Compile Data Set for Download or QSAR
Report error Found 701 Enz. Inhib. hit(s) with all data for entry = 50042279
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50097256((R)-N1-((S)-3,3-dimethyl-1-oxo-1-(pyridin-4-ylamin...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50106022((7S,8R,11S)-8-[3-(4-chloro-phenyl)-propyl]-9-oxo-2...)
Affinity DataIC50: 0.257nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50160843(1-[4-(4-Phenoxy-phenoxy)-phenyl]-1,7,9-triaza-spir...)
Affinity DataKi:  0.331nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50063910((R)-N*1*-((S)-2,2-Dimethyl-1-methylcarbamoyl-propy...)
Affinity DataIC50: 0.339nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50097252((R)-N'-((S)-3,3-dimethyl-1-oxo-1-((R)-1-phenylethy...)
Affinity DataIC50: 0.380nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM30359(BOC-piperidinyl glycine derivative, 34)
Affinity DataIC50: 0.398nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50097273((R)-N*1*-((S)-2,2-dimethyl-1-methylcarbamoyl-propy...)
Affinity DataIC50: 0.501nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50088118(N-Hydroxy-2-[(4-nitro-benzyl)-pentafluorobenzenesu...)
Affinity DataKi:  0.603nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50290442((R)-N4-hydroxy-N1-((S)-1-(methylamino)-1-oxo-3-phe...)
Affinity DataIC50: 0.603nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50086781(N-Hydroxy-2-[(4-nitro-benzyl)-pentafluorobenzenesu...)
Affinity DataKi:  0.603nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50088118(N-Hydroxy-2-[(4-nitro-benzyl)-pentafluorobenzenesu...)
Affinity DataKi:  0.692nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50086781(N-Hydroxy-2-[(4-nitro-benzyl)-pentafluorobenzenesu...)
Affinity DataKi:  0.692nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50102468(4-[Carboxy-(4'-methoxy-biphenyl-4-sulfonylamino)-m...)
Affinity DataIC50: 0.708nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50082545((S)-N-hydroxy-4-(4-methoxyphenylsulfonyl)-2,2-dime...)
Affinity DataIC50: 0.708nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50098924((R)-1-Cyclohexyl-3-(4-methoxy-benzenesulfonyl)-6-o...)
Affinity DataIC50: 0.708nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50160855(1-[4-(4-chloro-phenoxy)-phenyl]-1,7,9-triaza-spiro...)
Affinity DataKi:  0.724nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50160851(4-[4-(2,6,8,10-Tetraoxo-1,7,9-triaza-spiro[4.5]dec...)
Affinity DataKi:  0.724nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11341(2-[benzyl(2,3,4,5,6-pentafluorobenzene)sulfonamido...)
Affinity DataKi:  0.794nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11348(2-[benzyl(2,3,4,5,6-pentafluorobenzene)sulfonamido...)
Affinity DataKi:  0.794nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50100812(2-(N-(2-nitrobenzyl)-2,3,4,5,6-pentafluorophenylsu...)
Affinity DataKi:  0.794nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50106016((7S,8R,11S)-8-[3-(4-ethoxy-phenyl)-propyl]-9-oxo-2...)
Affinity DataIC50: 0.794nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50084726(4-(Biphenyl-4-carbonyl)-1-(4-methoxy-benzenesulfon...)
Affinity DataIC50: 0.891nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11336(2-[benzyl(2,3,4,5,6-pentafluorobenzene)sulfonamido...)
Affinity DataKi:  0.891nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50160855(1-[4-(4-chloro-phenoxy)-phenyl]-1,7,9-triaza-spiro...)
Affinity DataKi:  0.955nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50102479(4-[Carboxy-(4'-methylsulfanyl-biphenyl-4-sulfonyla...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50084759(4-(2-Hydroxy-3-methyl-butyryl)-1-(4-methoxy-benzen...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50097245((R)-N*1*-((S)-2,2-Dimethyl-1-phenylcarbamoyl-propy...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50096472(2-(N-benzyl-4-methoxyphenylsulfonamido)-N-hydroxy-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50102478(4-{Carboxy-[(4'-methoxy-biphenyl-4-sulfonyl)-(2-me...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50098915((R)-1-tert-Butyl-3-(4-methoxy-benzenesulfonyl)-6-o...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50084729(4-Acetyl-1-(4-methoxy-benzenesulfonyl)-piperazine-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50098918(1-BENZYL-3-(4-METHOXY-BENZENESULFONYL)-6-OXO-HEXAH...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50100812(2-(N-(2-nitrobenzyl)-2,3,4,5,6-pentafluorophenylsu...)
Affinity DataKi:  1nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50102476(4-[Carboxy-(4'-methoxy-biphenyl-4-sulfonylamino)-m...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50290456((R)-2-Heptyl-N*4*-hydroxy-N*1*-((S)-1-methylcarbam...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50290433((R)-N4-hydroxy-N1-((S)-1-(methylamino)-1-oxo-3-phe...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50290450((R)-2-Dodecyl-N*4*-hydroxy-N*1*-((S)-1-methylcarba...)
Affinity DataIC50: 1nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11348(2-[benzyl(2,3,4,5,6-pentafluorobenzene)sulfonamido...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11330(2-[benzyl(2,3,4,5,6-pentafluorobenzene)sulfonamido...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50160849(4-[4-(2,6,8,10-Tetraoxo-1,7,9-triaza-spiro[4.5]dec...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50102468(4-[Carboxy-(4'-methoxy-biphenyl-4-sulfonylamino)-m...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11341(2-[benzyl(2,3,4,5,6-pentafluorobenzene)sulfonamido...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50071839(4-benzoyl-N-hydroxy-1-(4-phenoxyphenylsulfonyl)-1,...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50097240((R)-N1-((S)-1-(cyclohexylamino)-3,3-dimethyl-1-oxo...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50423402(CHEMBL122711)
Affinity DataKi:  1.30nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11349(2-[benzyl(4-methoxybenzene)sulfonamido]-N-hydroxy-...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50086801(2-(N-(4-nitrobenzyl)-2,2,12,12,15,15,18,18,18-nona...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM11336(2-[benzyl(2,3,4,5,6-pentafluorobenzene)sulfonamido...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50423402(CHEMBL122711)
Affinity DataKi:  1.40nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50088128(N-Hydroxy-2-[(4-nitro-benzyl)-(nonafluorobutane-1-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
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