Compile Data Set for Download or QSAR
maximum 50k data
Found 25 of ki for UniProtKB: Q16512
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596594(CHEMBL5182936)
Affinity DataKi:  60nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM27400(1-ethyl-2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,...)
Affinity DataKi:  108nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM27344(2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyri...)
Affinity DataKi:  150nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM27401(1-(2-hydroxyethyl)-2-(pyridin-4-yl)-1H,4H,5H,6H,7H...)
Affinity DataKi:  220nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596601(CHEMBL5175087)
Affinity DataKi:  260nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi:  540nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596600(CHEMBL5202568)
Affinity DataKi:  650nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596595(CHEMBL5187643)
Affinity DataKi:  920nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596596(CHEMBL5170263)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545113(CHEMBL4647033)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM27394(1-methyl-2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545105(CHEMBL4635777)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545111(CHEMBL4634210)
Affinity DataKi:  1.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545109(CHEMBL4632420)
Affinity DataKi:  1.91E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM55759(2-(4-pyridyl)-1H-benzimidazole | 2-pyridin-4-yl-1H...)
Affinity DataKi:  2.24E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545101(CHEMBL4636367)
Affinity DataKi:  2.59E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545106(CHEMBL4649365)
Affinity DataKi:  2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545110(CHEMBL4638916)
Affinity DataKi:  2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545108(CHEMBL4646744)
Affinity DataKi:  2.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545104(CHEMBL4645636)
Affinity DataKi:  3.02E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545102(CHEMBL185288)
Affinity DataKi:  3.25E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545107(CHEMBL4637286)
Affinity DataKi:  4.88E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545112(CHEMBL160012)
Affinity DataKi:  5.37E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545103(CHEMBL4640475)
Affinity DataKi:  6.77E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged PKN1 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed