Affinity DataIC50: <1nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of D5D in rat RLN10 cells using [14C]DGLA as substrate preincubated for 30 mins followed by substrate addition measured after 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of D5D in Sprague-Dawley rat liver microsomes using [14C]DGLA as substrate preincubated for 5 mins measured after 120 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of D5D in rat RLN10 cells using [14C]DGLA as substrate preincubated for 30 mins followed by substrate addition measured after 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: >30nMAssay Description:Inhibition of rat microsomal Delta5-desaturaseMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of D5D in Sprague-Dawley rat liver microsomes using [14C]DGLA as substrate preincubated for 5 mins measured after 120 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.17E+3nMAssay Description:Inhibition of Delta(5) fatty acid desaturase in freshly isolated rat hepatocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]T-3364366 from D5D in rat liver microsomal membrane preincubated for 15 mins followed by radioligand addition measured after 150 ...More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of stearoyl-CoA delta5 desaturase in rat microsomeMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rat Delta(5) fatty acid desaturase by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of rat delta-5 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of rat delta-5 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of rat delta-5 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of rat delta-5 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of rat delta-5 desaturase activity expressed in human HEpG2 cellsMore data for this Ligand-Target Pair