YY; Lin, WH; Tsai, CH; Wang, WP; Chen, YT; Su, YC; Wang, PC; Chen, YF; Wu, ZW; Yeh, JY; Hung, MC; Wu, MH; Wang, JY; Chen, CP; Song, JS; Shih, C; Chen, CT; Chang, CP J Med Chem 64: 7312 -7330 (2021)
Tseng, CH; Tzeng, CC; Yang, CL; Lu, PJ; Chen, HL; Li, HY; Chuang, YC; Yang, CN; Chen, YL J Med Chem 53: 6164 -79 (2010)
Peng, YH; Ueng, SH; Tseng, CT; Hung, MS; Song, JS; Wu, JS; Liao, FY; Fan, YS; Wu, MH; Hsiao, WC; Hsueh, CC; Lin, SY; Cheng, CY; Tu, CH; Lee, LC; Cheng, MF; Shia, KS; Shih, C; Wu, SY J Med Chem 59: 282 -93 (2016)
Cheng, Y; Zhou, M; Tung, CH; Ji, M; Zhang, F Bioorg Med Chem Lett 20: 3329 -37 (2010)
Boyle, RG; Walker, DW; Boyce, RJ; Peterson, S; Farouz, F; Vo, CH US Patent US10973817 (2021)
Wang, CH; Wu, HT; Cheng, HM; Yen, TJ; Lu, IH; Chang, HC; Jao, SC; Shing, TK; Li, WS J Med Chem 54: 8574 -81 (2011)
Milne, JC; Lambert, PD; Schenk, S; Carney, DP; Smith, JJ; Gagne, DJ; Jin, L; Boss, O; Perni, RB; Vu, CB; Bemis, JE; Xie, R; Disch, JS; Ng, PY; Nunes, JJ; Lynch, AV; Yang, H; Galonek, H; Israelian, K; Choy, W; Iffland, A; Lavu, S; Medvedik, O; Sinclair, DA; Olefsky, JM; Jirousek, MR; Elliott, PJ; Westphal, CH Nature 450: 712 -716 (2007)
Hong, CC; Williams, CH; Singh, LR US Patent US12194027 (2025)
Hong, BT; Chen, CL; Fang, JM; Tsai, KC; Wang, SY; Huang, WI; Cheng, YS; Wong, CH Bioorg Med Chem 22: 6647 -54 (2015)
Tseng, SL; Hung, MS; Chang, CP; Song, JS; Tai, CL; Chiu, HH; Hsieh, WP; Lin, Y; Chung, WL; Kuo, CW; Wu, CH; Chu, CM; Tung, YS; Chao, YS; Shia, KS J Med Chem 51: 5397 -412 (2008)
Moschen, T; Grutsch, S; Juen, MA; Wunderlich, CH; Kreutz, C; Tollinger, M J Med Chem 59: 10788 -10793 (2016)
Wang, K; Xu, CH; Tong, L; Wang, B; Liu, AH; Li, SW; Mao, SC J Nat Prod 87: 121 -131 (2024)
Xiang, HY; Chen, JY; Huan, XJ; Chen, Y; Gao, ZB; Ding, J; Miao, ZH; Yang, CH Bioorg Med Chem Lett 31: (2021)
Yao, CH; Song, JS; Chen, CT; Yeh, TK; Hsieh, TC; Wu, SH; Huang, CY; Huang, YL; Wang, MH; Liu, YW; Tsai, CH; Kumar, CR; Lee, JC Eur J Med Chem 55: 32 -8 (2012)
Yu, WC; Yeh, TY; Ye, CH; Chong, PCT; Ho, YH; So, DK; Yap, KY; Peng, GR; Shao, CH; Jagtap, AD; Chern, JW; Lin, CS; Lin, SP; Lin, SL; Yu, SH; Yu, CW J Med Chem 66: 10528 -10557 (2023)
Adelstein, GW; Yen, CH; Haack, RA; Yu, S; Gullikson, G; Price, DV; Anglin, C; Decktor, DL; Tsai, H; Keith, RH J Med Chem 31: 1215 -20 (1988)
Yogo, T; Nagamiya, H; Seto, M; Sasaki, S; Shih-Chung, H; Ohba, Y; Tokunaga, N; Lee, GN; Rhim, CY; Yoon, CH; Cho, SY; Skene, R; Yamamoto, S; Satou, Y; Kuno, M; Miyazaki, T; Nakagawa, H; Okabe, A; Marui, S; Aso, K; Yoshida, M J Med Chem 59: 733 -49 (2016)
Zhong, M; Bui, M; Shen, W; Baskaran, S; Allen, DA; Elling, RA; Flanagan, WM; Fung, AD; Hanan, EJ; Harris, SO; Heumann, SA; Hoch, U; Ivy, SN; Jacobs, JW; Lam, S; Lee, H; McDowell, RS; Oslob, JD; Purkey, HE; Romanowski, MJ; Silverman, JA; Tangonan, BT; Taverna, P; Yang, W; Yoburn, JC; Yu, CH; Zimmerman, KM; O'Brien, T; Lew, W Bioorg Med Chem Lett 19: 5158 -61 (2009)
Yuan, CH; Filippova, M; Tungteakkhun, SS; Duerksen-Hughes, PJ; Krstenansky, JL Bioorg Med Chem Lett 22: 2125 -9 (2012)
Zhou, W; Ercan, D; Chen, L; Yun, CH; Li, D; Capelletti, M; Cortot, AB; Chirieac, L; Iacob, RE; Padera, R; Engen, JR; Wong, KK; Eck, MJ; Gray, NS; Jänne, PA Nature 462: 1070 -4
Zhang, CH; Chen, K; Jiao, Y; Li, LL; Li, YP; Zhang, RJ; Zheng, MW; Zhong, L; Huang, SZ; Song, CL; Lin, WT; Yang, J; Xiang, R; Peng, B; Han, JH; Lu, GW; Wei, YQ; Yang, SY J Med Chem 59: 9788 -9805 (2016)
Liu, J; Zheng, CH; Ren, XH; Zhou, F; Li, W; Zhu, J; Lv, JG; Zhou, YJ J Med Chem 55: 5720 -33 (2012)
Wang, LL; Battini, N; Bheemanaboina, RRY; Zhang, SL; Zhou, CH Eur J Med Chem 167: 105 -123 (2019)
Gu, YG; Weitzberg, M; Clark, RF; Xu, X; Li, Q; Lubbers, NL; Yang, Y; Beno, DW; Widomski, DL; Zhang, T; Hansen, TM; Keyes, RF; Waring, JF; Carroll, SL; Wang, X; Wang, R; Healan-Greenberg, CH; Blomme, EA; Beutel, BA; Sham, HL; Camp, HS J Med Chem 50: 1078 -82 (2007)
Lesuisse, D; Tiraboschi, G; Krick, A; Abecassis, PY; Dutruc-Rosset, G; Babin, D; Halley, F; Châtreau, F; Lachaud, S; Chevalier, A; Quarteronet, D; Burgevin, MC; Amara, C; Bertrand, P; Rooney, T Bioorg Med Chem Lett 20: 2344 -9 (2010)
Furet, P; Schoepfer, J; Radimerski, T; Chène, P Bioorg Med Chem Lett 19: 4014 -7 (2009)
Bienaymé, H; Chêne, L; Grisoni, S; Grondin, A; Kaloun, el-B; Poigny, S; Rahali, H; Tam, E Bioorg Med Chem Lett 16: 4830 -3 (2006)
Bernier, S; Dubois, DY; Therrien, M; Lapointe, J; Chênevert, R Bioorg Med Chem Lett 10: 2441 -4 (2001)
Degterev, A; Hitomi, J; Germscheid, M; Ch'en, IL; Korkina, O; Teng, X; Abbott, D; Cuny, GD; Yuan, C; Wagner, G; Hedrick, SM; Gerber, SA; Lugovskoy, A; Yuan, J Nat Chem Biol 4: 313 -21 (2008)
Bernier, S; Akochy, PM; Lapointe, J; Chênevert, R Bioorg Med Chem 13: 69 -75 (2005)
Bourderioux, A; Naus, P; Perlíková, P; Pohl, R; Pichová, I; Votruba, I; Dzubák, P; Konecný, P; Hajdúch, M; Stray, KM; Wang, T; Ray, AS; Feng, JY; Birkus, G; Cihlar, T; Hocek, M J Med Chem 54: 5498 -507 (2011)
Jiménez-Alonso, S; Pérez-Lomas, AL; Estévez-Braun, A; Muñoz Martinez, F; Chávez Orellana, H; Ravelo, AG; Gamarro, F; Castanys, S; López, M J Med Chem 51: 7132 -43 (2009)