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Found 4 Enz. Inhib. hit(s) with Target = 'Heparanase' and Ligand = 'BDBM50165636'
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165636(2-(4-(5-(4-(3-(4-bromophenyl)acrylamido)-2-chlorop...)
Affinity DataIC50:  398nMAssay Description:Inhibition of heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165636(2-(4-(5-(4-(3-(4-bromophenyl)acrylamido)-2-chlorop...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human heparanase assessed as reduction in basic fibroblast growth factor binding incubated for 2 hrs by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165636(2-(4-(5-(4-(3-(4-bromophenyl)acrylamido)-2-chlorop...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165636(2-(4-(5-(4-(3-(4-bromophenyl)acrylamido)-2-chlorop...)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant heparanase catalytic stie (unknown origin) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed