TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 0.340nMAssay Description:Binding affinity to rat brain histamine H3 receptor after 1 hr by gamma countingMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 1.82nMAssay Description:Antagonist activity at histamine H3 receptor in rat cortical hemispheres assessed as inhibition of forskolin stimulated cAMP accumulation after 6 hrsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 3.55nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 3.72nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 3.98nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 4.17nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 5.01nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 6.31nMAssay Description:Antagonist activity at histamine H3 receptor in rat cortical hemispheres assessed as inhibition of forskolin stimulated cAMP accumulation after 6 hrsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 6.92nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 9.55nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 11.5nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: 26.3nMAssay Description:Antagonist activity at rat histamine H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Eth Zurich (Swiss Federal Institute Of Technology)
Curated by ChEMBL
Affinity DataKd: >3.00E+3nMAssay Description:Binding affinity to rat histamine H3 receptor low affinity site after 1 hr by Schard plot analysisMore data for this Ligand-Target Pair