Found 3 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50145022'
Affinity DataKi: 1.57nMAssay Description:In vitro binding afinity at opioid sigma-1 receptorin guinea pig brain membranes by (+)-[3H]-pentazocine displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.57nMAssay Description:Displacement of [3H]pentazocine from Sigma1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Displacement of (+)-[3H]pentazocine from mouse sigma 1 receptor in TRAMP cell membraneMore data for this Ligand-Target Pair