Compile Data Set for Download or QSAR
Report error Found 160 Enz. Inhib. hit(s) with all data for entry = 50041839
TargetAngiopoietin-1 receptor(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5815BDBM5815(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 2nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5815BDBM5815(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 3.02nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8826BDBM8826(CHEMBL196363 | 3-(4-{4-aminothieno[2,3-d]pyrimidin...)
Affinity DataIC50: 3.02nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8870BDBM8870(KDR Kinase Inhibitor, 9 | N-[4-(4-Aminothieno[2,3-...)
Affinity DataIC50: 3.02nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8826BDBM8826(CHEMBL196363 | 3-(4-{4-aminothieno[2,3-d]pyrimidin...)
Affinity DataIC50: 6.03nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8813BDBM8813(CHEMBL537435 | KDR Kinase Inhibitor, 7 | CHEMBL371...)
Affinity DataIC50: 6.03nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8813BDBM8813(CHEMBL537435 | KDR Kinase Inhibitor, 7 | CHEMBL371...)
Affinity DataIC50: 8.91nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8862BDBM8862(CHEMBL425749 | 3-(4-{4-aminothieno[2,3-d]pyrimidin...)
Affinity DataIC50: 11.0nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8844BDBM8844(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 12.0nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8867BDBM8867(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-2-methox...)
Affinity DataIC50: 12.9nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8860BDBM8860(CHEMBL198297 | N-{4-[4-Amino-6-(3-hydroxypropyl)th...)
Affinity DataIC50: 15.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8833BDBM8833(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 15.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8847BDBM8847(3-[4-amino-5-(4-{[(3-methylphenyl)carbamoyl]amino}...)
Affinity DataIC50: 17.0nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8846BDBM8846(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 17.0nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8832BDBM8832(N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)...)
Affinity DataIC50: 19.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8858BDBM8858(CHEMBL197353 | 3-{4-[4-amino-6-(2-hydroxyethyl)thi...)
Affinity DataIC50: 19.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8865BDBM8865(CHEMBL371510 | N-[4-(4-Aminothieno[2,3-d]pyrimidin...)
Affinity DataIC50: 19.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8844BDBM8844(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 19.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5816BDBM5816(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 21.9nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8838BDBM8838(CHEMBL382517 | 3-(4-{4-amino-6-methylthieno[2,3-d]...)
Affinity DataIC50: 21.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8860BDBM8860(CHEMBL198297 | N-{4-[4-Amino-6-(3-hydroxypropyl)th...)
Affinity DataIC50: 25.7nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8853BDBM8853(N-[4-(4-Amino-6-propylthieno[2,3-d]pyrimidin-5-yl)...)
Affinity DataIC50: 26.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8824BDBM8824(N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)-...)
Affinity DataIC50: 26.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8835BDBM8835(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 26.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8862BDBM8862(CHEMBL425749 | 3-(4-{4-aminothieno[2,3-d]pyrimidin...)
Affinity DataIC50: 26.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8824BDBM8824(N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)-...)
Affinity DataIC50: 28.2nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5814BDBM5814(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 28.2nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8867BDBM8867(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-2-methox...)
Affinity DataIC50: 28.2nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8839BDBM8839(N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)...)
Affinity DataIC50: 28.8nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8812BDBM8812(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 32.4nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8836BDBM8836(N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)...)
Affinity DataIC50: 33.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8856BDBM8856(3-{4-[4-amino-6-(pyridin-3-ylmethyl)thieno[2,3-d]p...)
Affinity DataIC50: 33.9nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50416743BDBM50416743(CHEMBL372744)
Affinity DataIC50: 33.9nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8832BDBM8832(N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)...)
Affinity DataIC50: 34.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8838BDBM8838(CHEMBL382517 | 3-(4-{4-amino-6-methylthieno[2,3-d]...)
Affinity DataIC50: 34.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8812BDBM8812(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 36.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5810BDBM5810(N-{3-[4-amino-5-(4-phenylphenyl)furo[2,3-d]pyrimid...)
Affinity DataIC50: 36.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8858BDBM8858(CHEMBL197353 | 3-{4-[4-amino-6-(2-hydroxyethyl)thi...)
Affinity DataIC50: 37.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8865BDBM8865(CHEMBL371510 | N-[4-(4-Aminothieno[2,3-d]pyrimidin...)
Affinity DataIC50: 38.0nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8843BDBM8843(methyl 3-{[(4-{4-amino-6-methylthieno[2,3-d]pyrimi...)
Affinity DataIC50: 42.7nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8846BDBM8846(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 45.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8840BDBM8840(-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-...)
Affinity DataIC50: 45.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8841BDBM8841(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 47.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8831BDBM8831(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50: 50.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8869BDBM8869(3-(4-{4-amino-6-ethylthieno[2,3-d]pyrimidin-5-yl}p...)
Affinity DataIC50: 50.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8840BDBM8840(-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-...)
Affinity DataIC50: 50.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8857BDBM8857(3-{4-[4-amino-6-(pyridin-4-ylmethyl)thieno[2,3-d]p...)
Affinity DataIC50: 52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8842BDBM8842(N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)...)
Affinity DataIC50: 52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8830BDBM8830(CHEMBL198267 | 3-(4-{4-amino-6-methylthieno[2,3-d]...)
Affinity DataIC50: 52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Dalian University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8836BDBM8836(N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)...)
Affinity DataIC50: 52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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