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Found 12 with Last Name = 'kauschke' and Initial = 'sg'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228359(CHEMBL254815 | methyl 2-chloro-6,8-dihydroxy-9-{1-...)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228360(CHEMBL254814 | methyl 9-[1-(acetyloxyethyl)]-2-chl...)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228358(CHEMBL253120 | methyl 2-chloro-9-ethyl-6,8-dihydro...)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228361(2-chloro-6,8-dihydroxy-1-methoxy-3,9-dimethyltetra...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228359(CHEMBL254815 | methyl 2-chloro-6,8-dihydroxy-9-{1-...)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228360(CHEMBL254814 | methyl 9-[1-(acetyloxyethyl)]-2-chl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228361(2-chloro-6,8-dihydroxy-1-methoxy-3,9-dimethyltetra...)
Affinity DataIC50:  4.40E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228358(CHEMBL253120 | methyl 2-chloro-9-ethyl-6,8-dihydro...)
Affinity DataIC50:  7.00E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228359(CHEMBL254815 | methyl 2-chloro-6,8-dihydroxy-9-{1-...)
Affinity DataEC50:  130nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228361(2-chloro-6,8-dihydroxy-1-methoxy-3,9-dimethyltetra...)
Affinity DataEC50:  260nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228358(CHEMBL253120 | methyl 2-chloro-9-ethyl-6,8-dihydro...)
Affinity DataEC50:  180nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228360(CHEMBL254814 | methyl 9-[1-(acetyloxyethyl)]-2-chl...)
Affinity DataEC50:  160nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed