Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 3577
TargetDual specificity protein kinase TTK(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM36486(US9266890, I-10 | Scaffold, B13 | 9-Cyclopentyl-2-...)
Affinity DataIC50: 145nMpH: 7.5 T: 2°CAssay Description:ATP-site competition binding assay using Mps1 Kinase inhibitors in LanthaScreen Eu time-resolved FRET (TR-FRET) technology from Invitrogen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2011
Entry Details Article
PubMed
TargetDual specificity protein kinase TTK(Human)
Dana-Farber Cancer Institute

LigandPNGBDBM36485(1-(4-(4-(2-(Isopropylsulfonyl)phenylamino)-1H-pyrr...)
Affinity DataIC50: 367nMpH: 7.5 T: 2°CAssay Description:ATP-site competition binding assay using Mps1 Kinase inhibitors in LanthaScreen Eu time-resolved FRET (TR-FRET) technology from Invitrogen.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2011
Entry Details Article
PubMed