Found 4 Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Ligand = 'BDBM50261184'
TargetGonadotropin-releasing hormone receptor(Mus musculus)
Norwegian Medical Cyclotron Centre
Curated by ChEMBL
Norwegian Medical Cyclotron Centre
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Binding affinity to mouse gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity at rat GnRH receptor by competition binding assayMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity to rat gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Norwegian Medical Cyclotron Centre
Curated by ChEMBL
Norwegian Medical Cyclotron Centre
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity to human gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair