TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: >0.000100nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.0210nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.0407nMAssay Description:Displacement of [3H]DAMGO from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.0480nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Fujisawa Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]pCCK-8 from cholecystokinin type B receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 0.148nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.178nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Parke-Davis Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:The compound was evaluated for the inhibition of binding of [3H]-PD 140376 to Cholecystokinin type B receptor in mouse cortex.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.209nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.224nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Fujisawa Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Displacement of 0.2 nM [3H]-pCCK-8 from guinea pig brain membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.251nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of 0.2 nM [3H]-pCCK-8 from guinea pig brain membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.288nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.295nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity of the compound against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]pCCK-8 from cholecystokinin type B receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.302nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Affinity DataKi: 0.310nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.331nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.355nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.372nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.398nMAssay Description:Inhibition of specific binding of [125I]-ET-1 (endothelin 1) to the endothelin A receptor of rat aorta membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Compound was tested for the affinity against Cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of binding of [125I]-PD 142308 to CCK-B receptor was determinedMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
Fujisawa Pharmaceutical Co., Ltd
Curated by PDSP Ki Database
