Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50027013
TargetB1 bradykinin receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50202412(methyl 3-chloro-3'-fluoro-4'-{(1R)-1-[({1-[(triflu...)
Affinity DataKi:  0.440nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50127438(1-(2-Oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-benzo...)
Affinity DataKi:  0.590nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264141(1-Benzyl-1H-benzoimidazole-2-carboxylic acid {2-[6...)
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50127438(1-(2-Oxo-5-phenethyl-1-propyl-2,3-dihydro-1H-benzo...)
Affinity DataKi:  0.920nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264189(5-(2-chlorobenzamido)-4-methyl-N-(2-(1-(1-methylpi...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264141(1-Benzyl-1H-benzoimidazole-2-carboxylic acid {2-[6...)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264298(N-(2-((4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)(met...)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264140(N-(2-((4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)(met...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264589(N-(2-((4-(1-methyl-4,5-dihydro-1H-imidazol-2-yl)be...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264368(1-benzyl-N-ethyl-N-(2-(4-(1-methylpiperidin-4-yl)p...)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264368(1-benzyl-N-ethyl-N-(2-(4-(1-methylpiperidin-4-yl)p...)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264370(1-benzyl-N-(2-(4-(1-methylpiperidin-4-yl)piperazin...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264370(1-benzyl-N-(2-(4-(1-methylpiperidin-4-yl)piperazin...)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264446(N-(3-((4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)(met...)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264298(N-(2-((4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)(met...)
Affinity DataIC50: 155nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264497(1-(1-Benzyl-1H-benzoimidazole-2-carbonyl)-piperidi...)
Affinity DataIC50: 188nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264632(N-(2-((4-(piperidin-1-ylmethyl)benzyl)(methyl)amin...)
Affinity DataIC50: 196nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264331(1-benzyl-N-methyl-N-(2-(4-(1-methylpiperidin-4-yl)...)
Affinity DataIC50: 268nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264332(1-benzyl-N-ethyl-N-(2-oxo-2-(4-(pyridin-4-yl)piper...)
Affinity DataIC50: 278nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264296(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50: 310nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264631(N-(2-((4-(pyrimidin-2-yl)benzyl)(methyl)amino)-2-o...)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264140(N-(2-((4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)(met...)
Affinity DataIC50: 345nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264369(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50: 355nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264369(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50: 396nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264630(N-(2-((4-(pyridin-2-yl)benzyl)(methyl)amino)-2-oxo...)
Affinity DataIC50: 407nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264296(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50: 417nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264400(1-benzyl-N-isopropyl-N-(2-(4-(1-methylpiperidin-4-...)
Affinity DataIC50: 465nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264399(1-Benzyl-1H-benzoimidazole-2-carboxylic acid [2-(1...)
Affinity DataIC50: 524nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264445(1-benzyl-N-(3-(4-(1-methylpiperidin-4-yl)piperazin...)
Affinity DataIC50: 601nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264591(N-(2-((4-(1H-imidazol-1-yl)benzyl)(methyl)amino)-2...)
Affinity DataIC50: 626nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264297(1-benzyl-N-(2-(4-(1-methylpiperidin-4-yl)piperazin...)
Affinity DataIC50: 686nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264590(N-(2-((4-(5-methyl-1,2,4-oxadiazol-3-yl)benzyl)(me...)
Affinity DataIC50: 718nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264715(N-(3-(3H-benzo[d]imidazol-5-ylamino)-3-oxopropyl)-...)
Affinity DataIC50: 744nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264531((1-Benzyl-1H-benzoimidazol-2-yl)-{(S)-2-[4-(1-meth...)
Affinity DataIC50: 884nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264401(1-benzyl-N-(3-oxo-3-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50: 962nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264268(N-(4-(4,5-dihydro-1H-imidazol-2-yl)benzyl)-1-benzy...)
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264677(N-(2-((4-(thiazol-2-yl)benzyl)(methyl)amino)-2-oxo...)
Affinity DataIC50: 1.17E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264330(1-benzyl-N-methyl-N-(2-oxo-2-(4-(pyridin-4-yl)pipe...)
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264329(1-benzyl-N-(1-(4-(1-methylpiperidin-4-yl)piperazin...)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50202412(methyl 3-chloro-3'-fluoro-4'-{(1R)-1-[({1-[(triflu...)
Affinity DataKi:  1.60E+3nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264712(1-Benzyl-1H-benzoimidazole-2-carboxylic acid [3-(3...)
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264678(N-(2-((4-(1H-pyrazol-5-yl)benzyl)(methyl)amino)-2-...)
Affinity DataIC50: 2.13E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264447([1-(1-Benzyl-1H-benzoimidazole-2-carbonyl)-piperid...)
Affinity DataIC50: 2.31E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264713(1-Benzyl-1H-benzoimidazole-2-carboxylic acid [3-(2...)
Affinity DataIC50: 2.91E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264529((1-Benzyl-1H-benzoimidazol-2-yl)-{(R)-2-[4-(1-meth...)
Affinity DataIC50: 3.22E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264496([1-(1-Benzyl-1H-benzoimidazole-2-carbonyl)-piperid...)
Affinity DataIC50: 4.02E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264498((1-Benzyl-1H-benzoimidazol-2-yl)-[(R)-2-(4-pyridin...)
Affinity DataIC50: 4.07E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264680(1-Benzyl-1H-benzoimidazole-2-carboxylic acid [3-(9...)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264679(N-(2-((4-(1H-tetrazol-5-yl)benzyl)(methyl)amino)-2...)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Crab-eating macaque)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264714(1-Benzyl-1H-benzoimidazole-2-carboxylic acid [3-ox...)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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