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Found 4 Enz. Inhib. hit(s) with Target = 'Sterol O-acyltransferase 1' and Ligand = 'BDBM50028867'
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50028867((3R,4S)-1,4-Bis-(4-methoxy-phenyl)-3-(3-phenyl-pro...)
Affinity DataIC50:  1.10E+4nMAssay Description:The concentration required for 50% inhibition of Acyl coenzyme A:cholesterol acyltransferase activity was measured at the dosage by using microsomal ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50028867((3R,4S)-1,4-Bis-(4-methoxy-phenyl)-3-(3-phenyl-pro...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase (ACAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50028867((3R,4S)-1,4-Bis-(4-methoxy-phenyl)-3-(3-phenyl-pro...)
Affinity DataIC50:  1.80E+4nMAssay Description:Concentration required for 50% inhibition of Acyl coenzyme A:cholesterol acyltransferase activity using microsomal ACAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50028867((3R,4S)-1,4-Bis-(4-methoxy-phenyl)-3-(3-phenyl-pro...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase (ACAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed