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Report error Found 96 of ec50 for UniProtKB: P18089
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50090256(ascorbic acid | (R)-5-((S)-1,2-dihydroxyethyl)-3,4...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human adrenergic alpha2B receptor expressed in HEK293 cells coexpressing Gqi5 protein by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50212995(CHEMBL75030)
Affinity DataEC50:  3.5nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50473228(AGN-190837 | CHEMBL297752)
Affinity DataEC50:  9.30nMAssay Description:Alpha-2B adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataEC50:  9.30nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50212996(CHEMBL306377)
Affinity DataEC50:  35nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50415140(CHEMBL569933)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  62nMAssay Description:Agonistic potency at human adrenergic alpha-2B receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50052880(Imidazolidin-2-ylidene-(5-methyl-quinoxalin-6-yl)-...)
Affinity DataEC50:  78nMAssay Description:Alpha-2B adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50019646(CHEMBL17860 | lofexidine | 2-(alpha-(2,6-Dichlorop...)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419890(CHEMBL1956191)
Affinity DataEC50:  162nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-2-imidazoline | 2-(2,6-dic...)
Affinity DataEC50:  166nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50412258(CHEMBL451229)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419873(CHEMBL1956203)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50212993(CHEMBL305928)
Affinity DataEC50:  214nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419875(CHEMBL1956193)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419876(CHEMBL266613)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419888(CHEMBL1956202)
Affinity DataEC50:  295nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419883(CHEMBL1956201)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human alpha2B ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419885(CHEMBL157206)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50412244(CHEMBL495096)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50473224(CHEMBL296660)
Affinity DataEC50:  562nMAssay Description:Alpha-2B adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  646nMAssay Description:Agonistic potency at human adrenergic alpha-2B receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  646nMAssay Description:Agonist activity at human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  646nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  646nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataEC50:  692nMAssay Description:Agonistic potency at human adrenergic alpha-2B receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataEC50:  692nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataEC50:  724nMAssay Description:Agonistic activity towards human Alpha-2B adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50027031((2-Chloro-phenyl)-(4,5-dihydro-1H-imidazol-2-ylmet...)
Affinity DataEC50:  776nMAssay Description:Agonist activity at human alpha2b-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50213028(CHEMBL74283)
Affinity DataEC50:  891nMAssay Description:Alpha-2B adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50000214(CHEMBL337862)
Affinity DataEC50:  955nMAssay Description:Agonist activity at human alpha2b-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2018
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50473154(CHEMBL14107)
Affinity DataEC50:  977nMAssay Description:Agonist activity at human alpha2B ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50415139(CHEMBL576623)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50002905(CHEMBL373535)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic potency at human adrenergic alpha-2B receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50417349(CHEMBL1276248)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor mic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50027060(2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imi...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50476178(CHEMBL223829)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50002905(CHEMBL373535)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50419884(CHEMBL157955)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50415136(CHEMBL570973)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-2-imidazoline | 2-(2,6-dic...)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at human alpha2B adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50493432(CHEMBL2431279)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human alpha2B ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
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