Report error Found 123 Enz. Inhib. hit(s) with all data for entry = 50045069
Affinity DataKi: 51nMAssay Description:Binding affinity to RORc (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Binding affinity to RORc (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 111nMAssay Description:Binding affinity to RORc-LBD (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Binding affinity to RORa (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 172nMAssay Description:Binding affinity to RORa-LBD (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Displacement of [3H2]25-hydroxycholesterol from RoRc-LBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [3H2]25-hydroxycholesterol from RoRc-LBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <16nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Displacement of [3H2]25-hydroxycholesterol from RoRc-LBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Displacement of [3H2]25-hydroxycholesterol from RoRc-LBD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Binding affinity to RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Binding affinity to RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]T0901317 from human RoRc expressed in HepG2 cells by scintillation proximity binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Displacement of [3H]T0901317 from human RoRc expressed in HepG2 cells by scintillation proximity binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]T0901317 from human RoRc expressed in HepG2 cells by scintillation proximity binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Displacement of [3H]T0901317 from human RoRc expressed in HepG2 cells by scintillation proximity binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to RORc-LBD (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of RORc (unknown origin) assessed as inhibition of coactivator recruitment by GAL4-nuclear receptor LBD assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of thymus-specific isoform RORgamma (unknown origin) transcriptional activity by luciferase-based cotransfection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of RORa (unknown origin) assessed as inhibition of coactivator recruitment by GAL4-nuclear receptor LBD assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Displacement of fluorescein-labelled 25-HC from human RoRgamma-LBD by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Binding affinity to RORgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Agonist activity at RoRc-LBD (unknown origin) expressed in HEK293 cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: <1.50E+4nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: <1.50E+4nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Agonist activity at RoRc-LBD (unknown origin) expressed in HEK293 cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Agonist activity at RoRc-LBD (unknown origin) expressed in HEK293 cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: <1.50E+4nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as SRC1 to 2 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Activity at human RoRc in human Jurkat cells assessed as inhibition of IL-17 promoterMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Activity at human RoRc in human Jurkat cells assessed as inhibition of IL-17 promoterMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Activity at human RoRc in human Jurkat cells assessed as inhibition of IL-17 promoterMore data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Activity at human RoRc in human Jurkat cells assessed as inhibition of IL-17 promoterMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Activity at human RoRc in human Jurkat cells assessed as inhibition of IL-17 promoterMore data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:Agonist activity at human RoRc-LBD expressed in CHO cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at human RoRc-LBD expressed in CHO cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Agonist activity at human RoRc-LBD expressed in CHO cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Agonist activity at human RoRc-LBD expressed in CHO cells assessed as transcriptional activity by GAL4 reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at human RoRc-LBD in human PBMC cells assessed as inhibition of IL-17A production by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at human RoRc-LBD in human PBMC cells assessed as inhibition of IL-17A production by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at human RoRc-LBD in human PBMC cells assessed as inhibition of IL-17A production by luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Inverse agonist activity at human RoRc-LBD fusion protein with GST expressed in BL-21 (BL3) cells assessed as SRC1 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: <32nMAssay Description:Inverse agonist activity at human RoRc-LBD fusion protein with GST expressed in BL-21 (BL3) cells assessed as SRC1 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Inverse agonist activity at human RoRc-LBD fusion protein with GST expressed in BL-21 (BL3) cells assessed as SRC1 coactivator peptide recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Inverse agonist activity at human RoRc-LBD fusion protein with GST expressed in BL-21 (BL3) cells assessed as SRC1 coactivator peptide recruitmentMore data for this Ligand-Target Pair