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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-adrenergic receptor kinase 1' and Ligand = 'BDBM50554259'
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554259(CHEMBL4788026)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554259(CHEMBL4788026)
Affinity DataKd:  3.33E+3nMAssay Description:Binding affinity to full length human GRK2 by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB