Compile Data Set for Download or QSAR
Report error Found 376 Enz. Inhib. hit(s) with all data for entry = 50047218
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154890BDBM50154890(CHEMBL3774425 | US10273244, Example 113 | US105841...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154896BDBM50154896(CHEMBL3774462 | US10273244, Example 51 | US1058413...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154898BDBM50154898(CHEMBL3774431 | US10273244, Example 61 | US1058413...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154878BDBM50154878(CHEMBL3774895 | US10273244, Example 114 | US105841...)
Affinity DataKi:  0.316nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154852BDBM50154852(CHEMBL3775737 | US10273244, Example 41 | US1058413...)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154852BDBM50154852(CHEMBL3775737 | US10273244, Example 41 | US1058413...)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154894BDBM50154894(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154852BDBM50154852(CHEMBL3775737 | US10273244, Example 41 | US1058413...)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154895BDBM50154895(CHEMBL3775534 | US10273244, Example 7 | US10584135...)
Affinity DataKi:  0.631nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154896BDBM50154896(CHEMBL3774462 | US10273244, Example 51 | US1058413...)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154850BDBM50154850(CHEMBL3774588 | US10273244, Example 22 | US1058413...)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154898BDBM50154898(CHEMBL3774431 | US10273244, Example 61 | US1058413...)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154896BDBM50154896(CHEMBL3774462 | US10273244, Example 51 | US1058413...)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154877BDBM50154877(CHEMBL3774621 | US10273244, Example 96 | US1058413...)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154898BDBM50154898(CHEMBL3774431 | US10273244, Example 61 | US1058413...)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154869BDBM50154869(CHEMBL3774519 | US10273244, Example 133 | US105841...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154891BDBM50154891(CHEMBL3775872 | US10273244, Example 25 | US1058413...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154843BDBM50154843(CHEMBL3775226 | US10273244, Example 17 | US1058413...)
Affinity DataKi:  1.26nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154842BDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataKi:  1.26nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154867BDBM50154867(CHEMBL3775810 | US10273244, Example 134 | US105841...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154842BDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154843BDBM50154843(CHEMBL3775226 | US10273244, Example 17 | US1058413...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154843BDBM50154843(CHEMBL3775226 | US10273244, Example 17 | US1058413...)
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by [35S]GTP-gamma-S binding assay in presence of 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154859BDBM50154859(CHEMBL3775554 | US10273244, Example 160 | US105841...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154853BDBM50154853(CHEMBL3775243 | US10273244, Example 81 | US1058413...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154853BDBM50154853(CHEMBL3775243 | US10273244, Example 81 | US1058413...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154851BDBM50154851(CHEMBL3774683 | US10273244, Example 89 | US1058413...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154842BDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by [35S]GTP-gamma-S binding assay in presence of 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154902BDBM50154902(CHEMBL3774540 | US10273244, Example 2 | US10584135...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154851BDBM50154851(CHEMBL3774683 | US10273244, Example 89 | US1058413...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154860BDBM50154860(CHEMBL3774490 | US10273244, Example 153 | US105841...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154875BDBM50154875(CHEMBL3775667 | US10273244, Example 94 | US1058413...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154888BDBM50154888(CHEMBL3774996 | US10273244, Example 95 | US1058413...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154863BDBM50154863(CHEMBL3775256 | US10273244, Example 162 | US105841...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154870BDBM50154870(CHEMBL3775771 | US10273244, Example 99 | US1058413...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154862BDBM50154862(CHEMBL3775482 | US10273244, Example 163 | US105841...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154892BDBM50154892(CHEMBL3775967 | US10273244, Example 27 | US1058413...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154889BDBM50154889(CHEMBL3774783 | US10273244, Example 120 | US105841...)
Affinity DataKi:  2.51nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154902BDBM50154902(CHEMBL3774540 | US10273244, Example 2 | US10584135...)
Affinity DataKi:  3.16nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154853BDBM50154853(CHEMBL3775243 | US10273244, Example 81 | US1058413...)
Affinity DataKi:  3.16nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154902BDBM50154902(CHEMBL3774540 | US10273244, Example 2 | US10584135...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154873BDBM50154873(CHEMBL3775753 | US10273244, Example 125 | US105841...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154900BDBM50154900(CHEMBL3775005 | US10273244, Example 30 | US1058413...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154861BDBM50154861(CHEMBL3775604 | US10273244, Example 141 | US105841...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154864BDBM50154864(CHEMBL3775036 | US10273244, Example 152 | US105841...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154847BDBM50154847(CHEMBL3775350 | US10273244, Example 208 | US105841...)
Affinity DataKi:  3.98nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154844BDBM50154844(CHEMBL3775197 | US10273244, Example 147 | US105841...)
Affinity DataKi:  3.98nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154851BDBM50154851(CHEMBL3774683 | US10273244, Example 89 | US1058413...)
Affinity DataKi:  3.98nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154848BDBM50154848(CHEMBL3774591 | US10273244, Example 102 | US105841...)
Affinity DataKi:  3.98nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Aptuit

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154848BDBM50154848(CHEMBL3774591 | US10273244, Example 102 | US105841...)
Affinity DataKi:  3.98nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2017
Entry Details Article
PubMed
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