Found 4 Enz. Inhib. hit(s) with Target = 'G-protein coupled receptor homolog US28' and Ligand = 'BDBM50027216'
TargetG-protein coupled receptor homolog US28(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Vrije Universiteit
Curated by PDSP Ki Database
Vrije Universiteit
Curated by PDSP Ki Database
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibitory concentration against chemokine receptor US28 expressed in COS-7 cells using [125I]-CCL5More data for this Ligand-Target Pair
TargetG-protein coupled receptor homolog US28(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Vrije Universiteit
Curated by PDSP Ki Database
Vrije Universiteit
Curated by PDSP Ki Database
Affinity DataEC50: 4.57E+3nMAssay Description:Allosteric modulatory activity at FLAG-tagged wild type human cytomegalovirus US28 receptor expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
TargetG-protein coupled receptor homolog US28(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Vrije Universiteit
Curated by PDSP Ki Database
Vrije Universiteit
Curated by PDSP Ki Database
Affinity DataEC50: 4.50E+3nMAssay Description:Allosteric modulatory activity at FLAG-tagged wild type human cytomegalovirus US28 receptor expressed in HEK293T cells by PathDetectElk1 assayMore data for this Ligand-Target Pair
TargetG-protein coupled receptor homolog US28(Human cytomegalovirus (strain AD169) (HHV-5) (Huma...)
Vrije Universiteit
Curated by PDSP Ki Database
Vrije Universiteit
Curated by PDSP Ki Database
Affinity DataEC50: 3.20E+3nMAssay Description:Effective concentration against US28-mediated inositol phosphate production in COS-7 cellsMore data for this Ligand-Target Pair