Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50014339
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31373(CHEMBL28137 | terephthalamide scaffold, 9)
Affinity DataKi:  781nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31374(CHEMBL286715 | terephthalamide scaffold, 10)
Affinity DataKi:  839nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31381(CHEMBL282624 | terephthalamide scaffold, 29)
Affinity DataKi:  1.01E+3nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31379(CHEMBL28872 | terephthalamide scaffold, 27)
Affinity DataKi:  1.79E+3nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31378(CHEMBL284686 | terephthalamide scaffold, 26)
Affinity DataKi:  1.85E+3nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31385(CHEMBL281240 | terephthalamide scaffold, 17)
Affinity DataKi:  3.31E+3nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31376(CHEMBL433422 | terephthalamide scaffold, 24)
Affinity DataKi:  5.85E+3nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50141117((S)-2-[4-Diisopropylcarbamoyl-2-(naphthalen-1-ylox...)
Affinity DataKi:  7.63E+3nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50141118((S)-(4-Diisopropylcarbamoyl-2-isopropoxy-benzoylam...)
Affinity DataKi:  1.09E+4nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31375(CHEMBL28504 | terephthalamide scaffold, 23)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50141122((S)-2-[4-(1-Carboxy-3-methyl-butylcarbamoyl)-2-phe...)
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50141121((S)-2-{4-[(1-Carboxy-ethyl)-isobutyl-carbamoyl]-2-...)
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50141120((S)-2-{4-[(1-Carboxy-2-methyl-propyl)-isobutyl-car...)
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50141119((S)-2-[4-(1-Carboxy-3-methyl-butylcarbamoyl)-2-(na...)
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM31389(CHEMBL29180 | terephthalamide scaffold, 36)
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity for Bcl-xL was assessed by a fluorescence polarizationassay using a fluorescently labeled 16-mer Bak-peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed