Compile Data Set for Download or QSAR
Report error Found 165 Enz. Inhib. hit(s) with all data for entry = 50017800
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410903(CHEMBL207598)
Affinity DataKi:  0.5nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410898(CHEMBL205757)
Affinity DataKi:  0.510nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410901(CHEMBL206413)
Affinity DataKi:  0.650nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410904(CHEMBL377532)
Affinity DataKi:  0.720nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410899(CHEMBL383674)
Affinity DataKi:  0.720nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186686(benzenesulfonyl-Glu(OtBu)-Ser-LeuVSMe | CHEMBL2049...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186721(Cbz-Ile-NeopentylAsn-Ala-LeuVSMe | CHEMBL382203)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186710(pTosyl-Glu(OtBu)-Ala-LeuVSMe | CHEMBL207016)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50069984((R)-1-((S)-2-((S)-2-(benzyloxycarbonyl)-4-methylpe...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186697(benzyl (2S,3S)-3-methyl-1-((S)-1-((S)-1-((S,E)-5-m...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186709(Cbz-Ile-Glu(OtBu)-Ala-LeuVSMe | CHEMBL207162)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186712(Cbz-Glu(OtBu)-Ser-LeuVSMe | CHEMBL206206)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186706(Cbz-Ile-t-ButylGln-Ala-LeuVSMe | CHEMBL438612)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50069985({1-[(S)-(S)-1-((S)-1-Formyl-3-methyl-butylcarbamoy...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50185154((2S,3S)-2-(Acetyl-methyl-amino)-3-methyl-pentanoic...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186696(pTosyl-NeopentylAsn-Ala-LeuVSMe | CHEMBL206001)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410906(CHEMBL207160)
Affinity DataKi:  5.70nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186707(pTosyl-NeopentylAsn-Ser-LeuVSMe | CHEMBL204946)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186685(Cbz-Glu(OtBu)-Ala-LeuVSMe | CHEMBL208015)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186691((S)-tert-butyl 4-(2,2-diphenylacetamido)-5-((S)-1-...)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186724(Cbz-Ile-CyclohexylGlu-Ala-LeuVSMe | CHEMBL207669)
Affinity DataIC50: 10nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186694(benzoyl-Glu(OtBu)-Ala-LeuVSMe | CHEMBL207336)
Affinity DataIC50: 17nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186698(Cbz-Ile-t-ButylhomoGlu-Ala-LeuVSMe | CHEMBL207196)
Affinity DataIC50: 24nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186717(Cbz-Ile-hPhe-Ala-LeuVSMe | CHEMBL446443)
Affinity DataIC50: 27nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410900(CHEMBL207425)
Affinity DataKi:  32nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186702(Ac-hPhe-Leu-Phe-LeuVSMe | CHEMBL379669)
Affinity DataIC50: 35nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410896(CHEMBL383122)
Affinity DataKi:  38nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186690(Cbz-Ile-trans-StyrylAla-Ala-LeuVSMe | CHEMBL208159)
Affinity DataIC50: 44nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410907(CHEMBL437311)
Affinity DataKi:  45nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186708(Cbz-Ile-NeopentylGln-Ala-LeuVSMe | CHEMBL378901)
Affinity DataIC50: 49nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186693(Cbz-Ile-Ser(OBn)-Ala-LeuVSMe | CHEMBL379772)
Affinity DataIC50: 49nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186711(Cbz-Ile-iPrGln-Ala-LeuVSMe | CHEMBL437115)
Affinity DataIC50: 52nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186687(Cbz-Ile-Leu-Ala-LeuVSMe | CHEMBL207403)
Affinity DataIC50: 69nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186705(Cbz-Ile-Asp-(OtBu)-Ala-LeuVSMe | CHEMBL379771)
Affinity DataIC50: 78nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186692(Cbz-Ile-hGln-Ala-LeuVSMe | CHEMBL437882)
Affinity DataIC50: 120nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186716(Ac-hPhe-Leu-Ala-LeuVSMe | CHEMBL207579)
Affinity DataIC50: 120nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410902(CHEMBL205687)
Affinity DataKi:  130nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410908(CHEMBL381931)
Affinity DataKi:  140nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186702(Ac-hPhe-Leu-Phe-LeuVSMe | CHEMBL379669)
Affinity DataIC50: 150nMAssay Description:Inhibition of cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50185154((2S,3S)-2-(Acetyl-methyl-amino)-3-methyl-pentanoic...)
Affinity DataIC50: 160nMAssay Description:Inhibition of trypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186695(Cbz-Glu(OtBu)-Gly-LeuVSMe | CHEMBL208019)
Affinity DataIC50: 170nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186689(Ac-Glu(OtBu)-Ala-LeuVSMe | CHEMBL383529)
Affinity DataIC50: 260nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50069985({1-[(S)-(S)-1-((S)-1-Formyl-3-methyl-butylcarbamoy...)
Affinity DataKi:  330nMAssay Description:Inhibition of trypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186720(Cbz-BocDab-Ser-LeuVSMe | CHEMBL381884)
Affinity DataIC50: 430nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186688(Cbz-Ile-Phe-Ala-LeuVSMe | CHEMBL207284)
Affinity DataIC50: 460nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50069985({1-[(S)-(S)-1-((S)-1-Formyl-3-methyl-butylcarbamoy...)
Affinity DataKi:  470nMAssay Description:Inhibition of post glutamyl peptide hydrolase-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50410905(CHEMBL379476)
Affinity DataKi:  500nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186713((S)-tert-butyl 2-((S)-3-(benzyloxycarbonyl)-4-((S)...)
Affinity DataIC50: 540nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186700(Cbz-Ile-Gln-Ala-LeuVSMe | CHEMBL382180)
Affinity DataIC50: 570nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50186687(Cbz-Ile-Leu-Ala-LeuVSMe | CHEMBL207403)
Affinity DataIC50: 700nMAssay Description:Inhibition of cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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