- D., AE; W., AS; Jean, BC; R., CK; C., IT; KOLAKOWSKI, KG; Manoj, K; A., ME; L., MM; Alexander, MJ; Tiphaine, M; J., MM; Dino, PT; Alexander, PM; Marta, P WIPO WO2022098970 (2022)
- Huffman, JW; Yu, S; Showalter, V; Abood, ME; Wiley, JL; Compton, DR; Martin, BR; Bramblett, RD; Reggio, PH J Med Chem 39: 3875-7 (1996)
- Erickson, RH; Hiner, RN; Feeney, SW; Blake, PR; Rzeszotarski, WJ; Hicks, RP; Costello, DG; Abreu, ME J Med Chem 34: 1431-5 (1991)
- Hudson, AR; Higuchi, RI; Roach, SL; Adams, ME; Vassar, A; Syka, PM; Mais, DE; Miner, JN; Marschke, KB; Zhi, L Bioorg Med Chem Lett 21: 1697-700 (2011)
- Salerno, L; Modica, MN; Romeo, G; Pittalà, V; Siracusa, MA; Amato, ME; Acquaviva, R; Di Giacomo, C; Sorrenti, V Eur J Med Chem 49: 118-26 (2012)
- Arango ME
- Tomassini, J; Selnick, H; Davies, ME; Armstrong, ME; Baldwin, J; Bourgeois, M; Hastings, J; Hazuda, D; Lewis, J; McClements, W Antimicrob Agents Chemother 38: 2827-37 (1995)
- Gouleni, N; Di Rienzo, A; Yılmaz, A; Selvitopi, H; Arslan, ME; Mardinoglu, A; Turkez, H; Di Stefano, A; Vassiliou, S; Cacciatore, I RSC Med Chem 14: 2315-2326 (2023)
- Krause-Heuer, AM; Fraser-Spears, R; Dobrowolski, JC; Ashford, ME; Wyatt, NA; Roberts, MP; Gould, GG; Cheah, WC; Ng, CKL; Bhadbhade, M; Zhang, B; Greguric, I; Wheate, NJ; Kumar, N; Koek, W; Callaghan, PD; Daws, LC; Fraser, BH Eur J Med Chem 137: 476-487 (2017)
- Khanapure, SP; Augustyniak, ME; Earl, RA; Garvey, DS; Letts, LG; Martino, AM; Murty, MG; Schwalb, DJ; Shumway, MJ; Trocha, AM; Young, DV; Zemtseva, IS; Janero, DR J Med Chem 48: 3930-4 (2005)
- Li, R; Cheng, C; Balasis, ME; Liu, Y; Garner, TP; Daniel, KG; Li, J; Qin, Y; Gavathiotis, E; Sebti, SM Eur J Med Chem 90: 315-31 (2015)
- Thorarensen, A; Dowty, ME; Banker, ME; Juba, B; Jussif, J; Lin, T; Vincent, F; Czerwinski, RM; Casimiro-Garcia, A; Unwalla, R; Trujillo, JI; Liang, S; Balbo, P; Che, Y; Gilbert, AM; Brown, MF; Hayward, M; Montgomery, J; Leung, L; Yang, X; Soucy, S; Hegen, M; Coe, J; Langille, J; Vajdos, F; Chrencik, J; Telliez, JB J Med Chem 60: 1971-1993 (2017)
- Ennis, MD; Baze, ME; Smith, MW; Lawson, CF; McCall, RB; Lahti, RA; Piercey, MF J Med Chem 35: 3058-66 (1992)
- Grabe, T; Jeyakumar, K; Niggenaber, J; Schulz, T; Koska, S; Kleinbölting, S; Beck, ME; Müller, MP; Rauh, D ACS Med Chem Lett 14: 591-598 (2023)
- Papillon, JP; Lou, C; Singh, AK; Adams, CM; Ksander, GM; Beil, ME; Chen, W; Leung-Chu, J; Fu, F; Gan, L; Hu, CW; Jeng, AY; LaSala, D; Liang, G; Rigel, DF; Russell, KS; Vest, JA; Watson, C J Med Chem 58: 9382-94 (2015)
- Bembenek, ME; Abell, CW; Chrisey, LA; Rozwadowska, MD; Gessner, W; Brossi, A J Med Chem 33: 147-52 (1990)
- López-Rodríguez, ML; Rosado, ML; Benhamú, B; Morcillo, MJ; Sanz, AM; Orensanz, L; Beneitez, ME; Fuentes, JA; Manzanares, J J Med Chem 39: 4439-50 (1996)
- López-Rodríguez, ML; Morcillo, MJ; Fernández, E; Porras, E; Orensanz, L; Beneytez, ME; Manzanares, J; Fuentes, JA J Med Chem 44: 186-97 (2001)
- Shishodia, S; Nuñez, R; Strohmier, BP; Bursch, KL; Goetz, CJ; Olp, MD; Jensen, DR; Fenske, TG; Ordonez-Rubiano, SC; Blau, ME; Roach, MK; Peterson, FC; Volkman, BF; Dykhuizen, EC; Smith, BC J Med Chem 65: 13714-13735 (2022)
- Bolitho, ME; Perez, LJ; Koch, MJ; Ng, WL; Bassler, BL; Semmelhack, MF Bioorg Med Chem 19: 6906-18 (2011)
- Bordeleau, ME; Mori, A; Oberer, M; Lindqvist, L; Chard, LS; Higa, T; Belsham, GJ; Wagner, G; Tanaka, J; Pelletier, J Nat Chem Biol 2: 213-20 (2006)
- Le Manach, C; Nchinda, AT; Paquet, T; Gonzàlez Cabrera, D; Younis, Y; Han, Z; Bashyam, S; Zabiulla, M; Taylor, D; Lawrence, N; White, KL; Charman, SA; Waterson, D; Witty, MJ; Wittlin, S; Botha, ME; Nondaba, SH; Reader, J; Birkholtz, LM; Jiménez-Díaz, MB; Martínez, MS; Ferrer, S; Angulo-Barturen, I; Meister, S; Antonova-Koch, Y; Winzeler, EA; Street, LJ; Chibale, K J Med Chem 59: 9890-9905 (2016)
- Deligia, F; Deiana, V; Gotti, C; Lazzari, P; Bottazzi, ME; Pucci, L; Fasoli, F; Ragusa, G; Pinna, GA; Murineddu, G Eur J Med Chem 103: 429-37 (2015)
- Boursier, ME; Manson, DE; Combs, JB; Blackwell, HE Bioorg Med Chem 26: 5336-5342 (2018)
- Hoveyda, HR; Dutheuil, G; Fraser, GL; Roy, M; Bousmaqui, ME; Batt, F US Patent US10683295 (2020)
- Lowe, DB; Magnuson, S; Qi, N; Campbell, AM; Cook, J; Hong, Z; Wang, M; Rodriguez, M; Achebe, F; Kluender, H; Wong, WC; Bullock, WH; Salhanick, AI; Witman-Jones, T; Bowling, ME; Keiper, C; Clairmont, KB Bioorg Med Chem Lett 14: 3155-9 (2004)
- Sullivan, TJ; Truglio, JJ; Boyne, ME; Novichenok, P; Zhang, X; Stratton, CF; Li, HJ; Kaur, T; Amin, A; Johnson, F; Slayden, RA; Kisker, C; Tonge, PJ ACS Chem Biol 1: 43-53 (2006)
- Roman, BI; De Ryck, T; Patronov, A; Slavov, SH; Vanhoecke, BW; Katritzky, AR; Bracke, ME; Stevens, CV Eur J Med Chem 101: 627-39 (2015)
- Bockman, CS; Bradley, ME; Dang, HK; Zeng, W; Scofield, MA; Dowd, FJ J Pharmacol Exp Ther 297: 718-26 (2001)
- Sarau, HM; Griswold, DE; Potts, W; Foley, JJ; Schmidt, DB; Webb, EF; Martin, LD; Brawner, ME; Elshourbagy, NA; Medhurst, AD; Giardina, GA; Hay, DW J Pharmacol Exp Ther 281: 1303-11 (1997)
- Yestrepsky, BD; Xu, Y; Breen, ME; Li, X; Rajeswaran, WG; Ryu, JG; Sorenson, RJ; Tsume, Y; Wilson, MW; Zhang, W; Sun, D; Sun, H; Larsen, SD Bioorg Med Chem 21: 1880-97 (2013)
- Zhao, G; Souers, AJ; Voorbach, M; Falls, HD; Droz, B; Brodjian, S; Lau, YY; Iyengar, RR; Gao, J; Judd, AS; Wagaw, SH; Ravn, MM; Engstrom, KM; Lynch, JK; Mulhern, MM; Freeman, J; Dayton, BD; Wang, X; Grihalde, N; Fry, D; Beno, DW; Marsh, KC; Su, Z; Diaz, GJ; Collins, CA; Sham, H; Reilly, RM; Brune, ME; Kym, PR J Med Chem 51: 380-3 (2008)
- Datta, S; Bucks, ME; Koley, D; Lim, PX; Savinov, SN Bioorg Med Chem 18: 6099-108 (2010)
- Trzupek, JD; Lee, KL; Bunnage, ME; Han, S; Hepworth, D; Lovering, FE; Mathias, JP; Papaioannou, N; Pierce, BS; Strohbach, JW; Wright, SW; Zapf, CW; Gavrin, LK; Lee, A; Anderson, DR; Curran, KJ; Dehnhardt, CM; Saiah, E; Goldberg, JA; Wang, X; Huang, H; Vargas, R; Lowe, MD; Patny, A US Patent US10329302 (2019)
- Jiang, Q; Payton-Stewart, F; Elliott, S; Driver, J; Rhodes, LV; Zhang, Q; Zheng, S; Bhatnagar, D; Boue, SM; Collins-Burow, BM; Sridhar, J; Stevens, C; McLachlan, JA; Wiese, TE; Burow, ME; Wang, G J Med Chem 53: 6153-63 (2010)
- Thurmond, J; Butchbach, ME; Palomo, M; Pease, B; Rao, M; Bedell, L; Keyvan, M; Pai, G; Mishra, R; Haraldsson, M; Andresson, T; Bragason, G; Thosteinsdottir, M; Bjornsson, JM; Coovert, DD; Burghes, AH; Gurney, ME; Singh, J J Med Chem 51: 449-69 (2008)
- López-Cara, LC; Carrión, MD; Entrena, A; Gallo, MA; Espinosa, A; López, A; Escames, G; Acuña-Castroviejo, D; Camacho, ME Eur J Med Chem 50: 129-39 (2012)
- Murray, CW; Berdini, V; Buck, IM; Carr, ME; Cleasby, A; Coyle, JE; Curry, JE; Day, JE; Day, PJ; Hearn, K; Iqbal, A; Lee, LY; Martins, V; Mortenson, PN; Munck, JM; Page, LW; Patel, S; Roomans, S; Smith, K; Tamanini, E; Saxty, G ACS Med Chem Lett 6: 798-803 (2015)
- Fontenla, JA; Osuna, J; Rosa, E; Castro, ME; G-Ferreiro, T; Loza-García, I; Calleja, JM; Sanz, F; Rodríguez, J; Raviña, E J Med Chem 37: 2564-73 (1994)
- Patel, SD; Habeski, WM; Min, H; Zhang, J; Roof, R; Snyder, B; Bora, G; Campbell, B; Li, C; Hidayetoglu, D; Johnson, DS; Chaudhry, A; Charlton, ME; Kablaoui, NM Bioorg Med Chem Lett 18: 5689-93 (2008)
- Chiari, ME; Vera, DM; Palacios, SM; Carpinella, MC Bioorg Med Chem 19: 3474-82 (2011)
- Galal, KA; Truong, A; Kwarcinski, F; de Silva, C; Avalani, K; Havener, TM; Chirgwin, ME; Merten, E; Ong, HW; Willis, C; Abdelwaly, A; Helal, MA; Derbyshire, ER; Zutshi, R; Drewry, DH J Med Chem 65: 13172-13197 (2022)
- Burkholder, TP; Cunningham, BE; Clayton, JR; Lander, PA; Brown, ML; Doti, RA; Durst, GL; Montrose-Rafizadeh, C; King, C; Osborne, HE; Amos, RM; Zink, RW; Stramm, LE; Burris, TP; Cardona, G; Konkol, DL; Reidy, C; Christe, ME; Genin, MJ Bioorg Med Chem Lett 25: 1377-80 (2015)
- Baldwin, JJ; Ponticello, GS; Anderson, PS; Christy, ME; Murcko, MA; Randall, WC; Schwam, H; Sugrue, MF; Springer, JP; Gautheron, P J Med Chem 32: 2510-3 (1989)
- Miknis, GF; Stevens, SJ; Smith, LE; Ostrov, DA; Churchill, ME Bioorg Med Chem Lett 25: 963-8 (2015)
- Wheelock, CE; Nishi, K; Ying, A; Jones, PD; Colvin, ME; Olmstead, MM; Hammock, BD Bioorg Med Chem 16: 2114-30 (2008)
- Condon, ME; Cimarusti, CM; Fox, R; Narayanan, VL; Reid, J; Sundeen, JE; Hauck, FP J Med Chem 21: 913-22 (1978)
- Guile, SD; Bantick, JR; Cooper, ME; Donald, DK; Eyssade, C; Ingall, AH; Lewis, RJ; Martin, BP; Mohammed, RT; Potter, TJ; Reynolds, RH; St-Gallay, SA; Wright, AD J Med Chem 50: 254-63 (2007)
- Mulchande, J; Simões, SI; Gaspar, MM; Eleutério, CV; Oliveira, R; Cruz, ME; Moreira, R; Iley, J J Enzyme Inhib Med Chem 26: 169-75 (2011)
- Xie, Y; Tummala, P; Oakley, AJ; Deora, GS; Nakano, Y; Rooke, M; Cuellar, ME; Strasser, JM; Dahlin, JL; Walters, MA; Casarotto, MG; Board, PG; Baell, JB J Med Chem 63: 2894-2914 (2020)
- McIntyre, CJ; McCauley, JA; Bednar, B; Bednar, RA; Butcher, JW; Claremon, DA; Cunningham, ME; Freidinger, RM; Gaul, SL; Homnick, CF; Koblan, KS; Mosser, SD; Romano, JJ; Liverton, NJ Bioorg Med Chem Lett 19: 5132-5 (2009)
- Xiao, HY; Watterson, SH; Langevine, CM; Srivastava, AS; Ko, SS; Zhang, Y; Cherney, RJ; Guo, WW; Gilmore, JL; Sheppeck, JE; Wu, DR; Li, P; Ramasamy, D; Arunachalam, P; Mathur, A; Taylor, TL; Shuster, DJ; McIntyre, KW; Shen, DR; Yarde, M; Cvijic, ME; Marino, AM; Balimane, PV; Yang, Z; Banas, DM; Cornelius, G; D'Arienzo, CJ; Warrack, BM; Lehman-McKeeman, L; Salter-Cid, LM; Xie, J; Barrish, JC; Carter, PH; Dyckman, AJ; Dhar, TG J Med Chem 59: 9837-9854 (2016)
- Xiao, HY; Balog, A; Attar, RM; Fairfax, D; Fleming, LB; Holst, CL; Martin, GS; Rossiter, LM; Chen, J; Cvjic, ME; Dell-John, J; Geng, J; Gottardis, MM; Han, WC; Nation, A; Obermeier, M; Rizzo, CA; Schweizer, L; Spires, T; Shan, W; Gavai, A; Salvati, ME; Vite, G Bioorg Med Chem Lett 20: 4491-5 (2010)
- Doherty, JB; Ashe, BM; Barker, PL; Blacklock, TJ; Butcher, JW; Chandler, GO; Dahlgren, ME; Davies, P; Dorn, CP; Finke, PE J Med Chem 33: 2513-21 (1990)
- Litaudon, M; Bousserouel, H; Awang, K; Nosjean, O; Martin, MT; Dau, ME; Hadi, HA; Boutin, JA; Sévenet, T; Guéritte, F J Nat Prod 72: 480-3 (2010)
- Tomassini, J; Selnick, H; Davies, ME; Armstrong, ME; Baldwin, J; Bourgeois, M; Hastings, J; Hazuda, D; Lewis, J; McClements, W Antimicrob Agents Chemother 38: 2827-37 (1995)
- Sutton, JC; Bolton, SA; Davis, ME; Hartl, KS; Jacobson, B; Mathur, A; Ogletree, ML; Slusarchyk, WA; Zahler, R; Seiler, SM; Bisacchi, GS Bioorg Med Chem Lett 14: 2233-9 (2004)
- Velagapudi, UK; Langelier, MF; Delgado-Martin, C; Diolaiti, ME; Bakker, S; Ashworth, A; Patel, BA; Shao, X; Pascal, JM; Talele, TT J Med Chem 62: 5330-5357 (2019)
- Wang, X; Moon, J; Dodge, ME; Pan, X; Zhang, L; Hanson, JM; Tuladhar, R; Ma, Z; Shi, H; Williams, NS; Amatruda, JF; Carroll, TJ; Lum, L; Chen, C J Med Chem 56: 2700-4 (2013)
- Cheng, M; De, B; Pikul, S; Almstead, NG; Natchus, MG; Anastasio, MV; McPhail, SJ; Snider, CE; Taiwo, YO; Chen, L; Dunaway, CM; Gu, F; Dowty, ME; Mieling, GE; Janusz, MJ; Wang-Weigand, S J Med Chem 43: 369-80 (2000)
- Maresso, AW; Wu, R; Kern, JW; Zhang, R; Janik, D; Missiakas, DM; Duban, ME; Joachimiak, A; Schneewind, O J Biol Chem 282: 23129-39 (2007)
- Marín-Rubio, JL; Peltier-Heap, RE; Dueñas, ME; Heunis, T; Dannoura, A; Inns, J; Scott, J; Simpson, AJ; Blair, HJ; Heidenreich, O; Allan, JM; Watt, JE; Martin, MP; Saxty, B; Trost, M J Med Chem 65: 12014-12030 (2022)
- Engers, DW; Melancon, BJ; Gregro, AR; Bertron, JL; Bollinger, SR; Felts, AS; Konkol, LC; Wood, MR; Bollinger, KA; Luscombe, VB; Rodriguez, AL; Jones, CK; Bubser, M; Yohn, SE; Wood, MW; Brandon, NJ; Dugan, ME; Niswender, CM; Conn, PJ; Bridges, TM; Lindsley, CW Bioorg Med Chem Lett 29: 1714-1718 (2019)
- Lindsley, CW; Zhao, Z; Leister, WH; Robinson, RG; Barnett, SF; Defeo-Jones, D; Jones, RE; Hartman, GD; Huff, JR; Huber, HE; Duggan, ME Bioorg Med Chem Lett 15: 761-4 (2005)
- Dumas, ME; Chen, GY; Kendrick, ND; Xu, G; Larsen, SD; Jana, S; Waterson, AG; Bauer, JA; Hancock, W; Sulikowski, GA; Ohi, R Bioorg Med Chem Lett 29: 148-154 (2019)
- Butler, TW; Blake, JF; Bordner, J; Butler, P; Chenard, BL; Collins, MA; DeCosta, D; Ducat, MJ; Eisenhard, ME; Menniti, FS; Pagnozzi, MJ; Sands, SB; Segelstein, BE; Volberg, W; White, WF; Zhao, D J Med Chem 41: 1172-84 (1998)
- Bylund, J; Ek, ME; Gravenfors, Y; Nordvall, G; Minidis, A; Vallin, KS; Viklund, J; Holenz, J; Von Berg, S; Sohn, D US Patent US9145380 (2015)
- Allam, HA; Fahim, SH; F Abo-Ashour, M; Nocentini, A; Elbakry, ME; Abdelrahman, MA; Eldehna, WM; Ibrahim, HS; Supuran, CT Eur J Med Chem 179: 547-556 (2019)
- Kline, RH; Eshleman, AJ; Wright, J; Eldefrawi, ME J Med Chem 37: 2249-52 (1994)
- Hamer, RR; Tegeler, JJ; Kurtz, ES; Allen, RC; Bailey, SC; Elliott, ME; Hellyer, L; Helsley, GC; Przekop, P; Freed, BS; White, J; Martin, LL J Med Chem 39: 246-52 (1996)
- Zacharie, B; Abbott, SD; Bienvenu, JF; Cameron, AD; Cloutier, J; Duceppe, JS; Ezzitouni, A; Fortin, D; Houde, K; Lauzon, C; Moreau, N; Perron, V; Wilb, N; Asselin, M; Doucet, A; Fafard, ME; Gaudreau, D; Grouix, B; Sarra-Bournet, F; St-Amant, N; Gagnon, L; Penney, CL J Med Chem 53: 1138-45 (2010)
- Balasubramanian, N; St Laurent, DR; Federici, ME; Meanwell, NA; Wright, JJ; Schumacher, WA; Seiler, SM J Med Chem 36: 300-3 (1993)
- Apsel, B; Blair, JA; Gonzalez, B; Nazif, TM; Feldman, ME; Aizenstein, B; Hoffman, R; Williams, RL; Shokat, KM; Knight, ZA Nat Chem Biol 4: 691-9 (2008)
- Cebrián-Torrejón, G; Assad Kahn, S; Lagarde, N; Castellano, F; Leblanc, K; Rodrigo, J; Molinier-Frenkel, V; Rojas de Arias, A; Ferreira, ME; Thirant, C; Fournet, A; Figadère, B; Chneiweiss, H; Poupon, E J Nat Prod 75: 257-61 (2012)
- Petrov, RR; Ferrini, ME; Jaffar, Z; Thompson, CM; Roberts, K; Diaz, P Bioorg Med Chem Lett 21: 5859-62 (2011)
- Phillips, AJ; Nasveschuk, CG; Henderson, JA; Liang, Y; Fitzgerald, ME; He, M; Michael, RE US Patent US10646575 (2020)
- Brown, MF; Fenwick, AE; Flanagan, ME; Gonzales, A; Johnson, TA; Kaila, N; Mitton-Fry, MJ; Strohbach, JW; TenBrink, RE; Trzupek, JD; Unwalla, RJ; Vazquez, ML; Parikh, MD US Patent US9035074 (2015)
- Flaugh, ME; Mullen, DL; Fuller, RW; Mason, NR J Med Chem 31: 1746-53 (1988)
- Breslin, MJ; Fraley, ME; Ford, MC; Jones, SR., KL; Roecker, AJ; Schirripa, KM; Tong, L US Patent US20230391758 (2023)
- Francisco, ME; Seltzman, HH; Gilliam, AF; Mitchell, RA; Rider, SL; Pertwee, RG; Stevenson, LA; Thomas, BF J Med Chem 45: 2708-19 (2002)
- Qian, Y; Hamilton, M; Sidduri, A; Gabriel, S; Ren, Y; Peng, R; Kondru, R; Narayanan, A; Truitt, T; Hamid, R; Chen, Y; Zhang, L; Fretland, AJ; Sanchez, RA; Chang, KC; Lucas, M; Schoenfeld, RC; Laine, D; Fuentes, ME; Stevenson, CS; Budd, DC J Med Chem 55: 7920-39 (2012)
- Kyle, DJ; Goehring, RR; Fundytus, ME US Patent US8530494 (2013)
- Ganapathy, ME; Huang, W; Wang, H; Ganapathy, V; Leibach, FH Biochem Biophys Res Commun 246: 470-5 (1998)
- Melnick, JS; Janes, J; Kim, S; Chang, JY; Sipes, DG; Gunderson, D; Jarnes, L; Matzen, JT; Garcia, ME; Hood, TL; Beigi, R; Xia, G; Harig, RA; Asatryan, H; Yan, SF; Zhou, Y; Gu, XJ; Saadat, A; Zhou, V; King, FJ; Shaw, CM; Su, AI; Downs, R; Gray, NS; Schultz, PG; Warmuth, M; Caldwell, JS Proc Natl Acad Sci U S A 103: 3153-8 (2006)
- Munk, SA; Lai, RK; Burke, JE; Arasasingham, PN; Kharlamb, AB; Manlapaz, CA; Padillo, EU; Wijono, MK; Hasson, DW; Wheeler, LA; Garst, ME J Med Chem 39: 1193-5 (1996)
- Bylund, DB; Gerety, ME; Happe, HK; Murrin, LC J Neurosci Methods 105: 159-66 (2001)
- Babler, M; Gerritsen, ME US Patent US9572811 (2017)
- Giusepponi, ME; Cifani, C; Micioni Di Bonaventura, MV; Mattioli, L; Hudson, A; Diamanti, E; Del Bello, F; Giannella, M; Mammoli, V; Paoletti, CD; Piergentili, A; Pigini, M; Quaglia, W ACS Med Chem Lett 7: 956-961 (2016)
- Leblanc, E; Ban, F; Cavga, AD; Lawn, S; Huang, CF; Mohan, S; Chang, MEK; Flory, MR; Ghaidi, F; Lingadahalli, S; Chen, G; Yu, IPL; Morin, H; Lallous, N; Gleave, ME; Mohammed, H; Young, RN; Rennie, PS; Lack, NA; Cherkasov, A J Med Chem 64: 14968-14982 (2021)
- Jones, CD; Blaszczak, LC; Goettel, ME; Suarez, T; Crowell, TA; Mabry, TE; Ruenitz, PC; Srivatsan, V J Med Chem 35: 931-8 (1992)
- Boehm, MF; McClurg, MR; Pathirana, C; Mangelsdorf, D; White, SK; Hebert, J; Winn, D; Goldman, ME; Heyman, RA J Med Chem 37: 408-14 (1994)
- Louvet, P; Schweizer, D; Gourdel, ME; Riguet, E; Yue, C; Marcy, VR; Lin, YG; Gruner, J; Lesur, B; Bacon, ER; Chatterjee, S Eur J Med Chem 54: 949-51 (2012)
- Wagner, CE; Jurutka, PW; Marshall, PA; Groy, TL; van der Vaart, A; Ziller, JW; Furmick, JK; Graeber, ME; Matro, E; Miguel, BV; Tran, IT; Kwon, J; Tedeschi, JN; Moosavi, S; Danishyar, A; Philp, JS; Khamees, RO; Jackson, JN; Grupe, DK; Badshah, SL; Hart, JW J Med Chem 52: 5950-66 (2009)
- Hill, T; Odell, LR; Edwards, JK; Graham, ME; McGeachie, AB; Rusak, J; Quan, A; Abagyan, R; Scott, JL; Robinson, PJ; McCluskey, A J Med Chem 48: 7781-8 (2005)
- Pettersson, M; Johnson, DS; Subramanyam, C; Bales, KR; am Ende, CW; Fish, BA; Green, ME; Kauffman, GW; Mullins, PB; Navaratnam, T; Sakya, SM; Stiff, CM; Tran, TP; Xie, L; Zhang, L; Pustilnik, LR; Vetelino, BC; Wood, KM; Pozdnyakov, N; Verhoest, PR; O'Donnell, CJ J Med Chem 57: 1046-62 (2014)
- Grimes ME
- Sun, S; Jia, Q; Zenova, AY; Chafeev, M; Zhang, Z; Lin, S; Kwan, R; Grimwood, ME; Chowdhury, S; Young, C; Cohen, CJ; Oballa, RM Bioorg Med Chem Lett 24: 4397-401 (2014)
- Jacobs, MR; Olivero, JE; Ok Choi, H; Liao, CP; Kashemirov, BA; Katz, JE; Gross, ME; McKenna, CE Bioorg Med Chem 92: (2023)
- Daher, R; Coinçon, M; Fonvielle, M; Gest, PM; Guerin, ME; Jackson, M; Sygusch, J; Therisod, M J Med Chem 53: 7836-42 (2010)
- Thurmond, J; Butchbach, ME; Palomo, M; Pease, B; Rao, M; Bedell, L; Keyvan, M; Pai, G; Mishra, R; Haraldsson, M; Andresson, T; Bragason, G; Thosteinsdottir, M; Bjornsson, JM; Coovert, DD; Burghes, AH; Gurney, ME; Singh, J J Med Chem 51: 449-69 (2008)
- Han, G; Haskell-Luevano, C; Kendall, L; Bonner, G; Hadley, ME; Cone, RD; Hruby, VJ J Med Chem 47: 1514-26 (2004)
- Allen, MP; Blake, JF; Bryce, DK; Haggan, ME; Liras, S; McLean, S; Segelstein, BE Bioorg Med Chem Lett 10: 523-6 (2000)
- Millen, J; Riley, TN; Waters, IW; Hamrick, ME J Med Chem 28: 12-7 (1985)
- Huff, SE; Mohammed, FA; Yang, M; Agrawal, P; Pink, J; Harris, ME; Dealwis, CG; Viswanathan, R J Med Chem 61: 666-680 (2018)
- Hart, ME; Suchland, KL; Miyakawa, M; Bunzow, JR; Grandy, DK; Scanlan, TS J Med Chem 49: 1101-12 (2006)
- Maggiora, L; Chang, CT; Hasson, ME; Bigge, CF; Mertes, MP J Med Chem 26: 1028-36 (1983)
- Su, BN; Cuendet, M; Hawthorne, ME; Kardono, LB; Riswan, S; Fong, HH; Mehta, RG; Pezzuto, JM; Kinghorn, AD J Nat Prod 65: 163-9 (2002)
- Hayes, ME; Breinlinger, EC; Wallace, GA; Grongsaard, P; Miao, W; McPherson, MJ; Stoffel, RH; Green, DW; Roth, GP Bioorg Med Chem Lett 18: 2414-9 (2008)
- Hegazy, ME; El-Hamd H Mohamed, A; El-Halawany, AM; Djemgou, PC; Shahat, AA; Paré, PW J Nat Prod 74: 937-42 (2011)
- Snyder, KR; Story, SC; Heidt, ME; Murray, TF; DeLander, GE; Aldrich, JV J Med Chem 35: 4330-3 (1992)
- Deng, JZ; Starck, SR; Hecht, SM; Ijames, CF; Hemling, ME J Nat Prod 62: 1000-2 (1999)
- Jerome, KD; Hepperle, ME; Walker, JK; Xing, L; Devraj, RV; Benson, AG; Baldus, JE; Selness, SR Bioorg Med Chem Lett 20: 3146-9 (2010)
- Mayer, SC; Kreft, AF; Harrison, B; Abou-Gharbia, M; Antane, M; Aschmies, S; Atchison, K; Chlenov, M; Cole, DC; Comery, T; Diamantidis, G; Ellingboe, J; Fan, K; Galante, R; Gonzales, C; Ho, DM; Hoke, ME; Hu, Y; Huryn, D; Jain, U; Jin, M; Kremer, K; Kubrak, D; Lin, M; Lu, P; Magolda, R; Martone, R; Moore, W; Oganesian, A; Pangalos, MN; Porte, A; Reinhart, P; Resnick, L; Riddell, DR; Sonnenberg-Reines, J; Stock, JR; Sun, SC; Wagner, E; Wang, T; Woller, K; Xu, Z; Zaleska, MM; Zeldis, J; Zhang, M; Zhou, H; Jacobsen, JS J Med Chem 51: 7348-51 (2008)
- Sams, AG; Mikkelsen, GK; Larsen, M; Langgård, M; Howells, ME; Schrøder, TJ; Brennum, LT; Torup, L; Jørgensen, EB; Bundgaard, C; Kreilgård, M; Bang-Andersen, B J Med Chem 54: 751-64 (2012)
- Fast, W; Huff, ME; Silverman, RB Bioorg Med Chem Lett 7: 1449-1454 (1997)
- LEE, K; DUGGIRALA, KB; CHOI, GD; CHAE, CH; JUNG, ME; LEE, Y; CHO, BC US Patent US20240343694 (2024)
- Jacobs ME
- Jimenez, ME; Bush, K; Pawlik, J; Sower, L; Peterson, JW; Gilbertson, SR Bioorg Med Chem Lett 18: 4215-8 (2008)
- Wu, J; Vaid, TM; Kim, H; Lu, J; Li, M; Fung, LW; Johnson, ME US Patent US20250059159 (2025)
- Knutsen, LJ; Lau, J; Petersen, H; Thomsen, C; Weis, JU; Shalmi, M; Judge, ME; Hansen, AJ; Sheardown, MJ J Med Chem 42: 3463-77 (1999)
- Kang, SY; Park, EJ; Park, WK; Kim, HJ; Choi, G; Jung, ME; Seo, HJ; Kim, MJ; Pae, AN; Kim, J; Lee, J Bioorg Med Chem 18: 6156-69 (2010)
- Smith, RA; Barbosa, J; Blum, CL; Bobko, MA; Caringal, YV; Dally, R; Johnson, JS; Katz, ME; Kennure, N; Kingery-Wood, J; Lee, W; Lowinger, TB; Lyons, J; Marsh, V; Rogers, DH; Swartz, S; Walling, T; Wild, H Bioorg Med Chem Lett 11: 2775-8 (2001)
- Kavanagh, ME; Chenge, J; Zoufir, A; McLean, KJ; Coyne, AG; Bender, A; Munro, AW; Abell, C Biochemistry 56: 1559-1572 (2017)
- Bock, MG; DiPardo, RM; Rittle, KE; Evans, BE; Freidinger, RM; Veber, DF; Chang, RS; Chen, TB; Keegan, ME; Lotti, VJ J Med Chem 29: 1941-5 (1986)
- Cumming, JN; Smith, EM; Wang, L; Misiaszek, J; Durkin, J; Pan, J; Iserloh, U; Wu, Y; Zhu, Z; Strickland, C; Voigt, J; Chen, X; Kennedy, ME; Kuvelkar, R; Hyde, LA; Cox, K; Favreau, L; Czarniecki, MF; Greenlee, WJ; McKittrick, BA; Parker, EM; Stamford, AW Bioorg Med Chem Lett 22: 2444-9 (2012)
- Newton, E; Starcovic, SA; Menze, M; Konkle, ME; Long, TE; Hazlehurst, LA; Huber, JD; Robart, AR; Geldenhuys, WJ Bioorg Med Chem Lett 89: (2023)
- Clapham, B; Cox, PB; Dart, MJ; Gomtsyan, A; Jinkerson, TK; Keddy, RG; Kort, ME; Kym, PR; Matulenko, M; Schmidt, RG; Villamil, CI; Voight, EA; Woller, KR US Patent US9012651 (2015)
- Kuehne, ME; He, L; Jokiel, PA; Pace, CJ; Fleck, MW; Maisonneuve, IM; Glick, SD; Bidlack, JM J Med Chem 46: 2716-30 (2003)
- Zheng, W; Padia, J; Urban, DJ; Jadhav, A; Goker-Alpan, O; Simeonov, A; Goldin, E; Auld, D; LaMarca, ME; Inglese, J; Austin, CP; Sidransky, E Proc Natl Acad Sci U S A 104: 13192-7 (2007)
- Ward, YD; Thomson, DS; Frye, LL; Cywin, CL; Morwick, T; Emmanuel, MJ; Zindell, R; McNeil, D; Bekkali, Y; Girardot, M; Hrapchak, M; DeTuri, M; Crane, K; White, D; Pav, S; Wang, Y; Hao, MH; Grygon, CA; Labadia, ME; Freeman, DM; Davidson, W; Hopkins, JL; Brown, ML; Spero, DM; Giradot, M J Med Chem 45: 5471-82 (2002)
- Wilkinson, RA; Pincus, SH; Song, K; Shepard, JB; Weaver, AJ; Labib, ME; Teintze, M Bioorg Med Chem Lett 23: 2197-201 (2013)
- Haadsma-Svensson, SR; Cleek, KA; Dinh, DM; Duncan, JN; Haber, CL; Huff, RM; Lajiness, ME; Nichols, NF; Smith, MW; Svensson, KA; Zaya, MJ; Carlsson, A; Lin, CH J Med Chem 44: 4716-32 (2001)
- Reiter, LA; Robinson, RP; McClure, KF; Jones, CS; Reese, MR; Mitchell, PG; Otterness, IG; Bliven, ML; Liras, J; Cortina, SR; Donahue, KM; Eskra, JD; Griffiths, RJ; Lame, ME; Lopez-Anaya, A; Martinelli, GJ; McGahee, SM; Yocum, SA; Lopresti-Morrow, LL; Tobiassen, LM; Vaughn-Bowser, ML Bioorg Med Chem Lett 14: 3389-95 (2004)
- Uehling, DE; Shearer, BG; Donaldson, KH; Chao, EY; Deaton, DN; Adkison, KK; Brown, KK; Cariello, NF; Faison, WL; Lancaster, ME; Lin, J; Hart, R; Milliken, TO; Paulik, MA; Sherman, BW; Sugg, EE; Cowan, C J Med Chem 49: 2758-71 (2006)
- Jung, KY; Wang, H; Teriete, P; Yap, JL; Chen, L; Lanning, ME; Hu, A; Lambert, LJ; Holien, T; Sundan, A; Cosford, ND; Prochownik, EV; Fletcher, S J Med Chem 58: 3002-24 (2015)
- Wu, Z; Yang, C; Graham, TH; Verras, A; Chabin, RM; Xu, S; Tong, X; Xie, D; Lassman, ME; Bhatt, UR; Garcia-Calvo, MM; Shen, Z; Chen, Q; Bleasby, K; Sinharoy, R; Hale, JJ; Tata, JR; Pinto, S; Colletti, SL; Shen, DM Bioorg Med Chem Lett 22: 1727-30 (2012)
- McDonald, IA; Nyce, PL; Muench, DM; Gates, CA; Blohm, TR; Laughlin, ME; Weintruab, PM Bioorg Med Chem Lett 4: 847-851 (1994)
- Shi, Q; Canada, EJ; Xu, Y; Warshawsky, AM; Etgen, GJ; Broderick, CL; Clutinger, CK; Irwin, LA; Laurila, ME; Montrose-Rafizadeh, C; Oldham, BA; Wang, M; Winneroski, LL; Xie, C; York, JS; Yumibe, NP; Zink, RW; Mantlo, N Bioorg Med Chem Lett 17: 6744-9 (2008)
- Layton, ME; Kern, JC; Hartingh, TJ; Shipe, WD; Raheem, I; Kandebo, M; Hayes, RP; Huszar, S; Eddins, D; Ma, B; Fuerst, J; Wollenberg, GK; Li, J; Fritzen, J; McGaughey, GB; Uslaner, JM; Smith, SM; Coleman, PJ; Cox, CD J Med Chem 66: 1157-1171 (2023)
- Xu, YC; Johnson, KW; Phebus, LA; Cohen, M; Nelson, DL; Schenck, K; Walker, CD; Fritz, JE; Kaldor, SW; LeTourneau, ME; Murff, RE; Zgombick, JM; Calligaro, DO; Audia, JE; Schaus, JM J Med Chem 44: 4031-4 (2001)
- Powell, DA; Ramtohul, Y; Lebrun, ME; Oballa, R; Bhat, S; Falgueyret, JP; Guiral, S; Huang, Z; Skorey, K; Tawa, P; Zhang, L Bioorg Med Chem Lett 20: 6366-9 (2010)
- Szychowski, J; Papp, R; Dietrich, E; Liu, B; Vallée, F; Leclaire, ME; Fourtounis, J; Martino, G; Perryman, AL; Pau, V; Yin, SY; Mader, P; Roulston, A; Truchon, JF; Marshall, CG; Diallo, M; Duffy, NM; Stocco, R; Godbout, C; Bonneau-Fortin, A; Kryczka, R; Bhaskaran, V; Mao, D; Orlicky, S; Beaulieu, P; Turcotte, P; Kurinov, I; Sicheri, F; Mamane, Y; Gallant, M; Black, WC J Med Chem 65: 10251-10284 (2022)
- Boschelli, DH; Kramer, JB; Connor, DT; Lesch, ME; Schrier, DJ; Ferin, MA; Wright, CD J Med Chem 37: 717-8 (1994)
- Zhang, CH; Spasov, KA; Reilly, RA; Hollander, K; Stone, EA; Ippolito, JA; Liosi, ME; Deshmukh, MG; Tirado-Rives, J; Zhang, S; Liang, Z; Miller, SJ; Isaacs, F; Lindenbach, BD; Anderson, KS; Jorgensen, WL ACS Med Chem Lett 12: 1325-1332 (2021)
- Nikolovska-Coleska, Z; Xu, L; Hu, Z; Tomita, Y; Li, P; Roller, PP; Wang, R; Fang, X; Guo, R; Zhang, M; Lippman, ME; Yang, D; Wang, S J Med Chem 47: 2430-40 (2004)
- Shuttleworth, SJ; Lizarzaburu, ME; Chai, A; Coward, P Bioorg Med Chem Lett 14: 3037-42 (2004)
- Venepalli, BR; Aimone, LD; Appell, KC; Bell, MR; Dority, JA; Goswami, R; Hall, PL; Kumar, V; Lawrence, KB; Logan, ME J Med Chem 35: 374-8 (1992)
- Zimmermann, TJ; Niesen, FH; Pilka, ES; Knapp, S; Oppermann, U; Maier, ME Bioorg Med Chem 17: 530-6 (2009)
- Zerfas, BL; Maresh, ME; Trader, DJ J Med Chem 63: 1841-1858 (2020)
- Artico, M; Di Santo, R; Costi, R; Novellino, E; Greco, G; Massa, S; Tramontano, E; Marongiu, ME; De Montis, A; La Colla, P J Med Chem 41: 3948-60 (1998)
- Baumhover, NJ; Martin, ME; Parameswarappa, SG; Kloepping, KC; O'Dorisio, MS; Pigge, FC; Schultz, MK Bioorg Med Chem Lett 21: 5757-61 (2011)
- Gomez, L; Massari, ME; Vickers, T; Freestone, G; Vernier, W; Ly, K; Xu, R; McCarrick, M; Marrone, T; Metz, M; Yan, YG; Yoder, ZW; Lemus, R; Broadbent, NJ; Barido, R; Warren, N; Schmelzer, K; Neul, D; Lee, D; Andersen, CB; Sebring, K; Aertgeerts, K; Zhou, X; Tabatabaei, A; Peters, M; Breitenbucher, JG J Med Chem 60: 2037-2051 (2017)
- Allen, JG; Bourbeau, MP; Wohlhieter, GE; Bartberger, MD; Michelsen, K; Hungate, R; Gadwood, RC; Gaston, RD; Evans, B; Mann, LW; Matison, ME; Schneider, S; Huang, X; Yu, D; Andrews, PS; Reichelt, A; Long, AM; Yakowec, P; Yang, EY; Lee, TA; Oliner, JD J Med Chem 52: 7044-53 (2009)
- Mattmann, ME; Geske, GD; Worzalla, GA; Chandler, JR; Sappington, KJ; Greenberg, EP; Blackwell, HE Bioorg Med Chem Lett 18: 3072-5 (2008)
- Matyskiela, ME; Zhang, W; Man, HW; Muller, G; Khambatta, G; Baculi, F; Hickman, M; LeBrun, L; Pagarigan, B; Carmel, G; Lu, CC; Lu, G; Riley, M; Satoh, Y; Schafer, P; Daniel, TO; Carmichael, J; Cathers, BE; Chamberlain, PP J Med Chem 61: 535-542 (2017)
- Zhong, W; Pasunooti, KK; Balamkundu, S; Wong, YH; Nah, Q; Gadi, V; Gnanakalai, S; Chionh, YH; McBee, ME; Gopal, P; Lim, SH; Olivier, N; Buurman, ET; Dick, T; Liu, CF; Lescar, J; Dedon, PC J Med Chem 62: 7788-7805 (2019)
- Shen, DM; Brady, EJ; Candelore, MR; Dallas-Yang, Q; Ding, VD; Feeney, WP; Jiang, G; McCann, ME; Mock, S; Qureshi, SA; Saperstein, R; Shen, X; Tong, X; Tota, LM; Wright, MJ; Yang, X; Zheng, S; Chapman, KT; Zhang, BB; Tata, JR; Parmee, ER Bioorg Med Chem Lett 21: 76-81 (2010)
- Gleason, JG; Hall, RF; Perchonock, CD; Erhard, KF; Frazee, JS; Ku, TW; Kondrad, K; McCarthy, ME; Mong, S; Crooke, ST J Med Chem 30: 959-61 (1987)
- Reitz, AB; Baxter, EW; Codd, EE; Davis, CB; Jordan, AD; Maryanoff, BE; Maryanoff, CA; McDonnell, ME; Powell, ET; Renzi, MJ; Schott, MR; Scott, MK; Shank, RP; Vaught, JL J Med Chem 41: 1997-2009 (1998)
- Katz, BA; Luong, C; Ho, JD; Somoza, JR; Gjerstad, E; Tang, J; Williams, SR; Verner, E; Mackman, RL; Young, WB; Sprengeler, PA; Chan, H; Mortara, K; Janc, JW; McGrath, ME J Mol Biol 344: 527-47 (2004)
- Mainolfi, N; Powers, J; Amin, J; Long, D; Lee, W; McLaughlin, ME; Jaffee, B; Brain, C; Elliott, J; Sivak, JM J Med Chem 56: 5464-72 (2013)
- Mertzman, ME; Dzierba, CD; Guernon, JM; Hart, AC; Luo, G; Macor, JE; Pitts, WJ; Shi, J; Spergel, SH US Patent US11440913 (2022)
- Xu, S; Sun, L; Dick, A; Zalloum, WA; Huang, T; Meuser, ME; Zhang, X; Tao, Y; Cherukupalli, S; Ding, D; Ding, X; Gao, S; Jiang, X; Kang, D; De Clercq, E; Pannecouque, C; Cocklin, S; Liu, X; Zhan, P Eur J Med Chem 227: (2022)
- Meyer, ME; Doshi, A; Polgar, WE; Zaveri, NT Bioorg Med Chem 92: (2023)
- Parker, MH; Smith-Swintosky, VL; McComsey, DF; Huang, Y; Brenneman, D; Klein, B; Malatynska, E; White, HS; Milewski, ME; Herb, M; Finley, MF; Liu, Y; Lubin, ML; Qin, N; Iannucci, R; Leclercq, L; Cuyckens, F; Reitz, AB; Maryanoff, BE J Med Chem 52: 7528-36 (2009)
- Blevitt, JM; Hack, MD; Herman, KL; Jackson, PF; Krawczuk, PJ; Lebsack, AD; Liu, AX; Mirzadegan, T; Nelen, MI; Patrick, AN; Steinbacher, S; Milla, ME; Lumb, KJ J Med Chem 60: 3511-3517 (2017)
- Million, ME; Boiziau, J; Parker, F; Tocque, B; Roques, BP; Garbay, C J Med Chem 38: 4693-703 (1995)
- Kim, HY; Sohn, J; Wijewickrama, GT; Edirisinghe, P; Gherezghiher, T; Hemachandra, M; Lu, PY; Chandrasena, RE; Molloy, ME; Tonetti, DA; Thatcher, GR Bioorg Med Chem 18: 809-21 (2010)
- Monteiro, ME; Lechuga, G; Lara, LS; Souto, BA; Viganó, MG; Bourguignon, SC; Calvet, CM; Oliveira, FOR; Alves, CR; Souza-Silva, F; Santos, MS; Pereira, MCS Eur J Med Chem 182: (2019)
- Ortega, MA; Montoya, ME; Zarranz, B; Jaso, A; Aldana, I; Leclerc, S; Meijer, L; Monge, A Bioorg Med Chem 10: 2177-84 (2002)
- Morgan ME
- Hopper, AT; Juhl, M; Hornberg, J; Badolo, L; Kilburn, JP; Thougaard, A; Smagin, G; Song, D; Calice, L; Menon, V; Dale, E; Zhang, H; Cajina, M; Nattini, ME; Gandhi, A; Grenon, M; Jones, K; Khayrullina, T; Chandrasena, G; Thomsen, C; Zorn, SH; Brodbeck, R; Poda, SB; Staal, R; Möller, T J Med Chem 64: 4891-4902 (2021)
- Averina, EB; Vasilenko, DA; Gracheva, YA; Grishin, YK; Radchenko, EV; Burmistrov, VV; Butov, GM; Neganova, ME; Serkova, TP; Redkozubova, OM; Shevtsova, EF; Milaeva, ER; Kuznetsova, TS; Zefirov, NS Bioorg Med Chem 24: 712-20 (2016)
- Babaoglu, K; Simeonov, A; Irwin, JJ; Nelson, ME; Feng, B; Thomas, CJ; Cancian, L; Costi, MP; Maltby, DA; Jadhav, A; Inglese, J; Austin, CP; Shoichet, BK J Med Chem 51: 2502-11 (2008)
- Morisseau, C; Pakhomova, S; Hwang, SH; Newcomer, ME; Hammock, BD Bioorg Med Chem Lett 23: 3818-21 (2013)
- Macor, JE; Burkhart, CA; Heym, JH; Ives, JL; Lebel, LA; Newman, ME; Nielsen, JA; Ryan, K; Schulz, DW; Torgersen, LK J Med Chem 33: 2087-93 (1990)
- Carbain, B; Paterson, DJ; Anscombe, E; Campbell, AJ; Cano, C; Echalier, A; Endicott, JA; Golding, BT; Haggerty, K; Hardcastle, IR; Jewsbury, PJ; Newell, DR; Noble, ME; Roche, C; Wang, LZ; Griffin, RJ J Med Chem 57: 56-70 (2014)
- Hancock, AA; Bennani, YL; Bush, EN; Esbenshade, TA; Faghih, R; Fox, GB; Jacobson, P; Knourek-Segel, V; Krueger, KM; Nuss, ME; Pan, JB; Shapiro, R; Witte, DG; Yao, BB Eur J Pharmacol 487: 183-97 (2004)
- Lee, D; Long, SA; Murray, JH; Adams, JL; Nuttall, ME; Nadeau, DP; Kikly, K; Winkler, JD; Sung, CM; Ryan, MD; Levy, MA; Keller, PM; DeWolf, WE J Med Chem 44: 2015-26 (2001)
- Charrier, JD; Durrant, SJ; Golec, JM; Kay, DP; Knegtel, RM; MacCormick, S; Mortimore, M; O'Donnell, ME; Pinder, JL; Reaper, PM; Rutherford, AP; Wang, PS; Young, SC; Pollard, JR J Med Chem 54: 2320-30 (2011)
- Olah, ME; Gallo-Rodriguez, C; Jacobson, KA; Stiles, GL Mol Pharmacol 45: 978-82 (1994)
- Olson, ME; Abate-Pella, D; Perkins, AL; Li, M; Carpenter, MA; Rathore, A; Harris, RS; Harki, DA J Med Chem 58: 7419-30 (2015)
- Reitz, AB; Baxter, EW; Bennett, DJ; Codd, EE; Jordan, AD; Malloy, EA; Maryanoff, BE; McDonnell, ME; Ortegon, ME; Renzi, MJ J Med Chem 38: 4211-22 (1995)
- Hoorens, MWH; Ourailidou, ME; Rodat, T; van der Wouden, PE; Kobauri, P; Kriegs, M; Peifer, C; Feringa, BL; Dekker, FJ; Szymanski, W Eur J Med Chem 179: 133-146 (2019)
- Blois, J; Yuan, H; Smith, A; Pacold, ME; Weissleder, R; Cantley, LC; Josephson, L J Med Chem 51: 4699-707 (2008)
- Leach, CA; Brown, TH; Ife, RJ; Keeling, DJ; Laing, SM; Parsons, ME; Price, CA; Wiggall, KJ J Med Chem 35: 1845-52 (1992)
- Cockerill, GS; Angell, RM; Bedernjak, A; Chuckowree, I; Fraser, I; Gascon-Simorte, J; Gilman, MSA; Good, JAD; Harland, R; Johnson, SM; Ludes-Meyers, JH; Littler, E; Lumley, J; Lunn, G; Mathews, N; McLellan, JS; Paradowski, M; Peeples, ME; Scott, C; Tait, D; Taylor, G; Thom, M; Thomas, E; Villalonga Barber, C; Ward, SE; Watterson, D; Williams, G; Young, P; Powell, K J Med Chem 64: 3658-3676 (2021)
- Maillard, MC; Perlman, ME; Amitay, O; Baxter, D; Berlove, D; Connaughton, S; Fischer, JB; Guo, JQ; Hu, LY; McBurney, RN; Nagy, PI; Subbarao, K; Yost, EA; Zhang, L; Durant, GJ J Med Chem 41: 3048-61 (1998)
- Brant, MG; Garnett, GAE; Guedia, J; Lasalle, M; Lawn, S; Petersen, ME; Duan, R; Mendez-Campos, J; Hirkala-Schaefer, T; Winters, GC; Barnscher, SD Bioorg Med Chem Lett 91: (2023)
- Hopkins, CR; O'neil, SV; Laufersweiler, MC; Wang, Y; Pokross, M; Mekel, M; Evdokimov, A; Walter, R; Kontoyianni, M; Petrey, ME; Sabatakos, G; Roesgen, JT; Richardson, E; Demuth, TP Bioorg Med Chem Lett 16: 5659-63 (2006)
- Murphy, JM; Armijo, AL; Nomme, J; Lee, CH; Smith, QA; Li, Z; Campbell, DO; Liao, HI; Nathanson, DA; Austin, WR; Lee, JT; Darvish, R; Wei, L; Wang, J; Su, Y; Damoiseaux, R; Sadeghi, S; Phelps, ME; Herschman, HR; Czernin, J; Alexandrova, AN; Jung, ME; Lavie, A; Radu, CG J Med Chem 56: 6696-708 (2013)
- Carini, DJ; Duncia, JV; Aldrich, PE; Chiu, AT; Johnson, AL; Pierce, ME; Price, WA; Santella, JB; Wells, GJ; Wexler, RR J Med Chem 34: 2525-47 (1991)
- Pierson, ME; Comstock, JM; Simmons, RD; Julien, R; Kaiser, F; Rosamond, JD J Med Chem 43: 2350-5 (2000)
- Teng, M; Duong, TT; Klein, ES; Pino, ME; Chandraratna, RA J Med Chem 39: 3035-8 (1996)
- Klopfenstein, SR; Evdokimov, AG; Colson, AO; Fairweather, NT; Neuman, JJ; Maier, MB; Gray, JL; Gerwe, GS; Stake, GE; Howard, BW; Farmer, JA; Pokross, ME; Downs, TR; Kasibhatla, B; Peters, KG Bioorg Med Chem Lett 16: 1574-8 (2006)
- Arabaci, G; Yi, T; Fu, H; Porter, ME; Beebe, KD; Pei, D Bioorg Med Chem Lett 12: 3047-50 (2002)
- Plescia, J; Hédou, D; Pousse, ME; Labarre, A; Dufresne, C; Mittermaier, A; Moitessier, N Eur J Med Chem 240: (2022)
- Harris, DA; Powers, ME; Romesberg, FE Bioorg Med Chem Lett 19: 3787-90 (2009)
- Minassi, A; Rogati, F; Cruz, C; Prados, ME; Galera, N; Jinénez, C; Appendino, G; Bellido, ML; Calzado, MA; Caprioglio, D; Muñoz, E J Nat Prod 81: 2235-2243 (2018)
- Prime, ME; Brookfield, FA; Courtney, SM; Gaines, S; Marston, RW; Ichihara, O; Li, M; Vaidya, D; Williams, H; Pedret-Dunn, A; Reed, L; Schaertl, S; Toledo-Sherman, L; Beconi, M; Macdonald, D; Muñoz-Sanjuan, I; Dominguez, C; Wityak, J ACS Med Chem Lett 3: 731-735 (2012)
- Lacivita, E; Niso, M; Stama, ML; Arzuaga, A; Altamura, C; Costa, L; Desaphy, JF; Ragozzino, ME; Ciranna, L; Leopoldo, M Eur J Med Chem 199: (2020)
- Obeng, S; Kamble, SH; Reeves, ME; Restrepo, LF; Patel, A; Behnke, M; Chear, NJ; Ramanathan, S; Sharma, A; León, F; Hiranita, T; Avery, BA; McMahon, LR; McCurdy, CR J Med Chem 63: 433-439 (2020)
- Toms, NJ; Reid, ME; Phillips, W; Kemp, MC; Roberts, PJ Neuropharmacology 36: 1483-8 (1997)
- Sensfuss, U; Kruse, T; Skyggebjerg, RB; Uldam, HK; Vestergaard, B; Huus, K; Vinther, TN; Reinau, ME; Schéele, S; Clausen, TR J Med Chem 62: 1407-1419 (2019)
- Brown, DA; Kharkar, PS; Parrington, I; Reith, ME; Dutta, AK J Med Chem 51: 7806-19 (2008)
- Rawson, TE; Somers, TC; Marsters, JC; Wan, DT; Reynolds, ME; Burdick, DJ Bioorg Med Chem Lett 5: 1335-1338 (1995)
- Zhang, M; Bailey, DL; Bastian, JA; Briggs, SL; Chirgadze, NY; Clawson, DK; Denney, ML; Gifford-Moore, DS; Harper, RW; Johnson, LM; Klimkowski, VJ; Kohn, TJ; Lin, HS; McCowan, JR; Richett, ME; Sall, DJ; Smith, AJ; Smith, GF; Snyder, DW; Takeuchi, K; Utterback, BG; Yan, SC Bioorg Med Chem Lett 9: 775-80 (1999)
- Raviña, E; Negreira, J; Cid, J; Masaguer, CF; Rosa, E; Rivas, ME; Fontenla, JA; Loza, MI; Tristán, H; Cadavid, MI; Sanz, F; Lozoya, E; Carotti, A; Carrieri, A J Med Chem 42: 2774-97 (1999)
- Sestito, S; Bacci, A; Chiarugi, S; Runfola, M; Gado, F; Margheritis, E; Gul, S; Riveiro, ME; Vazquez, R; Huguet, S; Manera, C; Rezai, K; Garau, G; Rapposelli, S Eur J Med Chem 226: (2021)
- Valdameri, G; Genoux-Bastide, E; Peres, B; Gauthier, C; Guitton, J; Terreux, R; Winnischofer, SM; Rocha, ME; Boumendjel, A; Di Pietro, A J Med Chem 55: 966-70 (2012)
- Fell, JB; Fischer, JP; Baer, BR; Blake, JF; Bouhana, K; Briere, DM; Brown, KD; Burgess, LE; Burns, AC; Burkard, MR; Chiang, H; Chicarelli, MJ; Cook, AW; Gaudino, JJ; Hallin, J; Hanson, L; Hartley, DP; Hicken, EJ; Hingorani, GP; Hinklin, RJ; Mejia, MJ; Olson, P; Otten, JN; Rhodes, SP; Rodriguez, ME; Savechenkov, P; Smith, DJ; Sudhakar, N; Sullivan, FX; Tang, TP; Vigers, GP; Wollenberg, L; Christensen, JG; Marx, MA J Med Chem 63: 6679-6693 (2020)
- Rogers, ME; Wilkinson, DS; Thweatt, JR; Halenda, SP J Med Chem 23: 688-90 (1980)
- Guo, H; Hathaway, H; Royce, ME; Prossnitz, ER; Miao, Y Bioorg Med Chem Lett 23: 5484-7 (2013)
- Coppola, GM; Zhang, YL; Schuster, HF; Russell, ME; Hughes, TE Bioorg Med Chem Lett 10: 1555-8 (2000)
- Chen, Z; Kim, SH; Barbosa, SA; Huynh, T; Tortolani, DR; Leavitt, KJ; Wei, DD; Manne, V; Ricca, CS; Gullo-Brown, J; Poss, MA; Vaccaro, W; Salvati, ME Bioorg Med Chem Lett 16: 628-32 (2005)
- Wang, H; Ruan, Z; Li, JJ; Simpkins, LM; Smirk, RA; Wu, SC; Hutchins, RD; Nirschl, DS; Van Kirk, K; Cooper, CB; Sutton, JC; Ma, Z; Golla, R; Seethala, R; Salyan, ME; Nayeem, A; Krystek, SR; Sheriff, S; Camac, DM; Morin, PE; Carpenter, B; Robl, JA; Zahler, R; Gordon, DA; Hamann, LG Bioorg Med Chem Lett 18: 3168-72 (2008)
- Alvarez, F; Ghérardi, A; Nebois, P; Sarciron, ME; Pétavy, AF; Walchshofer, N Bioorg Med Chem Lett 12: 977-9 (2002)
- Zhang, L; Schaner, ME; Giacomini, KM J Pharmacol Exp Ther 286: 354-61 (1998)
- Fernández-Bachiller, MI; Hwang, S; Schembri, ME; Lindemann, P; Guberman, M; Herziger, S; Specker, E; Matter, H; Will, DW; Czech, J; Wagner, M; Bauer, A; Schreuder, H; Ritter, K; Urmann, M; Wehner, V; Sun, H; Nazaré, M J Med Chem 65: 13013-13028 (2022)
- Schnute, ME US Patent US9920054 (2018)
- Huryn, DM; Wipf, P; Grandis, JR; LaPorte, MG; Johnston, PA; Schurdak, ME; Colombo, R US Patent US10618914 (2020)
- Scott, ME; Guerin, D; Molinari, D; Kattar, S; Fuller, P; Dinsmore, C; Kong, N; Bai, Y; Fu, J; Liu, Y; Zheng, Z US Patent US10072025 (2018)
- Sridhar, J; Sfondouris, ME; Bratton, MR; Nguyen, TL; Townley, I; Klein Stevens, CL; Jones, FE Bioorg Med Chem Lett 24: 126-31 (2014)
- Byun, DH; Cai, ZR; Canales, EY; Debien, LP; Hansen, TR; Huang, R; Jansa, P; Lee, RA; Loyer-Drew, JA; McFadden, R; Mitchell, ML; Pyun, H; Saito, RD; Sangi, MS; Schrier, AJ; Shatskikh, ME; Taylor, JG; Van Veldhuizen, JJ; Xu, L US Patent US11878965 (2024)
- Buck, IM; Black, JW; Cooke, T; Dunstone, DJ; Gaffen, JD; Griffin, EP; Harper, EA; Hull, RA; Kalindjian, SB; Lilley, EJ; Linney, ID; Low, CM; McDonald, IM; Pether, MJ; Roberts, SP; Shankley, NP; Shaxted, ME; Steel, KI; Sykes, DA; Tozer, MJ; Watt, GF; Walker, MK; Wright, L; Wright, PT J Med Chem 48: 6803-12 (2005)
- Soltan, OM; Shoman, ME; Abdel-Aziz, SA; Narumi, A; Konno, H; Abdel-Aziz, M Eur J Med Chem 225: (2021)
- Liu, JJ; Dermatakis, A; Lukacs, C; Konzelmann, F; Chen, Y; Kammlott, U; Depinto, W; Yang, H; Yin, X; Chen, Y; Schutt, A; Simcox, ME; Luk, KC Bioorg Med Chem Lett 13: 2465-8 (2003)
- Huang, HC; Tremont, SJ; Lee, LF; Keller, BT; Carpenter, AJ; Wang, CC; Banerjee, SC; Both, SR; Fletcher, T; Garland, DJ; Huang, W; Jones, C; Koeller, KJ; Kolodziej, SA; Li, J; Manning, RE; Mahoney, MW; Miller, RE; Mischke, DA; Rath, NP; Reinhard, EJ; Tollefson, MB; Vernier, WF; Wagner, GM; Rapp, SR; Beaudry, J; Glenn, K; Regina, K; Schuh, JR; Smith, ME; Trivedi, JS; Reitz, DB J Med Chem 48: 5853-68 (2005)
- McNemar, C; Snow, ME; Windsor, WT; Prongay, A; Mui, P; Zhang, R; Durkin, J; Le, HV; Weber, PC Biochemistry 36: 10006-14 (1997)
- Chakraborti, AK; Gopalakrishnan, B; Sobhia, ME; Malde, A Bioorg Med Chem Lett 13: 2473-9 (2003)
- Nayak, BV; Ciftci-Yabanoglu, S; Bhakat, S; Timiri, AK; Sinha, BN; Ucar, G; Soliman, ME; Jayaprakash, V Bioorg Chem 58: 72-80 (2015)
- Gallagher, TF; Fier-Thompson, SM; Garigipati, RS; Sorenson, ME; Smietana, JM; Lee, D; Bender, PE; Lee, JC; Laydon, JT; Griswold, DE; Chabot-Fletcher, MC; Breton, JJ; Adams, JL Bioorg Med Chem Lett 5: 1171-1176 (1995)
- Pungitore, CR; Ayub, MJ; García, M; Borkowski, EJ; Sosa, ME; Ciuffo, G; Giordano, OS; Tonn, CE J Nat Prod 67: 357-61 (2004)
- Verdine, GL; Bowman, BR; Sowa, ME; Blodgett, JA; Robison, KE; Stiles, DT; Morgenstern, JP; Townson, SA; Shigdel, UK US Patent US11059830 (2021)
- Cheng, H; Orr, STM; Bailey, S; Brooun, A; Chen, P; Deal, JG; Deng, YL; Edwards, MP; Gallego, GM; Grodsky, N; Huang, B; Jalaie, M; Kaiser, S; Kania, RS; Kephart, SE; Lafontaine, J; Ornelas, MA; Pairish, M; Planken, S; Shen, H; Sutton, S; Zehnder, L; Almaden, CD; Bagrodia, S; Falk, MD; Gukasyan, HJ; Ho, C; Kang, X; Kosa, RE; Liu, L; Spilker, ME; Timofeevski, S; Visswanathan, R; Wang, Z; Meng, F; Ren, S; Shao, L; Xu, F; Kath, JC J Med Chem 64: 644-661 (2021)
- Ko, KS; Steffey, ME; Brandvold, KR; Soellner, MB ACS Med Chem Lett 4: 779-783 (2013)
- Soper, DL; Milbank, JB; Mieling, GE; Dirr, MJ; Kende, AS; Cooper, R; Jee, WS; Yao, W; Chen, JL; Bodman, M; Lundy, MW; De, B; Stella, ME; Ebetino, FH; Wang, Y; deLong, MA; Wos, JA J Med Chem 44: 4157-69 (2001)
- Park, HJ; Kim, YS; Kim, JS; Lee, EJ; Yi, YJ; Hwang, HJ; Suh, ME; Ryu, CK; Lee, SK Bioorg Med Chem Lett 14: 3385-8 (2004)
- Lis, R; Morgan, TK; DeVita, RJ; Davey, DD; Lumma, WC; Wohl, RA; Diamond, J; Wong, SS; Sullivan, ME J Med Chem 30: 696-704 (1987)
- Touaibia, M; Surette, ME US Patent US20240425441 (2024)
- Gleave, RJ; Beswick, PJ; Brown, AJ; Giblin, GM; Haslam, CP; Livermore, D; Moses, A; Nicholson, NH; Page, LW; Slingsby, B; Swarbrick, ME Bioorg Med Chem Lett 19: 6578-81 (2009)
- Liu, Y; Garnham, CP; Roll-Mecak, A; Tanner, ME Bioorg Med Chem Lett 23: 4408-12 (2013)
- Li, X; Chu, S; Feher, VA; Khalili, M; Nie, Z; Margosiak, S; Nikulin, V; Levin, J; Sprankle, KG; Tedder, ME; Almassy, R; Appelt, K; Yager, KM J Med Chem 46: 5663-73 (2003)
- Becker, GL; Sielaff, F; Than, ME; Lindberg, I; Routhier, S; Day, R; Lu, Y; Garten, W; Steinmetzer, T J Med Chem 53: 1067-75 (2010)
- Theoclitou, ME; Aquila, B; Block, MH; Brassil, PJ; Castriotta, L; Code, E; Collins, MP; Davies, AM; Deegan, T; Ezhuthachan, J; Filla, S; Freed, E; Hu, H; Huszar, D; Jayaraman, M; Lawson, D; Lewis, PM; Nadella, MV; Oza, V; Padmanilayam, M; Pontz, T; Ronco, L; Russell, D; Whitston, D; Zheng, X J Med Chem 54: 6734-50 (2011)
- Syrjänen, L; Tolvanen, ME; Hilvo, M; Vullo, D; Carta, F; Supuran, CT; Parkkila, S Bioorg Med Chem 21: 1516-21 (2013)
- Roberts, K; Ursini, A; Barnaby, R; Cassarà, PG; Corsi, M; Curotto, G; Donati, D; Feriani, A; Finizia, G; Marchioro, C; Niccolai, D; Oliosi, B; Polinelli, S; Ratti, E; Reggiani, A; Tedesco, G; Tranquillini, ME; Trist, DG; van Amsterdam, FT Bioorg Med Chem 19: 4257-73 (2011)
- He, S; Lai, Z; Ye, Z; Dobbelaar, PH; Shah, SK; Truong, Q; Du, W; Guo, L; Liu, J; Jian, T; Qi, H; Bakshi, RK; Hong, Q; Dellureficio, J; Reibarkh, M; Samuel, K; Reddy, VB; Mitelman, S; Tong, SX; Chicchi, GG; Tsao, KL; Trusca, D; Wu, M; Shao, Q; Trujillo, ME; Fernandez, G; Nelson, D; Bunting, P; Kerr, J; Fitzgerald, P; Morissette, P; Volksdorf, S; Eiermann, GJ; Li, C; Zhang, B; Howard, AD; Zhou, YP; Nargund, RP; Hagmann, WK ACS Med Chem Lett 5: 748-53 (2014)
- Zheng, GZ; Bhatia, P; Daanen, J; Kolasa, T; Patel, M; Latshaw, S; El Kouhen, OF; Chang, R; Uchic, ME; Miller, L; Nakane, M; Lehto, SG; Honore, MP; Moreland, RB; Brioni, JD; Stewart, AO J Med Chem 48: 7374-88 (2005)
- Obermoser, V; Urban, ME; Murgueitio, MS; Wolber, G; Kintscher, U; Gust, R Eur J Med Chem 124: 138-152 (2016)
- Reis, J; Cagide, F; Valencia, ME; Teixeira, J; Bagetta, D; Pérez, C; Uriarte, E; Oliveira, PJ; Ortuso, F; Alcaro, S; Rodríguez-Franco, MI; Borges, F Eur J Med Chem 158: 781-800 (2018)
- Cherney, RJ; Duan, JJ; Voss, ME; Chen, L; Wang, L; Meyer, DT; Wasserman, ZR; Hardman, KD; Liu, RQ; Covington, MB; Qian, M; Mandlekar, S; Christ, DD; Trzaskos, JM; Newton, RC; Magolda, RL; Wexler, RR; Decicco, CP J Med Chem 46: 1811-23 (2003)
- WENZLER ME
- Lovelace, ES; Armishaw, CJ; Colgrave, ML; Wahlstrom, ME; Alewood, PF; Daly, NL; Craik, DJ J Med Chem 49: 6561-8 (2006)
- Pengsuparp, T; Cai, L; Fong, HH; Kinghorn, AD; Pezzuto, JM; Wani, MC; Wall, ME J Nat Prod 57: 415-8 (1994)
- Picconi, P; Hind, CK; Nahar, KS; Jamshidi, S; Di Maggio, L; Saeed, N; Evans, B; Solomons, J; Wand, ME; Sutton, JM; Rahman, KM J Med Chem 63: 6941-6958 (2020)
- Burkholder, TP; Kudlacz, EM; Le, TB; Knippenberg, RW; Shatzer, SA; Maynard, GD; Webster, ME; Horgan, SW Bioorg Med Chem Lett 6: 951-956 (1996)
- Welsch, ME; Zhou, J; Gao, Y; Yan, Y; Porter, G; Agnihotri, G; Li, Y; Lu, H; Chen, Z; Thomas, SB ACS Med Chem Lett 7: 1124-1129 (2016)
- Stebbins, JL; Zhang, Z; Chen, J; Wu, B; Emdadi, A; Williams, ME; Cashman, J; Pellecchia, M J Med Chem 50: 6607-17 (2007)
- Namanja-Magliano, HA; Bohn, K; Agrawal, N; Willoughby, ME; Hrycyna, CA; Chmielewski, J Bioorg Med Chem 25: 5128-5132 (2017)
- Grunewald, GL; Seim, MR; Bhat, SR; Wilson, ME; Criscione, KR Bioorg Med Chem 16: 542-59 (2008)
- Cipollina, JA; Ruediger, EH; New, JS; Wire, ME; Shepherd, TA; Smith, DW; Yevich, JP J Med Chem 34: 3316-28 (1991)
- Coates, DA; Frimpong, K; Holloway, WG; Jones, BS; Levinson, AM; Lugar, III, CW; Richett, ME; Watson, BM; Woodman, ME US Patent US12252491 (2025)
- Ma, Y; Zhao, S; Ren, Y; Cherukupalli, S; Li, Q; Woodson, ME; Bradley, DP; Tavis, JE; Liu, X; Zhan, P Eur J Med Chem 225: (2021)
- Cao, Y; Zhang, M; Wu, C; Lee, S; Wroblewski, ME; Whipple, T; Nagy, PI; Takács-Novák, K; Balázs, A; Torös, S; Messer, WS J Med Chem 46: 4273-86 (2003)
- Cheng, Y; Hua, R; Kellar, T; Li, W; Gibbons, P; Zak, ME US Patent US10189836 (2019)
- Areias, FM; Brea, J; Gregori-Puigjané, E; Zaki, ME; Carvalho, MA; Domínguez, E; Gutiérrez-de-Terán, H; Proença, MF; Loza, MI; Mestres, J Bioorg Med Chem 18: 3043-52 (2010)
- Chiaradia, LD; Mascarello, A; Purificação, M; Vernal, J; Cordeiro, MN; Zenteno, ME; Villarino, A; Nunes, RJ; Yunes, RA; Terenzi, H Bioorg Med Chem Lett 18: 6227-30 (2008)
- Nagarajan, SR; Devadas, B; Zupec, ME; Freeman, SK; Brown, DL; Lu, HF; Mehta, PP; Kishore, NS; McWherter, CA; Getman, DP; Gordon, JI; Sikorski, JA J Med Chem 40: 1422-38 (1997)
- Zhang, MQ; Zwaagstra, ME; Nederkoorn, PH; Timmerman, H Bioorg Med Chem Lett 7: 1331-1336 (1997)